Structure | Compound Name | Standard Type | Standard Values (in nM) |
|---|---|---|---|
| Ethyl 8-chloro-5,6-dihydro-5-methyl-6-oxo-4H-imidazo(1,5-a)(1,4)benzodiazepine-3-carboxylate | Ki | 0.85 [1], 54.6 [2] | |
| 8-Methyl-5-[4-(trifluoromethyl)-1-benzothiophen-2-yl]-1,9-dihydro-[1,3]oxazolo[4,5-h][2,3]benzodiazepin-2-one | IC50 | 201.0 [1], 500.0 [2] | |
| Saripidem | IC50 | 2.7 [1], 4.6 [2] | |
| Zolpidem | Ki | 15000.0 [1] | |
| Ethyl-8-azido-5,6-dihydro-5-methyl-6-oxo-4H-imidazo-1,4-benzodiazepine-3-carboxylate | Ki | 3.1 [1] | |
MLA | "Quest Database™ GABA receptor alpha-5 subunit Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 13 Dec. 2025, https://www.aatbio.com/data-sets/gaba-receptor-alpha-5-subunit-inhibitors-ic50-ki. | |
APA | AAT Bioquest, Inc. (2025, December 13). Quest Database™ GABA receptor alpha-5 subunit Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/gaba-receptor-alpha-5-subunit-inhibitors-ic50-ki. | |
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