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GABA receptor rho-1 subunit Inhibitors (IC50, Ki)

Structure
Compound Name
Standard Type
Standard Values (in nM)
(3-Aminopropyl)(n-butyl)phosphinic acidIC5062000.0 [1]
TpmpaIC502220.0 [1]
Butyl-[(4S)-4-[6-[(4-nitro-2,1,3-benzoxadiazol-7-yl)amino]hexanoylamino]cyclopenten-1-yl]phosphinic acidIC50193270.0 [1], 281420.0 [2]
Butyl-[(4S)-4-[6-[3-(2,2-difluoro-4,6,10,12-tetramethyl-3-aza-1-azonia-2-boranuidatricyclo[7.3.0.03,7]dodeca-1(12),4,6,8,10-pentaen-8-yl)propanoylamino]hexanoylamino]cyclopenten-1-yl]phosphinic acidIC5058610.0 [1], 103140.0 [2]
[(4S)-4-[6-[5-[(3As,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanoylamino]hexanoylamino]cyclopenten-1-yl]-butylphosphinic acidIC5076540.0 [1], 147920.0 [2]
Aminolevulinic acidIC5012900.0 [1]
LindaneIC5091.0 [1]
FipronilIC5010000.0 [1]
[(2R)-3-Amino-2-hydroxypropyl]-methylphosphinic acidIC505400.0 [1]
(+)-cis-2-Aminomethylcyclopropane carboxylic acidIC50800000.0 [1]
[(4S)-4-Aminocyclopenten-1-yl]-butylphosphinic acidIC509760.0 [1]
Phosphinic acid, P-[(2S)-3-amino-2-hydroxypropyl]-P-methyl-IC5017100.0 [1]
[(E)-3-Aminoprop-1-enyl]-methylphosphinic acidIC505500.0 [1]
4-Aminocyclopent-1-enecarboxylic acidIC506600.0 [1]
Endosulfan IIIC50800.0 [1]
cis-2-Aminocyclopropanecarboxylic acidIC50890000.0 [1]
(1-Hydroxy-1-oxo-1lambda5-phospholan-3-yl)methanamineIC5019910.0 [1]
4-Amino-N-hydroxycyclopentene-1-carboxamideIC5012900.0 [1]
4-Amino-N-methoxycyclopentene-1-carboxamideIC5081500.0 [1]
4-Amino-N-ethoxycyclopentene-1-carboxamideIC50153000.0 [1]
4-Amino-N-prop-2-enoxycyclopentene-1-carboxamideIC50115300.0 [1]
4-Amino-1-cyclopentene-1-carboxamideIC509600.0 [1]
4-Amino-N-methylcyclopentene-1-carboxamideIC50408300.0 [1]
4-Amino-N-propylcyclopentene-1-carboxamideIC50570000.0 [1]
(R)-2-Methyl-4-aminobutyric acidIC5016000.0 [1]



References

This online tool may be cited as follows

MLA

"Quest Database™ GABA receptor rho-1 subunit Inhibitors (IC50, Ki)." AAT Bioquest, Inc.9 May2024https://www.aatbio.com/data-sets/gaba-receptor-rho-1-subunit-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024May 9). Quest Database™ GABA receptor rho-1 subunit Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/gaba-receptor-rho-1-subunit-inhibitors-ic50-ki.
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