 | CID 11560787 | IC50 | 83.0 [1] |
 | Semagacestat | IC50 | 39.81 [1] |
 | Begacestat | IC50 | 11.0 [1] |
 | Avagacestat | IC50 | 0.27 [1] |
 | (4S,4As,10bS)-7,10-difluoro-4-(2-methylsulfonylethyl)-10b-[4-(trifluoromethyl)phenyl]sulfonyl-2,4,4a,5-tetrahydro-1H-pyrano[3,4-c]chromene | IC50 | 11.0 [1] |
 | CID 25164607 | IC50 | 1.3 [1] |
 | (4S,9E)-9-[[3-Methoxy-4-(4-methylimidazol-1-yl)phenyl]methylidene]-4-(3,4,5-trifluorophenyl)-4,6,7,8-tetrahydro-3H-pyrido[2,1-c][1,2,4]oxadiazine | IC50 | 33.0 [1], 123.0 [2] |
 | [(3S,8E)-3-(4-Fluorophenyl)-8-[[3-methoxy-4-(4-methylimidazol-1-yl)phenyl]methylidene]-6,7-dihydro-5H-[1,2,4]oxadiazolo[4,3-a]pyridin-3-yl]methanol | IC50 | 29.0 [1], 170.0 [2] |
 | 4-[[(4S,4As,10bS)-7,10-difluoro-4-(2-methylsulfonylethyl)-2,4,4a,5-tetrahydro-1H-pyrano[3,4-c]chromen-10b-yl]sulfonyl]benzonitrile | IC50 | 25.0 [1] |
 | Sulindac sulfide | IC50 | 53000.0 [1], 57100.0 [2], 82500.0 [3], 215000.0 [4], 332000.0 [5] |
 | l-685,458 | IC50 | 4.3 [1], 22.0 [2], 36.0 [3], 72.0 [4], 281.0 [5] |
 | Wpe-III-31C | IC50 | 10.0 [1], 220.0 [2], 400.0 [3], 18000.0 [4] |
 | 2-[6-Chloro-9-[2,4,6-tri(propan-2-yl)phenyl]sulfonylcarbazol-2-yl]propanoic acid | IC50 | 8500.0 [1], 9300.0 [2], 20000.0 [3] |
 | 2-[9-[2,4,6-Tri(propan-2-yl)phenyl]sulfonylcarbazol-2-yl]oxyacetic acid | IC50 | 7500.0 [1], 7800.0 [2], 19000.0 [3] |
 | Methyl (2S)-2-[[(2S)-2-[[benzyl-[(2R,3S)-2-hydroxy-3-[(2-methylpropan-2-yl)oxycarbonylamino]-4-phenylbutyl]carbamoyl]amino]-4-methylpentanoyl]amino]-4-methylpentanoate | IC50 | 30.0 [1], 600.0 [2], 650.0 [3], 9400.0 [4] |
 | [(9-Octyl-9H-carbazol-2-yl)oxy]acetic acid | IC50 | 19000.0 [1], 24000.0 [2], 40000.0 [3] |
 | (4R,6S)-5-(4-Chlorophenyl)sulfonyl-4,6-diethyl-1,4,6,7-tetrahydropyrazolo[4,3-c]pyridine | IC50 | 0.35 [1], 0.37 [2], 4.7 [3], 5.8 [4], 70.0 [5] |
 | 4-[[(4-Chlorophenyl)sulfonyl-pentan-3-ylamino]methyl]benzoic acid | IC50 | 120.0 [1], 130.0 [2], 10000.0 [3] |
 | (1S,2S)-2-[[(1S,2S)-2-[[(1S,2S)-2-[[(1S,2S)-2-[[(1S,2S)-2-[[(1S,2S)-2-[[(1S,2S)-2-[[(1S,2S)-2-[[(1S,2S)-2-[[(1S,2S)-2-[[(1S,2S)-2-[[(1S,2S)-2-Acetamidocyclopentanecarbonyl]amino]cyclopentanecarbonyl]amino]cyclopentanecarbonyl]amino]cyclopentanecarbonyl]amino]cyclopentanecarbonyl]amino]cyclopentanecarbonyl]amino]cyclopentanecarbonyl]amino]cyclopentanecarbonyl]amino]cyclopentanecarbonyl]amino]cyclopentanecarbonyl]amino]cyclopentanecarbonyl]amino]cyclopentane-1-carboxamide | IC50 | 8.81 [1], 9.93 [2], 20.4 [3], 626.0 [4], 1180.0 [5] |
 | (3S)-3-[[(1S,2S)-2-[[(1S,2S)-2-Acetamidocyclopentanecarbonyl]amino]cyclopentanecarbonyl]amino]-N'-[(1S,2S)-2-[[(1S,2S)-2-[[(1S,2S)-2-[[(1S,2S)-2-[[(1S,2S)-2-[[(1S,2S)-2-[[(1S,2S)-2-[[(1S,2S)-2-[[(1S,2S)-2-carbamoylcyclopentyl]carbamoyl]cyclopentyl]carbamoyl]cyclopentyl]carbamoyl]cyclopentyl]carbamoyl]cyclopentyl]carbamoyl]cyclopentyl]carbamoyl]cyclopentyl]carbamoyl]cyclopentyl]carbamoyl]cyclopentyl]pentanediamide | IC50 | 0.56 [1], 0.88 [2], 3.16 [3], 68.4 [4], 84.6 [5] |
 | (1S,2S)-2-[[(1S,2S)-2-[[(1S,2S)-2-[[(1S,2S)-2-[[(1S,2S)-2-[[(1S,2S)-2-[[(1S,2S)-2-[[(1S,2S)-2-[[(1S,2S)-2-[[(3S)-3-[[(1S,2S)-2-[[(1S,2S)-2-Acetamidocyclopentanecarbonyl]amino]cyclopentanecarbonyl]amino]-4-hydroxybutanoyl]amino]cyclopentanecarbonyl]amino]cyclopentanecarbonyl]amino]cyclopentanecarbonyl]amino]cyclopentanecarbonyl]amino]cyclopentanecarbonyl]amino]cyclopentanecarbonyl]amino]cyclopentanecarbonyl]amino]cyclopentanecarbonyl]amino]cyclopentane-1-carboxamide | IC50 | 0.4 [1], 0.83 [2], 41.3 [3], 84.2 [4], 86.4 [5] |
 | Nirogacestat | IC50 | 1.2 [1], 1.3 [2], 6.2 [3], 19.15 [4] |
 | N-[4-(4-Chlorophenyl)sulfonyl-4-(2,5-difluorophenyl)cyclohexyl]-1,1,1-trifluoromethanesulfonamide | IC50 | 0.65 [1], 5.0 [2], 14.3 [3], 15.0 [4] |
 | 4-[2-[(1R)-1-(N-(4-Chlorophenyl)sulfonyl-2,5-difluoroanilino)ethyl]-5-fluorophenyl]butanoic acid | IC50 | 7.1 [1], 12.0 [2], 25600.0 [3] |
 | Unii-7F5qgv49GL | IC50 | 0.34 [1], 5.3 [2], 6.6 [3] |
 | [(2R)-2-[5-Chloro-N-(4-chlorophenyl)sulfonyl-2-(hydroxymethyl)anilino]propyl] N-propylcarbamate | IC50 | 10.0 [1], 47.0 [2], 57.0 [3], 100.0 [4] |
 | 5-Chloro-N-[(2R)-4,4,4-trifluoro-1-hydroxy-3-(trifluoromethyl)butan-2-yl]thiophene-2-sulfonamide | IC50 | 8.0 [1], 15.0 [2], 10000.0 [3], 30000.0 [4] |
 | 2-(1-(4-Chlorophenylsulfonyl)cyclohexyl)-1,4-difluorobenzene | IC50 | 3.0 [1], 14.1 [2], 27.0 [3], 41.0 [4] |
 | (8E)-3-(4-Fluorophenyl)-8-[[3-methoxy-4-(4-methylimidazol-1-yl)phenyl]methylidene]-3-methyl-6,7-dihydro-5H-[1,2,4]oxadiazolo[4,3-a]pyridine | IC50 | 58.0 [1], 267.0 [2], 13702.0 [3] |
 | N-[(1S)-1-(4-Fluorophenyl)ethyl]-6-[3-methoxy-4-(4-methylimidazol-1-yl)phenyl]-4-methylpyridazin-3-amine | IC50 | 63.1 [1], 199.53 [2] |
 | N-[(1S)-1-(4-Fluorophenyl)ethyl]-6-[3-methoxy-4-(4-methylimidazol-1-yl)phenyl]pyridazin-3-amine | IC50 | 63.1 [1], 199.53 [2] |
 | [(9-Decyl-9H-carbazol-2-yl)oxy]acetic acid | IC50 | 11000.0 [1], 40000.0 [2] |
 | 2-[3,4-Bis[4-(trifluoromethyl)phenyl]phenyl]acetic acid | IC50 | 1995.26 [1], 19952.62 [2], 100000.0 [3] |
 | (2R)-2-[3-Phenylmethoxy-5-[4-(trifluoromethyl)phenyl]phenyl]pentanoic acid | IC50 | 4.8 [1], 3980.0 [2], 100000.0 [3] |
 | Methyl (2R)-2-[[(2R)-2-[[benzyl-[(2R,3R)-2-hydroxy-3-[(2-methylpropan-2-yl)oxycarbonylamino]-4-phenylbutyl]carbamoyl]amino]-4-methylpentanoyl]amino]-4-methylpentanoate | IC50 | 200.0 [1], 3000.0 [2], 9000.0 [3] |
 | Methyl (2R)-2-[[(2R)-2-[[benzyl-[(2R,3R)-2-hydroxy-3-[(2-methylpropan-2-yl)oxycarbonylamino]-4-phenylbutyl]carbamoyl]amino]-4-methylpentanoyl]amino]-3-methylbutanoate | IC50 | 100.0 [1], 2000.0 [2], 17000.0 [3] |
 | 2-[(2S,4R)-1-[(1R)-4-Methyl-1-[6-(trifluoromethyl)pyridin-3-yl]pentyl]-2-[4-(trifluoromethyl)phenyl]piperidin-4-yl]acetic acid | IC50 | 316.23 [1], 6309.57 [2], 39810.72 [3], 100000.0 [4] |
 | 2-[(2S,4R)-1-[(1R)-2-Methyl-1-[6-(trifluoromethyl)pyridin-3-yl]propyl]-2-[4-(trifluoromethyl)phenyl]piperidin-4-yl]acetic acid | IC50 | 3981.07 [1], 19952.62 [2], 100000.0 [3] |
 | 2-[(2S,4R)-1-[(R)-Cyclopropyl-[6-(trifluoromethyl)pyridin-3-yl]methyl]-2-[4-(trifluoromethyl)phenyl]piperidin-4-yl]acetic acid | IC50 | 7943.28 [1], 50118.72 [2], 100000.0 [3] |
 | 2-[(2S,4R)-2-[4-(Trifluoromethyl)phenyl]-1-[(1R)-1-[6-(trifluoromethyl)pyridin-3-yl]pentyl]piperidin-4-yl]acetic acid | IC50 | 630.96 [1], 15848.93 [2], 39810.72 [3], 100000.0 [4] |
 | 2-[(2S,4R)-2-[4-(Trifluoromethyl)phenyl]-1-[(1R)-1-[6-(trifluoromethyl)pyridin-3-yl]heptyl]piperidin-4-yl]acetic acid | IC50 | 501.19 [1], 15848.93 [2], 25118.86 [3], 100000.0 [4] |
 | [(1S)-2-Hydroxy-1-[(1S,4S,6R,8S,11R,12S,13R,16R,18S,21R)-11-hydroxy-4,6,12,17,17-pentamethyl-18-[(2S,3R,4S,5R)-3,4,5-trihydroxyoxan-2-yl]oxy-9-oxahexacyclo[11.9.0.01,21.04,12.05,10.016,21]docos-5(10)-en-8-yl]-2-methylpropyl] acetate | IC50 | 100.0 [1], 2700.0 [2], 6300.0 [3] |
 | LY-411575 | IC50 | 1.0 [1], 1200.0 [2] |
 | (2S)-2-[[(2S)-2-(3,5-Difluorophenyl)-2-hydroxyacetyl]amino]-N-[(5S)-3-methyl-4-oxo-5H-2,3-benzodiazepin-5-yl]propanamide | IC50 | 0.3 [1], 1.2 [2], 510.0 [3] |
 | Unii-19KW9LD704 | IC50 | 24000.0 [1], 100000.0 [2] |
 | 12-(4-Chlorophenyl)sulfonyl-4,5,12-triazatricyclo[6.3.1.02,6]dodeca-2(6),3-diene | IC50 | 2.0 [1], 879.0 [2] |
 | (2S,3R)-N'-[(3S)-1-Methyl-2-oxo-5-phenyl-3H-1,4-benzodiazepin-3-yl]-3-(2-methylpropyl)-2-propylbutanediamide | IC50 | 6.4 [1], 1060.0 [2] |
| (2S,3R)-N'-[(3S)-1-Methyl-2-oxo-5-phenyl-3H-1,4-benzodiazepin-3-yl]-3-(2-methylpropyl)-2-propylbutanediamide | Ki | 2.6 [1] |
 | (2S)-N-[(2S)-1-[Butyl(methyl)amino]-3-cyclohexyl-1-oxopropan-2-yl]-2-[[(2S)-2-hydroxy-2-phenylacetyl]amino]-4-methylpentanamide | IC50 | 1.0 [1] |
 | (R)-2-(4-Methoxy-3-(4-(trifluoromethyl)benzylcarbamoyl)benzyl)butanoic acid | IC50 | 34200.0 [1], 37800.0 [2], 100000.0 [3] |
 | 2-(6-Chloro-9-octylcarbazol-2-yl)propanoic acid | IC50 | 6900.0 [1], 40000.0 [2], 100000.0 [3] |
 | 5-(4-Chlorophenyl)sulfonyl-1,4-dihydropyrazolo[4,3-c]quinoline | IC50 | 27.0 [1], 250.0 [2], 327.0 [3] |
 | 4-Chloro-N-[(4-methoxyphenyl)methyl]-N-[(3R)-2-oxoazepan-3-yl]benzenesulfonamide | IC50 | 2.4 [1], 2.8 [2], 4.1 [3] |
 | (4S,4As,10bS)-10b-(4-chlorophenyl)sulfonyl-4-(2-ethylsulfonylethyl)-7,10-difluoro-2,4,4a,5-tetrahydro-1H-pyrano[3,4-c]chromene | IC50 | 2.0 [1], 3.0 [2], 5.0 [3] |
 | (4S,4As,10bS)-10b-(4-chlorophenyl)sulfonyl-7,10-difluoro-4-(2-propan-2-ylsulfonylethyl)-2,4,4a,5-tetrahydro-1H-pyrano[3,4-c]chromene | IC50 | 3.0 [1], 5.5 [2], 8.0 [3] |
 | 2-[2-[(4S,4As,10bS)-10b-(4-chlorophenyl)sulfonyl-7,10-difluoro-2,4,4a,5-tetrahydro-1H-pyrano[3,4-c]chromen-4-yl]ethylsulfonyl]ethanol | IC50 | 0.9 [1], 1.0 [2], 1.2 [3] |
 | [1-(4-Chlorophenyl)sulfonyl-6-(3-fluorophenyl)piperidin-2-yl]methyl 4-piperidin-1-ylpiperidine-1-carboxylate | IC50 | 3.0 [1], 7.7 [2], 11.2 [3] |
 | (4R)-5-(4-Chlorophenyl)sulfonyl-8-fluoro-4-methyl-1,4-dihydropyrazolo[4,3-c]quinoline | IC50 | 0.62 [1], 14.0 [2] |
 | N-[[(6Ar,7R,10aS)-1,4-difluoro-10a-[4-(trifluoromethyl)phenyl]sulfonyl-6,6a,7,8,9,10-hexahydrobenzo[c]chromen-7-yl]methyl]-1,1,1-trifluoromethanesulfonamide | IC50 | 32.0 [1], 54.0 [2], 73.0 [3] |
 | (1R,2S,4R,7R,10S)-4-Ethyl-12,15-difluoro-10-[4-(trifluoromethyl)phenyl]sulfonyl-17-oxa-5lambda6-thia-6-azatetracyclo[8.8.0.02,7.011,16]octadeca-11,13,15-triene 5,5-dioxide | IC50 | 1.9 [1], 2.0 [2], 5.0 [3] |
 | 10-Phenyl-12-[4-(trifluoromethyl)phenyl]sulfonyl-4,5,12-triazatricyclo[6.3.1.02,6]dodeca-2(6),3-diene | IC50 | 14.0 [1], 10932.0 [2] |
 | 2-[2-[(4S,4As,10bS)-10b-(4-chlorophenyl)sulfonyl-7,10-difluoro-2,4,4a,5-tetrahydro-1H-pyrano[3,4-c]chromen-4-yl]ethylsulfonyl]acetic acid | IC50 | 2.7 [1], 22.0 [2], 38.0 [3] |
 | Acetic acid, (9H-carbazol-2-yloxy)- | IC50 | 40000.0 [1] |
 | (3S)-6-Fluoro-3-[4-[2-methoxy-4-(4-methylimidazol-1-yl)phenyl]triazol-1-yl]-1-(2,2,2-trifluoroethyl)-4,5-dihydro-3H-1-benzazepin-2-one | IC50 | 11.0 [1], 73.0 [2], 30000.0 [3] |
 | (3S)-6-Fluoro-3-[4-[2-fluoro-4-(4-methylimidazol-1-yl)phenyl]triazol-1-yl]-1-(2,2,2-trifluoroethyl)-4,5-dihydro-3H-1-benzazepin-2-one | IC50 | 58.0 [1], 460.0 [2], 45000.0 [3] |
 | (3S)-6-Fluoro-3-[4-[3-fluoro-2-methoxy-4-(4-methylimidazol-1-yl)phenyl]triazol-1-yl]-1-(2,2,2-trifluoroethyl)-4,5-dihydro-3H-1-benzazepin-2-one | IC50 | 13.0 [1], 100.0 [2], 50000.0 [3] |
 | N-(2,5-Difluorophenyl)-4-fluoro-N-[[2-(oxan-4-yloxy)phenyl]methyl]benzenesulfonamide | IC50 | 360.0 [1], 400.0 [2], 620.0 [3] |
 | Tert-butyl N-[(2S,3R,5R)-5-benzyl-6-[[(2S)-1-[[(3R)-5-cyclohexyl-2-oxo-1,3-dihydro-1,4-benzodiazepin-3-yl]amino]-1-oxopropan-2-yl]amino]-3-hydroxy-6-oxo-1-phenylhexan-2-yl]carbamate | IC50 | 0.56 [1], 0.7 [2], 28.0 [3] |
 | N-[(2S,3R,5R)-5-Benzyl-6-[[(2S)-1-[[(3R)-5-cyclohexyl-2-oxo-1,3-dihydro-1,4-benzodiazepin-3-yl]amino]-1-oxopropan-2-yl]amino]-3-hydroxy-6-oxo-1-phenylhexan-2-yl]-4-(4-prop-2-ynoxybenzoyl)benzamide | IC50 | 0.91 [1], 1.0 [2], 20.0 [3] |
 | 5-(4-Chloro-benzenesulfonyl)-6-phenyl-4,5,6,7-tetrahydro-2H-pyrazolo[4,3-c]pyridine | IC50 | 7.7 [1], 598.0 [2], 6514.0 [3] |
 | 6-Benzyl-5-(4-chlorophenylsulfonyl)-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridine | IC50 | 80.9 [1], 1554.0 [2], 16625.0 [3] |
 | 5-(4-Chlorophenylsulfonyl)-6-isopropyl-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridine | IC50 | 16.1 [1], 87.0 [2], 6759.0 [3] |
 | 5-(4-Chlorophenylsulfonyl)-6-(4-fluorophenyl)-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridine | IC50 | 5.4 [1], 481.0 [2], 5319.0 [3] |
 | 6-(4-Chlorophenyl)-5-(4-chlorophenylsulfonyl)-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridine | IC50 | 3.4 [1], 311.0 [2], 2586.0 [3] |
 | 5-(4-Chlorophenylsulfonyl)-6-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridine | IC50 | 9.7 [1], 776.0 [2], 14126.0 [3] |
 | 5-(4-Chlorophenyl)sulfonyl-6-pyrimidin-5-yl-1,4,6,7-tetrahydropyrazolo[4,3-c]pyridine | IC50 | 536.0 [1], 10375.0 [2], 40000.0 [3] |
 | 5-(4-Chlorophenyl)sulfonyl-4-pyrimidin-5-yl-1,4,6,7-tetrahydropyrazolo[4,3-c]pyridine | IC50 | 12.0 [1], 120.0 [2], 2305.0 [3] |
 | Ethyl 5-(4-chlorophenyl)sulfonyl-1,4,6,7-tetrahydropyrazolo[4,3-c]pyridine-4-carboxylate | IC50 | 10.2 [1], 204.0 [2], 10263.0 [3] |
 | Ethyl 5-(4-chlorophenyl)sulfonyl-1,4,6,7-tetrahydropyrazolo[4,3-c]pyridine-6-carboxylate | IC50 | 431.0 [1], 5851.0 [2], 40000.0 [3] |
 | 2-[5-(4-Chlorophenyl)sulfonyl-1,4,6,7-tetrahydropyrazolo[4,3-c]pyridin-6-yl]-1,3-thiazole | IC50 | 244.0 [1], 5750.0 [2], 33565.0 [3] |
 | 2-[5-(4-Chlorophenyl)sulfonyl-1,4,6,7-tetrahydropyrazolo[4,3-c]pyridin-4-yl]-1,3-thiazole | IC50 | 29.1 [1], 858.0 [2], 6527.0 [3] |
 | [5-(4-Chlorophenyl)sulfonyl-1,4,6,7-tetrahydropyrazolo[4,3-c]pyridin-4-yl]methyl N,N-dimethylcarbamate | IC50 | 350.0 [1], 8251.0 [2], 40000.0 [3] |
 | (4S,4As,10bS)-10b-(4-chlorophenyl)sulfonyl-7,10-difluoro-4-[2-(trifluoromethylsulfonyl)ethyl]-2,4,4a,5-tetrahydro-1H-pyrano[3,4-c]chromene | IC50 | 4.4 [1], 7.4 [2], 13.0 [3] |
 | (4S,4As,10bS)-10b-(4-chlorophenyl)sulfonyl-7,10-difluoro-4-[2-(2,2,2-trifluoroethylsulfonyl)ethyl]-2,4,4a,5-tetrahydro-1H-pyrano[3,4-c]chromene | IC50 | 6.4 [1], 7.3 [2], 22.0 [3] |
 | (4S,4As,10bS)-10b-(4-chlorophenyl)sulfonyl-7,10-difluoro-4-(2-propylsulfonylethyl)-2,4,4a,5-tetrahydro-1H-pyrano[3,4-c]chromene | IC50 | 5.0 [1], 6.8 [2], 11.0 [3] |
 | (4S,4As,10bS)-10b-(4-bromophenyl)sulfonyl-7,10-difluoro-4-(2-methylsulfonylethyl)-2,4,4a,5-tetrahydro-1H-pyrano[3,4-c]chromene | IC50 | 0.6 [1], 2.5 [2], 2.9 [3] |
 | (4S,4As,10bS)-10b-(3,4-difluorophenyl)sulfonyl-7,10-difluoro-4-(2-methylsulfonylethyl)-2,4,4a,5-tetrahydro-1H-pyrano[3,4-c]chromene | IC50 | 1.4 [1], 14.0 [2], 31.0 [3] |
 | (6Ar,7S,10aS)-1,4-difluoro-7-(2-methylsulfonylethyl)-10a-[4-(trifluoromethyl)phenyl]sulfonyl-6,6a,7,8,9,10-hexahydrobenzo[c]chromene | IC50 | 21.0 [1], 43.0 [2], 63.0 [3] |
 | 4-[[(1R,2S,4R,7R,10S)-4-Ethyl-12,15-difluoro-5,5-dioxo-17-oxa-5lambda6-thia-6-azatetracyclo[8.8.0.02,7.011,16]octadeca-11,13,15-trien-10-yl]sulfonyl]benzonitrile | IC50 | 2.0 [1], 4.0 [2], 4.7 [3] |
 | (2R)-2-[3,5-Bis(trifluoromethyl)phenyl]-N-[4-(2-methylpyridin-4-yl)phenyl]propanamide | IC50 | 260.0 [1], 3100.0 [2], 11800.0 [3] |
 | 1-N'-[(1S)-1-Hydroxy-3-methylbutyl]-1-N-[(3S)-1-methyl-2-oxo-5-[4-(trifluoromethyl)phenyl]-3H-1,4-benzodiazepin-3-yl]cyclobutane-1,1-dicarboxamide | IC50 | 6.1 [1] |
| 1-N'-[(1S)-1-Hydroxy-3-methylbutyl]-1-N-[(3S)-1-methyl-2-oxo-5-[4-(trifluoromethyl)phenyl]-3H-1,4-benzodiazepin-3-yl]cyclobutane-1,1-dicarboxamide | Ki | 2.1 [1] |
 | {[9-(4-Methylbenzene-1-sulfonyl)-9H-carbazol-2-yl]oxy}acetic acid | IC50 | 13000.0 [1], 39000.0 [2], 40000.0 [3] |
 | 2-[9-[3,5-Bis(trifluoromethyl)phenyl]sulfonylcarbazol-2-yl]oxyacetic acid | IC50 | 40000.0 [1] |
 | {[9-([1,1'-Biphenyl]-4-sulfonyl)-9H-carbazol-2-yl]oxy}acetic acid | IC50 | 13000.0 [1], 24000.0 [2], 40000.0 [3] |
 | {[9-(4-Chlorobenzene-1-sulfonyl)-9H-carbazol-2-yl]oxy}acetic acid | IC50 | 32000.0 [1], 40000.0 [2] |
 | {[9-(3,5-Difluorobenzene-1-sulfonyl)-9H-carbazol-2-yl]oxy}acetic acid | IC50 | 13000.0 [1], 40000.0 [2] |
 | {[9-(2-Bromobenzene-1-sulfonyl)-9H-carbazol-2-yl]oxy}acetic acid | IC50 | 40000.0 [1] |
 | {[9-(3-Nitrobenzene-1-sulfonyl)-9H-carbazol-2-yl]oxy}acetic acid | IC50 | 16000.0 [1], 40000.0 [2] |
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