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GAR transformylase Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
LometrexolIC505.77 [1], 14.0 [2], 220.0 [3], 14000.0 [4]
LometrexolKi6.0 [1], 60.0 [2], 130.0 [3]
PemetrexedIC5030.0 [1], 30000.0 [2]
PemetrexedKi380.0 [1], 1000.0 [2]
N-(4-((3-(2,4-Diamino-1,6-dihydro-6-oxo-5-pyrimidinyl)propyl)amino)benzoyl)glutamic acidIC503000.0 [1]

References
This online resource may be cited as follows
MLA
"Quest DatabaseGAR transformylase Inhibitors (IC50, Ki)." AAT Bioquest, Inc.15 Dec2025https://www.aatbio.com/data-sets/gar-transformylase-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 15). Quest DatabaseGAR transformylase Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/gar-transformylase-inhibitors-ic50-ki.
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