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Ghrelin receptor Inhibitors (IC50, Ki)

Structure
Compound Name
Standard Type
Standard Values (in nM)
KwFwLL-NH2IC5061.0 [1]
KwFwLL-NH2Ki255.0 [1]
IbutamorenIC500.4 [1]
IbutamorenKi0.24 [1]
CID 44576256IC500.14 [1]
CID 44576256Ki0.7 [1]
6-Ethyl-5-[4-[(4-methylsulfonylphenyl)methylamino]phenyl]pyrimidine-2,4-diamineIC507.0 [1], 9.7 [2], 12.0 [3], 37.0 [4]
3-(2,6-Dichlorophenyl)-N-[4-(diethylamino)phenyl]-5-methyl-1,2-oxazole-4-carboxamideIC50130.0 [1], 180.0 [2]
1-[2-[(2,2-Dimethyl-3,4-dihydrochromen-6-yl)methyl]-2,7-diazaspiro[3.5]nonan-7-yl]-2-(4-methoxyphenoxy)ethanoneIC50211.0 [1], 213.8 [2]
1-[2-[(2,2-Dimethyl-3,4-dihydrochromen-6-yl)methyl]-2,7-diazaspiro[3.5]nonan-7-yl]-2-(4-methoxyphenoxy)ethanoneKi213.8 [1], 407.38 [2], 408.0 [3]
2-Amino-N-[(1R)-2-(1H-indol-3-yl)-1-[5-[2-(1H-indol-3-yl)ethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]ethyl]-2-methylpropanamideIC506.0 [1]
N-[(1R)-2-(1H-Indol-3-yl)-1-[5-[2-(1H-indol-3-yl)ethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]ethyl]piperidine-4-carboxamideIC500.3 [1], 0.6 [2]
2-(4-Methoxyphenyl)-1-[2-[(1R)-5-pyrimidin-2-yl-2,3-dihydro-1H-inden-1-yl]-2,7-diazaspiro[3.5]nonan-7-yl]ethanoneKi6.31 [1], 6.9 [2], 17.38 [3]
5-{4-[(4-Chlorobenzyl)amino]phenyl}-6-ethylpyrimidine-2,4-diamineIC50310.0 [1], 1380.0 [2], 1400.0 [3]
6-[(Benzyloxy)methyl]-5-(4-{[4-(methylsulfonyl)benzyl]amino}phenyl)pyrimidine-2,4-diamineIC500.3 [1], 7.1 [2], 7.2 [3]
6-Benzyloxymethyl-5-[4-(4-chloro-benzylamino)-phenyl]-pyrimidine-2,4-diamineIC5019.0 [1], 180.0 [2]
3-(2,6-Dichlorophenyl)-N-[4-(diethylamino)phenyl]-5-[2-(1,3-dioxan-2-yl)ethyl]-1,2-oxazole-4-carboxamideIC506.0 [1], 14.0 [2], 19.0 [3]
N-[(1R)-1-[5-[(1R)-1-Acetamido-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]pyridine-2-carboxamideIC501.3 [1], 2.0 [2], 4.0 [3]
N-[(1R)-1-[5-[(1R)-1-Acetamido-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]pyridine-2-carboxamideKi10.0 [1]
N-[(1R)-1-[5-[(1R)-1-Formamido-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]pyridine-2-carboxamideIC503.0 [1], 3.4 [2], 8.0 [3]
N-[(1R)-1-[5-[(1R)-1-Formamido-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]pyridine-2-carboxamideKi8.0 [1]
N-[(1R)-1-[5-[(1R)-1-Acetamido-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-hydroxyacetamideIC502.0 [1], 3.0 [2], 8.0 [3]
N-[(1R)-1-[5-[(1R)-1-Acetamido-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-hydroxyacetamideKi0.8 [1]
(2S)-N-[(1R)-1-[5-[(1R)-1-Acetamido-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]morpholine-2-carboxamideIC503.0 [1], 3.4 [2], 9.0 [3]
(2S)-N-[(1R)-1-[5-[(1R)-1-Acetamido-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]morpholine-2-carboxamideKi2.0 [1]
N-[(1R)-1-[5-[(1R)-1-Acetamido-2-(1H-indol-3-yl)ethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-amino-2-methylpropanamideIC501.4 [1], 19.0 [2], 22.0 [3]
N-[(1R)-1-[5-[(1R)-1-Acetamido-2-(1H-indol-3-yl)ethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-amino-2-methylpropanamideKi12.0 [1]
2-Amino-N-[(1R)-1-[5-[(1R)-1-formamido-2-(1H-indol-3-yl)ethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-methylpropanamideIC503.2 [1], 33.0 [2], 60.0 [3]
2-Amino-N-[(1R)-1-[5-[(1R)-1-formamido-2-(1H-indol-3-yl)ethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-methylpropanamideKi46.0 [1]
N-[(1R)-1-[5-[(1R)-1-Acetamido-2-(1H-indol-3-yl)ethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]pyridine-2-carboxamideIC500.6 [1], 2.0 [2], 3.0 [3]
N-[(1R)-1-[5-[(1R)-1-Acetamido-2-(1H-indol-3-yl)ethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]pyridine-2-carboxamideKi9.0 [1]
Growth hormone releasing hexapeptideIC506.08 [1], 6000.0 [2]
Growth hormone releasing hexapeptideKi6.0 [1]
CapromorelinIC5019.95 [1], 3000.0 [2]
CapromorelinKi7.0 [1]
1-[2-[[2-Chloro-4-(triazol-2-yl)phenyl]methyl]-2,7-diazaspiro[3.5]nonan-7-yl]-2-(2-methylimidazo[2,1-b][1,3]thiazol-6-yl)ethanoneIC504.6 [1]
1-[2-[[2-Chloro-4-(triazol-2-yl)phenyl]methyl]-2,7-diazaspiro[3.5]nonan-7-yl]-2-(2-methylimidazo[2,1-b][1,3]thiazol-6-yl)ethanoneKi5.5 [1], 7.0 [2]
2-Methylpropyl N-[2-[[4-(diethylamino)phenyl]carbamoyl]-8-methoxy-3,4-dihydro-1H-naphthalen-2-yl]-N-methylcarbamateIC5016.0 [1], 29.0 [2]
Wfwll-NH2IC50530.0 [1], 1000.0 [2]
3-(2,6-Dichlorophenyl)-N-[4-(diethylamino)phenyl]-5-[2-(2-oxopiperidin-1-yl)ethyl]-1,2-oxazole-4-carboxamideIC508.0 [1], 9.0 [2]
2-(5-Methoxypyridin-2-yl)-1-[2-[(1R)-5-(6-methylpyrimidin-4-yl)-2,3-dihydro-1H-inden-1-yl]-2,7-diazaspiro[3.5]nonan-7-yl]ethanoneKi12.88 [1], 14.0 [2], 16.98 [3]
2-(5-Methoxypyridin-2-yl)-1-[2-[(1R)-5-(5-methylpyrimidin-2-yl)-2,3-dihydro-1H-inden-1-yl]-2,7-diazaspiro[3.5]nonan-7-yl]ethanoneKi9.12 [1], 85.11 [2]
2-(5-Methoxypyridin-2-yl)-1-[2-[(1R)-5-pyrimidin-2-yl-2,3-dihydro-1H-inden-1-yl]-2,7-diazaspiro[3.5]nonan-7-yl]ethanoneKi25.12 [1], 29.51 [2]
N-[(1R)-2-(1H-Indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]pyridine-3-carboxamideIC50122.0 [1], 337.0 [2], 411.0 [3]
5-Bromo-N-[(1R)-2-(1H-indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]pyridine-3-carboxamideIC5084.0 [1], 88.0 [2], 222.0 [3]
2-Bromo-N-[(1R)-2-(1H-indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]pyridine-3-carboxamideIC50193.0 [1], 250.0 [2], 510.0 [3]
6-Chloro-N-[(1R)-2-(1H-indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]pyridine-3-carboxamideIC50130.0 [1], 771.0 [2], 1010.0 [3]
2-Amino-N-[(1R)-2-(1H-indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]pyridine-3-carboxamideIC50380.0 [1], 427.0 [2], 671.0 [3]
3-Fluoro-N-[(1R)-2-(1H-indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]pyridine-2-carboxamideIC503.0 [1], 7.0 [2], 8.8 [3]
6-Fluoro-N-[(1R)-2-(1H-indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]pyridine-2-carboxamideIC502.0 [1], 2.1 [2]
3,5-Difluoro-N-[(1R)-2-(1H-indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]pyridine-2-carboxamideIC502.8 [1], 4.0 [2], 4.6 [3]
N-[(1R)-2-(1H-Indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]-6-methylpyridine-2-carboxamideIC503.4 [1], 5.4 [2], 7.5 [3]
N-[(1R)-2-(1H-Indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]-6-methoxypyridine-2-carboxamideIC502.0 [1], 7.8 [2], 9.0 [3]
6-Amino-N-[(1R)-2-(1H-indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]pyridine-2-carboxamideIC506.0 [1], 21.0 [2], 25.0 [3]
3-Hydroxy-N-[(1R)-2-(1H-indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]pyridine-2-carboxamideIC50108.0 [1], 165.0 [2], 240.0 [3]
N-[(1R)-2-(1H-Indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]-1-oxidopyridin-1-ium-2-carboxamideIC5042.0 [1], 79.0 [2], 112.0 [3]
N-[(1R)-2-(1H-Indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]-5-pyrrolidin-1-ylpyridine-2-carboxamideIC5065.0 [1], 1210.0 [2], 2115.0 [3]
3-Benzoyl-N-[(1R)-2-(1H-indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]pyridine-2-carboxamideIC50230.0 [1], 240.0 [2], 313.0 [3]
N-[(1R)-2-(1H-Indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]isoquinoline-1-carboxamideIC5073.0 [1], 82.0 [2], 150.0 [3]
N-[(1R)-2-(1H-Indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]isoquinoline-3-carboxamideIC50100.0 [1], 126.0 [2], 404.0 [3]
N-[(1R)-1-[5-[(1S)-1-Acetamido-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-amino-2-methylpropanamideIC501000.0 [1]
N-[(1R)-1-[5-[(1S)-1-Acetamido-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-amino-2-methylpropanamideKi1000.0 [1]
2-Amino-N-[(1R)-1-[5-[(1S)-1-amino-2-(1H-indol-3-yl)ethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-methylpropanamideIC501000.0 [1]
2-Amino-N-[(1R)-1-[5-[(1S)-1-amino-2-(1H-indol-3-yl)ethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-methylpropanamideKi1000.0 [1]
N-[(1R)-1-[5-[(1R)-1-Acetamido-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-3,4-dihydro-2H-pyran-6-carboxamideIC503.0 [1], 4.0 [2]
N-[(1R)-1-[5-[(1R)-1-Acetamido-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-3,4-dihydro-2H-pyran-6-carboxamideKi9.0 [1]
N-[(1R)-1-[5-[(1S)-1-Formamido-2-(1H-indol-3-yl)ethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]pyridine-2-carboxamideIC50410.0 [1], 1200.0 [2]
N-[(1R)-1-[5-[(1S)-1-Formamido-2-(1H-indol-3-yl)ethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]pyridine-2-carboxamideKi154.0 [1]
N-[(1R)-1-[5-[(1S)-1-Acetamido-2-(1H-indol-3-yl)ethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]pyridine-2-carboxamideIC50100.0 [1], 190.0 [2]
N-[(1R)-1-[5-[(1S)-1-Acetamido-2-(1H-indol-3-yl)ethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]pyridine-2-carboxamideKi62.0 [1]
2-Amino-N-[(1R)-1-[5-[(1S)-1-amino-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-methylpropanamideIC501000.0 [1]
2-Amino-N-[(1R)-1-[5-[(1S)-1-amino-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-methylpropanamideKi1000.0 [1]
N-[(1R)-1-[5-[(1R)-1-Acetamido-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-3-fluoropyridine-2-carboxamideIC502.0 [1]
N-[(1R)-1-[5-[(1R)-1-Acetamido-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-3-fluoropyridine-2-carboxamideKi4.0 [1]
N-[(1R)-1-[5-[(1R)-1-Acetamido-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-4,6-difluoropyridine-2-carboxamideIC504.0 [1]
N-[(1R)-1-[5-[(1R)-1-Acetamido-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-4,6-difluoropyridine-2-carboxamideKi11.0 [1]
2-Amino-N-[(1R)-1-[5-[(1R)-1-amino-2-(1H-indol-3-yl)ethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-methylpropanamideIC5090.0 [1], 130.0 [2]
2-Amino-N-[(1R)-1-[5-[(1R)-1-amino-2-(1H-indol-3-yl)ethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-methylpropanamideKi131.0 [1]
N-[(1R)-1-[5-[(1S)-1-Acetamido-2-(1H-indol-3-yl)ethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-amino-2-methylpropanamideIC501000.0 [1]
N-[(1R)-1-[5-[(1S)-1-Acetamido-2-(1H-indol-3-yl)ethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-amino-2-methylpropanamideKi1000.0 [1]
N-[(1R)-1-[5-[(1S)-1-Amino-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]pyridine-2-carboxamideIC50150.0 [1], 320.0 [2]
N-[(1R)-1-[5-[(1S)-1-Amino-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]pyridine-2-carboxamideKi62.0 [1]
N-[(1R)-1-[5-[(1R)-1-Amino-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]pyridine-2-carboxamideIC504.0 [1], 7.0 [2]
N-[(1R)-1-[5-[(1R)-1-Amino-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]pyridine-2-carboxamideKi18.0 [1]
2-Amino-N-[(1R)-1-[5-[(1R)-1-amino-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-methylpropanamideIC50115.0 [1], 135.0 [2]
2-Amino-N-[(1R)-1-[5-[(1R)-1-amino-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-methylpropanamideKi154.0 [1]
N-[(1R)-2-(1H-Indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]pyridine-2-carboxamideIC500.7 [1], 4.5 [2], 6.0 [3]
2-Amino-N-[(1R)-1-[5-[(1R)-1-formamido-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-methylpropanamideIC5043.0 [1], 113.0 [2]
2-Amino-N-[(1R)-1-[5-[(1R)-1-formamido-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-methylpropanamideKi59.0 [1]
N-[(1R)-1-[5-[(1S)-1-Acetamido-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]pyridine-2-carboxamideIC5070.0 [1], 360.0 [2]
N-[(1R)-1-[5-[(1S)-1-Acetamido-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]pyridine-2-carboxamideKi17.0 [1]
N-[(1R)-1-[5-[(1R)-1-Acetamido-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-amino-2-methylpropanamideIC5070.0 [1], 90.0 [2]
N-[(1R)-1-[5-[(1R)-1-Acetamido-2-phenylethyl]-4-[(4-methoxyphenyl)methyl]-1,2,4-triazol-3-yl]-2-(1H-indol-3-yl)ethyl]-2-amino-2-methylpropanamideKi46.0 [1]
(6S,9S,12R)-12-Benzyl-6-[(2S)-butan-2-yl]-9-(hydroxymethyl)-8-methyl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),18,20-triene-7,10,13-trioneIC50500.0 [1]
(6S,9S,12R)-12-Benzyl-6-[(2S)-butan-2-yl]-9-(hydroxymethyl)-8-methyl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),18,20-triene-7,10,13-trioneKi100.0 [1]
ExamorelinIC5015.9 [1], 18.0 [2]
CID 121879IC502800.0 [1]
CID 121879Ki63.0 [1]
2-Amino-N-[(1R)-2-(1H-indol-3-yl)-1-[4-[(4-methoxyphenyl)methyl]-5-(2-phenylethyl)-1,2,4-triazol-3-yl]ethyl]acetamideIC5032.0 [1]



References

This online tool may be cited as follows

MLA

"Quest Database™ Ghrelin receptor Inhibitors (IC50, Ki)." AAT Bioquest, Inc.8 May2024https://www.aatbio.com/data-sets/ghrelin-receptor-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024May 8). Quest Database™ Ghrelin receptor Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/ghrelin-receptor-inhibitors-ic50-ki.
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