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Glutamate carboxypeptidase II Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
2-(Phosphonomethyl)pentanedioic acidIC500.3 [1], 1.1 [2]
2-(Phosphonomethyl)pentanedioic acidKi0.2 [1], 0.28 [2], 0.3 [3], 31.2 [4]
N-{[(1s)-1-Carboxy-5-{[(4-Iodophenyl)carbonyl]amino}pentyl]carbamoyl}-L-Glutamic AcidIC500.02 [1]
N-{[(1s)-1-Carboxy-5-{[(4-Iodophenyl)carbonyl]amino}pentyl]carbamoyl}-L-Glutamic AcidKi0.0 [1], 0.01 [2]
2-(3-Mercaptopropyl)pentanedioic acidIC5090.0 [1]
CID 11722553Ki0.58 [1], 0.75 [2], 1.08 [3]
(2S,2'S)-2,2'-Carbonylbis(Azanediyl)Dipentanedioic AcidIC5047.0 [1]
(2S,2'S)-2,2'-Carbonylbis(Azanediyl)Dipentanedioic AcidKi8.0 [1]
3-(2-Carboxy-5-mercaptopentyl)benzoic acidIC5015.0 [1]
N~2~-{[(1s)-1-Carboxy-3-(Methylsulfanyl)propyl]carbamoyl}-N~6~-(4-Iodobenzoyl)-L-LysineKi23.0 [1]
5-Sulfanylpentanoic AcidIC501400.0 [1]
N~2~-{[(1s)-1-Carboxybut-3-Yn-1-Yl]carbamoyl}-N~6~-(4-Iodobenzoyl)-L-LysineKi5.3 [1]
N~2~-{[(1s)-1-Carboxy-2-(Furan-2-Yl)ethyl]carbamoyl}-N~6~-(4-Iodobenzoyl)-L-LysineKi5.3 [1]
3-(2-Mercaptoethyl)-[1,1'-biphenyl]-2,3'-dicarboxylic acidIC502.0 [1]
3-(2-Mercaptoethyl)-[1,1'-biphenyl]-2,3'-dicarboxylic acidKi1.0 [1]
1-(3-Carboxyphenyl)-3-(2-mercapto-ethyl)-1H-indole-2-carboxylic acidIC5022.0 [1]
2-(2-Hydroxycarbamoyl-ethyl)-pentanedioic acidIC501200.0 [1]
(S)-2-(3-((S)-5-Amino-1-carboxypentyl)ureido)pentanedioic AcidIC50498.0 [1]
(S)-2-(3-((S)-5-Amino-1-carboxypentyl)ureido)pentanedioic AcidKi44.3 [1]
Tripotassium;(2S)-2-[[oxido(4-phenylbutoxy)phosphoryl]amino]pentanedioateIC50180.0 [1]
N~2~-{[(1s)-1-Carboxybut-3-En-1-Yl]carbamoyl}-N~6~-[(4-Iodophenyl)carbonyl]-L-LysineKi11.0 [1]
(S)-2-(3-(Carboxymethyl)ureido)-6-(4-iodobenzamido)hexanoic acidKi1320.0 [1], 4390.0 [2]
(S)-2-(3-((S)-1-Carboxybutyl)ureido)-6-(4-iodobenzamido)hexanoic acidKi52.3 [1], 145.0 [2]
(2S)-2-[[(1S)-1-Carboxy-2-thiophen-2-ylethyl]carbamoylamino]-6-[(4-iodobenzoyl)amino]hexanoic acidKi16.2 [1]
(2S)-2-[[(1S)-1-Carboxy-2-(1,3-thiazol-4-yl)ethyl]carbamoylamino]-6-[(4-iodobenzoyl)amino]hexanoic acidKi16.1 [1]
N-({(1s)-5-[Acetyl(4-Bromobenzyl)amino]-1-Carboxypentyl}carbamoyl)-L-Glutamic AcidKi0.04 [1]
(2S)-2-[[(1S)-5-Acetamido-1-carboxypentyl]carbamoylamino]pentanedioic acidKi0.17 [1]
4-[2-Carboxy-5-(hydroxyamino)-5-oxopentyl]benzoic acidIC5040.0 [1], 63.0 [2]
Benzyl (2S,3S)-3-[(4-hydroxyphenyl)methyl]-4-oxo-1-[2-(3-phenylmethoxycarbonylphenyl)acetyl]azetidine-2-carboxylateIC50226.0 [1], 348.0 [2]
4-[[(2S,3S)-3-[(4-Hydroxyphenyl)methyl]-4-oxo-1-[2-(3-phenylmethoxycarbonylphenyl)acetyl]azetidine-2-carbonyl]oxymethyl]benzoic acidIC503500.0 [1]
4-[[(2S,3S)-3-Benzyl-4-oxo-1-[2-(3-phenylmethoxycarbonylphenyl)acetyl]azetidine-2-carbonyl]oxymethyl]benzoic acidIC508980.0 [1]
3-Benzyl-1-[2-(3-carboxy-phenyl)-acetyl]-4-oxo-azetidine-2-carboxylic acid 4-carboxy-benzyl esterIC5030000.0 [1]
4-[[(2S,3S)-3-Benzyl-1-[2-[3-[(4-carboxyphenyl)methoxycarbonyl]phenyl]acetyl]-4-oxoazetidine-2-carbonyl]oxymethyl]benzoic acidIC505840.0 [1]
3-Benzyl-1-[2-(3-benzyloxycarbonyl-phenyl)-acetyl]-4-oxo-azetidine-2-carboxylic acid benzyl esterIC501430.0 [1]
(S)-2-(3-((S)-1-Carboxy-5-(4-fluorobenzamido)pentyl)ureido)pentanedioic acidKi0.19 [1], 0.26 [2]
(2S)-2-[[(1S)-1-Carboxy-5-[(5-iodopyridine-3-carbonyl)amino]pentyl]carbamoylamino]pentanedioic acidKi0.35 [1], 0.56 [2]
Glutamic acidIC50428000.0 [1]
PhosphoserineIC50523000.0 [1]
Quisqualic acidIC509500.0 [1]
WillardiineIC5067000.0 [1]
L-Serine O-sulfateIC50438000.0 [1]
Glutamine hydroxamateIC50100000.0 [1]
(2S)-2-(Phosphonoamino)pentanedioic AcidIC502.3 [1]
2-Benzyl-3-mercaptopropanoic acidKi11.0 [1]
L-Glutamic acid, N-((((1S)-1-carboxy-5-((((4-iodophenyl)amino)carbonyl)amino)pentyl)amino)carbonyl)-IC5010.0 [1]
1,2,4-Butanetricarboxylic acidIC5020000.0 [1]
4-(Hydroxyamino)-4-oxobutanoic acidIC5043000.0 [1]
2-({Hydroxy[(2,3,4,5,6-pentafluorophenyl)methyl]phosphoryl}methyl)pentanedioic acidIC5082.0 [1]
IofolastatIC5022.0 [1]
Pentanedioic acid, 2-mercapto-IC502600.0 [1]
2-(Phosphonomethyl)Succinic AcidKi700.0 [1]
(R)-2-(Phosphonomethyl)Pentanedioic AcidKi30.0 [1]
n-Hydroxy-d-asparagineIC50100000.0 [1]
2-[3-(1-Carboxy-2-mercapto-ethyl)-ureido]-pentanedioic acidKi376.0 [1]
N-Hydroxy-L-asparagineIC50100000.0 [1]
2-Hydroxycarbamoylmethyl-pentanedioic acidIC50220.0 [1]
2-Phosphonomethyl-hexanedioic acidIC50185.0 [1]
(2s)-2-(Phosphonomethyl)pentanedioic AcidKi0.1 [1]
3-(Mercaptomethyl)benzoic acidIC501300.0 [1]
(2S,4S)-2-[[(1S,3S)-1,3-Dicarboxybutyl]carbamoylamino]-4-methylpentanedioic acidKi1109.0 [1]
(2S,4R)-2-[[(1S,3R)-1,3-Dicarboxybutyl]carbamoylamino]-4-methylpentanedioic acidKi1285.0 [1]
Benzoic acid, 3-[(1-carboxy-4-mercaptobutyl)thio]-IC5032.0 [1]
2-Mercaptomethylglutaric acidIC506000.0 [1]
N~2~-[(1-Carboxycyclopropyl)carbamoyl]-N~6~-(4-Iodobenzoyl)-L-LysineKi318.0 [1]
N~2~-{[(S)-Carboxy(4-Hydroxyphenyl)methyl]carbamoyl}-N~6~-(4-Iodobenzoyl)-L-LysineKi85.1 [1]
N~2~-{[(1s)-1-Carboxy-2-(Pyridin-4-Yl)ethyl]carbamoyl}-N~6~-(4-Iodobenzoyl)-L-LysineKi105.0 [1]
2-[(3-Carboxyphenyl)methoxy]-5-(sulfanylmethyl)benzoic acidIC502.0 [1]
2-(2-Mercaptoethyl)Benzoic AcidIC50930.0 [1]
Benzoic acid, 3-(1-carboxy-4-mercaptobutoxy)-IC5014.0 [1]
3-(1-Oxo-3,4-dihydroisothiochromen-8-yl)benzoic acidIC5020000.0 [1]
1-[(4-Bromo-3-carboxyphenyl)methyl]-3-(2-mercaptoethyl)-1h-indole-2-carboxylic acidIC50140.0 [1]
2-(4-Mercapto-butyl)-pentanedioic acidIC501100.0 [1]
2-[(3-Carboxyphenyl)methoxy]-6-(2-sulfanylethyl)benzoic acidIC5069.0 [1]
3-(2-Mercaptoethyl)-1H-indole-2-carboxylic acidIC501200.0 [1]
3-(2-Mercaptoethyl)-1-(phenylmethyl)-1h-indole-2-carboxylic acidIC5012000.0 [1]
1-[[3-Carboxy-5-(1,1-dimethylethyl)phenyl]methyl]-3-(2-mercaptoethyl)-1h-indole-2-carboxylic acidIC5034.0 [1]
1-[(2-Carboxyphenyl)methyl]-3-(2-mercaptoethyl)-1h-indole-2-carboxylic acidIC5022.0 [1]
3-(2-Mercaptoethyl)-1-phenyl-1H-indole-2-carboxylic acidIC506100.0 [1]
1-[(4-Carboxyphenyl)methyl]-3-(2-mercaptoethyl)-1h-indole-2-carboxylic acidIC5094.0 [1]
1-[(3-Carboxyphenyl)methyl]-3-(2-mercaptoethyl)-1h-indole-2-carboxylic acidIC5022.0 [1]
3-{2-Carboxy-2-[(hydroxycarbamoyl)methyl]ethyl}benzoic acidIC5015000.0 [1]
2-[[Hydroxy(phenylmethoxy)phosphoryl]methyl]pentanedioic acidIC5012.5 [1]
3-[2-(2-Benzoyloxymethyl-3-benzyl-4-oxo-azetidin-1-yl)-2-oxo-ethyl]-benzoic acid benzyl esterIC50100000.0 [1]
Benzoic acid 3-benzyl-1-ethanesulfonyl-4-oxo-azetidin-2-ylmethyl esterIC502190.0 [1]
Benzoic acid 1-benzenesulfonyl-3-benzyl-4-oxo-azetidin-2-ylmethyl esterIC503080.0 [1]
1-Benzoyl-3-(4-hydroxy-benzyl)-4-oxo-azetidine-2-carboxylic acid benzyl esterIC509140.0 [1]
Benzoic acid 3-benzyl-1-(4-nitro-benzenesulfonyl)-4-oxo-azetidin-2-ylmethyl esterIC5011500.0 [1]
Benzoic acid 3-benzyl-4-oxo-1-(toluene-4-sulfonyl)-azetidin-2-ylmethyl esterIC504790.0 [1]
3-Benzyl-4-oxo-1-(toluene-4-sulfonyl)-azetidine-2-carboxylic acid benzyl esterIC5030000.0 [1]
Benzoic acid 1-benzoyl-3-benzyl-4-oxo-azetidin-2-ylmethyl esterIC501590.0 [1]
4-[[(2S,3S)-1-Benzoyl-3-benzyl-4-oxoazetidin-2-yl]methoxycarbonyl]benzoic acidIC50100000.0 [1]
1-Benzoyl-3-benzyl-4-oxo-azetidine-2-carboxylic acid 4-carboxy-benzyl esterIC5024300.0 [1]
2-(2-Phosphonooxy-ethyl)-pentanedioic acidIC501200.0 [1]
2-(5-Mercapto-pentyl)-pentanedioic acidIC502600.0 [1]
2-Phosphonopentanedioic AcidIC501400.0 [1]
2-[3-(4,6-Dicarboxy-hexyldisulfanyl)-propyl]-pentanedioic acidIC503100.0 [1]
2-(3-Tritylsulfanyl-propyl)-pentanedioic acidIC5010000.0 [1]
Tetralithium;(2S)-2-(phosphonatoamino)pentanedioateIC500.86 [1]
(2R,4S)-2-Benzyl-4-[[(1S,3R)-1,3-dicarboxy-4-phenylbutyl]carbamoylamino]pentanedioic acidKi392.0 [1]
3-[2-Carboxy-2-(phosphonomethyl)ethyl]benzoic acidIC50120.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Glutamate carboxypeptidase II Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 10 May. 2024, https://www.aatbio.com/data-sets/glutamate-carboxypeptidase-ii-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 10). Quest Database™ Glutamate carboxypeptidase II Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/glutamate-carboxypeptidase-ii-inhibitors-ic50-ki.
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