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Glutamate NMDA receptor; GRIN1/GRIN2A Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
MemantineIC500.95 [1], 911.0 [2], 4360.0 [3], 4400.0 [4], 5600.0 [5]
KetamineIC503310.0 [1], 6100.0 [2]
TacrineIC504900.0 [1]
DexoxadrolIC509.7 [1]
DexoxadrolKi19.0 [1]

References
This online resource may be cited as follows
MLA
"Quest DatabaseGlutamate NMDA receptor; GRIN1/GRIN2A Inhibitors (IC50, Ki)." AAT Bioquest, Inc.13 Jan2026https://www.aatbio.com/data-sets/glutamate-nmda-receptor-grin1-grin2a-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2026January 13). Quest DatabaseGlutamate NMDA receptor; GRIN1/GRIN2A Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/glutamate-nmda-receptor-grin1-grin2a-inhibitors-ic50-ki.
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