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Glutamate [NMDA] receptor subunit epsilon 1 Inhibitors (IC50, Ki)

Structure
Compound Name
Standard Type
Standard Values (in nM)
DizocilpineIC5029.0 [1]
N-(4-(2-Benzoylhydrazinecarbonyl)benzyl)-3-chloro-4-fluorobenzenesulfonamideIC50109.0 [1]
4-(Trifluoromethoxy)-N'-[[2-(trifluoromethyl)phenyl]methyl]benzenecarboximidamideIC5010000.0 [1]
4-[4-(4-Benzylpiperidino)-1-butynyl]phenolIC50100000.0 [1]
2-Methyl-5-[3-(4-benzylpiperidino)propylthio]-1,3,4-thiadiazoleIC50100000.0 [1]
N-(4-(Benzyloxy)phenethyl)pyridin-4-amineIC5020000.0 [1]
5-[2-(4-Benzylpiperidino)ethylthio]-1H-1,2,4-triazole-3-amineIC50100000.0 [1]
1-[3-(Phenylthio)propyl]-4-benzylpiperidineIC5085000.0 [1]
5-[3-(4-Benzylpiperidino)propylthio]-1H-1,2,4-triazole-3-amineIC5077000.0 [1]
2-[3-(4-Benzylpiperidino)propylthio]-1H-imidazoleIC5077000.0 [1]
3-Methyl-5-[3-(4-benzylpiperidino)propylthio]-1H-1,2,4-triazoleIC50100000.0 [1]
5-[3-(4-Benzylpiperidino)propylthio]-1,3,4-thiadiazole-2-amineIC5073000.0 [1]
2-[3-(4-Benzylpiperidino)propylthio]-5-nitro-1H-benzimidazoleIC5061000.0 [1]
2-[3-(4-Benzylpiperidino)propylthio]-1H-benzimidazoleIC5064000.0 [1]
1-[2-(Phenylthio)ethyl]-4-benzylpiperidineIC50100000.0 [1]
3,4-Dichloro-N-(3-chloro-benzyl)-benzamidineIC5010000.0 [1]
5-[2-(4-Benzylpiperidino)ethylthio]-1,3,4-thiadiazole-2-amineIC50100000.0 [1]
4-[2-(4-Benzylpiperidino)ethylthio]phenolIC5035000.0 [1]
2-[2-(4-Benzylpiperidino)ethylthio]-1H-benzimidazoleIC5075000.0 [1]
2-[2-(4-Benzylpiperidino)ethylthio]-3H-imidazo[4,5-b]pyridineIC50100000.0 [1]
2-[2-(4-Benzylpiperidino)ethylthio]-5-nitro-1H-benzimidazoleIC50100000.0 [1]
2-[3-(4-Benzylpiperidino)propylthio]-3H-imidazo[4,5-b]pyridineIC50100000.0 [1]
3-Methyl-5-[2-(4-benzylpiperidino)ethylthio]-1H-1,2,4-triazoleIC50100000.0 [1]
3-[3-(4-Benzylpiperidino)propylthio]-2H-1,2,4-triazoleIC5051000.0 [1]
2-Methyl-5-[2-(4-benzylpiperidino)ethylthio]-1,3,4-thiadiazoleIC50100000.0 [1]
3,4-Dichloro-N-(2-trifluoromethoxy-benzyl)-benzamidineIC5010000.0 [1]
N-(3,5-Dimethyl-benzyl)-4-trifluoromethoxy-benzamidineIC5010000.0 [1]
N-(3,5-Dichloro-benzyl)-4-trifluoromethoxy-benzamidineIC5010000.0 [1]
2-[2-(4-Benzylpiperidino)ethylthio]-1H-imidazoleIC50100000.0 [1]
5-[2-(4-Benzylpiperidino)ethylthio]-1H-1,2,4-triazoleIC50100000.0 [1]



References

This online tool may be cited as follows

MLA

"Quest Database™ Glutamate [NMDA] receptor subunit epsilon 1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.9 May2024https://www.aatbio.com/data-sets/glutamate-nmda-receptor-subunit-epsilon-1-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024May 9). Quest Database™ Glutamate [NMDA] receptor subunit epsilon 1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/glutamate-nmda-receptor-subunit-epsilon-1-inhibitors-ic50-ki.
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