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Glutamate receptor ionotropic, AMPA 1 Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
PerampanelIC50243.0 [1], 485.0 [2], 623.0 [3], 1180.0 [4], 6510.0 [5]
4-[Methyl-(4-pyridin-2-yl-1,3-thiazol-2-yl)amino]phenolIC502970.0 [1], 83300.0 [2]
Glutamic acidKi1360.0 [1], 1362.0 [2]
Kainic acidKi7449.0 [1], 7450.0 [2], 7500.0 [3]
Argiotoxin 636IC50350.0 [1], 3400.0 [2]

References
This online resource may be cited as follows
MLA
"Quest DatabaseGlutamate receptor ionotropic, AMPA 1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.7 Dec2025https://www.aatbio.com/data-sets/glutamate-receptor-ionotropic-ampa-1-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 7). Quest DatabaseGlutamate receptor ionotropic, AMPA 1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/glutamate-receptor-ionotropic-ampa-1-inhibitors-ic50-ki.
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