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Glutamate receptor ionotropic kainate 1 Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
2,3-Dioxo-6-nitro-7-sulfamoylbenzo(f)quinoxalineIC5037000.0 [1], 50000.0 [2]
2,3-Dioxo-6-nitro-7-sulfamoylbenzo(f)quinoxalineKi11730.0 [1]
(2S,4R)-2-Amino-4-[(E)-3-naphthalen-2-ylprop-2-enyl]pentanedioic acidKi14.0 [1], 14.8 [2], 15.0 [3], 10000.0 [4]
4-Chloro-2-(3-(naphthalen-2-yl)ureido)benzoic acidIC501200.0 [1], 30000.0 [2], 69000.0 [3]
2-(3-(3-Bromophenyl)ureido)-4-chlorobenzoic acidIC504800.0 [1], 30000.0 [2]

References
This online resource may be cited as follows
MLA
"Quest DatabaseGlutamate receptor ionotropic kainate 1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.4 Feb2026https://www.aatbio.com/data-sets/glutamate-receptor-ionotropic-kainate-1-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2026February 4). Quest DatabaseGlutamate receptor ionotropic kainate 1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/glutamate-receptor-ionotropic-kainate-1-inhibitors-ic50-ki.
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