Glutaminase liver isoform, mitochondrial Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	(5Z)-5-{[1-(4-Bromophenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-4-hydroxy-1,3-thiazol-2(5H)-one	IC50	100000.0 [1]
	5-[3-[(Z)-(2,4-Dioxo-1,3-thiazolidin-5-ylidene)methyl]-2,5-dimethylpyrrol-1-yl]-2-[4-[(Z)-(2,4-dioxo-1,3-thiazolidin-5-ylidene)methyl]-3-ethylphenyl]benzonitrile	IC50	1185.0 [1]
	(5Z)-5-[[4-[4-[3-[(Z)-(2,4-Dioxo-1,3-thiazolidin-5-ylidene)methyl]-2,5-dimethylpyrrol-1-yl]-2-methoxyphenyl]-2-ethylphenyl]methylidene]-1,3-thiazolidine-2,4-dione	IC50	1189.0 [1]
	(5Z)-5-[[4-[4-[3-[(Z)-(2,4-Dioxo-1,3-thiazolidin-5-ylidene)methyl]-2,5-diphenylpyrrol-1-yl]-2-methoxyphenyl]phenyl]methylidene]-1,3-thiazolidine-2,4-dione	IC50	787.0 [1]
	(5Z)-5-[[4-[4-[3-[(Z)-(2,4-Dioxo-1,3-thiazolidin-5-ylidene)methyl]-2,5-dimethylpyrrol-1-yl]-2-methoxyphenyl]phenyl]methylidene]-1,3-thiazolidine-2,4-dione	IC50	2142.0 [1]
	(5Z)-5-[[4-[4-[3-[(Z)-(2,4-Dioxo-1,3-thiazolidin-5-ylidene)methyl]-2,5-dimethylpyrrol-1-yl]phenyl]-2-ethylphenyl]methylidene]-1,3-thiazolidine-2,4-dione	IC50	1031.0 [1]
	(5Z)-5-[[2-Chloro-4-[4-[3-[(Z)-(2,4-dioxo-1,3-thiazolidin-5-ylidene)methyl]-2,5-dimethylpyrrol-1-yl]phenyl]phenyl]methylidene]-1,3-thiazolidine-2,4-dione	IC50	4188.0 [1]
	(5Z)-5-[[1-(4-Bromophenyl)-2,5-diphenylpyrrol-3-yl]methylidene]-1,3-thiazolidine-2,4-dione	IC50	11753.0 [1]
	(5Z)-5-[[4-[4-[3-[(Z)-(2,4-Dioxo-1,3-thiazolidin-5-ylidene)methyl]-2,5-diphenylpyrrol-1-yl]phenyl]-2-ethylphenyl]methylidene]-1,3-thiazolidine-2,4-dione	IC50	1244.0 [1]
	(5Z)-5-[[4-[4-[3-[(Z)-(2,4-Dioxo-1,3-thiazolidin-5-ylidene)methyl]-2,5-diphenylpyrrol-1-yl]phenyl]phenyl]methylidene]-1,3-thiazolidine-2,4-dione	IC50	261.0 [1]
	(5Z)-5-[[4-[4-[3-[(Z)-(2,4-Dioxo-1,3-thiazolidin-5-ylidene)methyl]-2,5-dimethylpyrrol-1-yl]-2-hydroxyphenyl]phenyl]methylidene]-1,3-thiazolidine-2,4-dione	IC50	5725.0 [1]
	(5Z)-5-[[4-[4-[3-[(Z)-(2,4-Dioxo-1,3-thiazolidin-5-ylidene)methyl]-2,5-dithiophen-2-ylpyrrol-1-yl]phenyl]phenyl]methylidene]-1,3-thiazolidine-2,4-dione	IC50	102.0 [1]
	(5Z)-5-[[4-[4-[3-[(Z)-(2,4-Dioxo-1,3-thiazolidin-5-ylidene)methyl]-2,5-dithiophen-2-ylpyrrol-1-yl]-2-methoxyphenyl]phenyl]methylidene]-1,3-thiazolidine-2,4-dione	IC50	269.0 [1]
	(5Z)-5-[[4-[4-[3-[(Z)-(2,4-Dioxo-1,3-thiazolidin-5-ylidene)methyl]-2,5-dimethylpyrrol-1-yl]phenyl]phenyl]methylidene]-1,3-thiazolidine-2,4-dione	IC50	1188.0 [1]
	(5Z)-5-[[1-(4-Bromophenyl)-2,5-dithiophen-2-ylpyrrol-3-yl]methylidene]-1,3-thiazolidine-2,4-dione	IC50	3778.0 [1]
	(5Z)-5-[[4-[4-[3-[(Z)-(2,4-Dioxo-1,3-thiazolidin-5-ylidene)methyl]-2,5-dithiophen-2-ylpyrrol-1-yl]phenyl]-2-ethylphenyl]methylidene]-1,3-thiazolidine-2,4-dione	IC50	1716.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 16 ⟨⟩

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References

This online tool may be cited as follows

MLA	"Quest Database™ Glutaminase liver isoform, mitochondrial Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/glutaminase-liver-isoform-mitochondrial-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, May 9). Quest Database™ Glutaminase liver isoform, mitochondrial Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/glutaminase-liver-isoform-mitochondrial-inhibitors-ic50-ki.
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