Name: GRIA1/CACNG8 Inhibitors (IC50, Ki)
Creator: AAT Bioquest
License: https://www.aatbio.com/tou.html

GRIA1/CACNG8 Inhibitors (IC50, Ki)

Structure	Compound Name	Standard Type	Standard Values (in nM)
	5-[2-Chloro-6-(trifluoromethoxy)phenyl]-1,3-dihydrobenzimidazol-2-one	IC50	10.0 ^[1]
	5-[3-Chloro-5-(trifluoromethoxy)pyridin-4-yl]-7-methyl-1,3-dihydroindol-2-one	IC50	2.51 ^[1]
	AMPA Receptor Modulator-1	IC50	0.2 ^[1]
	5-[3-Chloro-5-(difluoromethoxy)pyridin-4-yl]-7-methyl-1,3-dihydroindol-2-one	IC50	7.94 ^[1]
	5-[2-Chloro-6-(trifluoromethoxy)phenyl]-1,3-dihydroindol-2-one	IC50	15.85 ^[1]
Rows per page: 1–5 of 18

References

This online resource may be cited as follows

MLA	"Quest Database™ GRIA1/CACNG8 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 6 Feb. 2026, https://www.aatbio.com/data-sets/gria1-cacng8-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2026, February 6). Quest Database™ GRIA1/CACNG8 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/gria1-cacng8-inhibitors-ic50-ki.
BibTeX	EndNote	RefMan