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Group X secretory phospholipase A2 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
▲
▼
Standard Values (in nM)
▲
▼
VarespladibIC5041.0 [1], 75.0 [2], 107.15 [3], 150.0 [4]
Spla2-X inhibitor 31IC5026.0 [1], 270.0 [2], 310.0 [3]
4-(3,5-Didodecanoyl-2,4,6-trihydroxyphenyl)-7-hydroxy-2-(4-hydroxyphenyl)chromanIC50200.0 [1], 1600.0 [2]
Mesyl-2-(3-(2-amino-2-oxoacetyl)-1-benzyl-2-isobutyl-1H-indol-4-yloxy)acetamideIC507.0 [1]
1-[3-(Trifluoromethyl)phenyl]indole-2-carboxamideIC506900.0 [1]
3-[3-(2-Carbamoyl-6-chloroindol-1-yl)phenyl]propanoic acidIC5090.0 [1], 1100.0 [2]
3-[3-(2-Carbamoyl-6-cyclopropylindol-1-yl)phenyl]propanoic acidIC50160.0 [1], 1900.0 [2]
3-[3-(2-Carbamoyl-6-cyanoindol-1-yl)phenyl]propanoic acidIC50110.0 [1], 990.0 [2]
3-[3-[2-Carbamoyl-6-(difluoromethoxy)indol-1-yl]phenyl]propanoic acidIC5068.0 [1], 370.0 [2]
3-[2-[2-Carbamoyl-6-(trifluoromethoxy)indol-1-yl]pyridin-4-yl]propanoic acidIC50110.0 [1], 640.0 [2]
3-[3-[2-Carbamoyl-6-(trifluoromethoxy)indol-1-yl]phenyl]-2-methylpropanoic acidIC50100.0 [1], 2800.0 [2]
(3S)-3-[3-[2-Carbamoyl-6-(trifluoromethoxy)indol-1-yl]phenyl]butanoic acidIC5015.0 [1], 110.0 [2]
3-[3-[2-Carbamoyl-6-(trifluoromethyl)indol-1-yl]phenyl]propanoic acidIC5043.0 [1], 480.0 [2]
3-[3-[2-Carbamoyl-6-(2,2,2-trifluoroethoxy)indol-1-yl]phenyl]propanoic acidIC5093.0 [1], 740.0 [2]
3-[6-[2-Carbamoyl-6-(trifluoromethoxy)indol-1-yl]pyridin-2-yl]propanoic acidIC5029.0 [1], 250.0 [2]
3-[4-[2-Carbamoyl-6-(trifluoromethoxy)indol-1-yl]pyridin-2-yl]propanoic acidIC50240.0 [1], 1600.0 [2]
3-[2-[2-Carbamoyl-6-(trifluoromethoxy)indol-1-yl]pyridin-4-yl]-2-methylpropanoic acidIC50360.0 [1], 3400.0 [2]
AmentoflavoneIC50100000.0 [1]
IndoxamIC501600.0 [1]
OchnaflavoneIC50100000.0 [1]
N-Hexadecanoyl-leucineIC501660.0 [1]
6-(4-Oxo-2-phenyl-chromen-6-yl)-2-phenyl-chromen-4-oneIC50100000.0 [1]
DidodecanoylphloroglucinolIC501600.0 [1]
2-(3-(2-Amino-2-oxoacetyl)-1-benzyl-2-ethyl-1H-indol-4-yloxy)propanoic acidIC5022.0 [1]
2-(1-Benzyl-6-methoxy-2-methyl-1H-indol-3-yl)-2-hydroxy-acetamideIC50250000.0 [1]
2-{4-[4-(4-Oxo-4H-chromen-2-yl)phenyl]phenyl}-4H-chromen-4-oneIC50100000.0 [1]
6-[3-(4-Oxo-4H-chromen-2-yl)-phenyl]-2-phenyl-chromen-4-oneIC5027600.0 [1]
2-{4-[3-(4-Oxo-4H-chromen-2-yl)phenyl]phenyl}-4H-chromen-4-oneIC50100000.0 [1]
6-[4-(4-Oxo-4H-chromen-2-yl)-phenyl]-2-phenyl-chromen-4-oneIC50100000.0 [1]
3-(4-(4-Oxo-4H-chromen-2-yl)phenyl)-2-phenyl-4H-chromen-4-oneIC50100000.0 [1]
Me-indoxamIC504570.0 [1]
((3-(2-Amino-1,2-dioxoethyl)-2-methyl-1-(phenylmethyl)-1H-indol-4-yl)oxy)acetic acidIC502000.0 [1]
2-[2-Ethyl-3-oxamoyl-1-(phenylmethyl)benzo[g]indol-4-yl]oxyacetic acidIC5020.0 [1]
2-Phenoxy-6-methoxyquinoline-4-carboxamideIC5010000.0 [1]
(S)-4-((S)-(E)-Dec-3-enoylamino)-5-(naphthalen-2-ylsulfanyl)-pentanoic acidIC50380.0 [1]
2-Phenoxy-6-methoxyquinoline-4-acetamideIC501000.0 [1]
(R)-2-((S)-Hexadecanoylamino)-4-methyl-pentanoic acidIC5030000.0 [1]
(3S)-4-(4-Benzylphenyl)sulfanyl-3-[[(E)-dec-3-enoyl]amino]butanoic acidIC50120.0 [1]
2-[4-[2-(Benzenesulfonamido)-2-oxoethoxy]-1-benzyl-2-(2-methylpropyl)indol-3-yl]-2-oxoacetamideIC5021.0 [1]
2-(3-(2-Amino-2-oxoacetyl)-1-benzyl-2-isobutyl-1H-indol-4-yloxy)acetic acidIC5050.0 [1]
(S)-4-((S)-Hexadecanoylamino)-6-methyl-heptanoic acidIC504500.0 [1]
(S)-3-((S)-(E)-Dec-3-enoylamino)-4-(naphthalen-2-ylsulfanyl)-butyric acidIC50790.0 [1]
(S)-3-((S)-(E)-Dec-3-enoylamino)-4-phenylsulfanyl-butyric acidIC502200.0 [1]
(R)-3-((S)-Decanoylamino)-5-methyl-hexanoic acidIC5015000.0 [1]
(R)-3-((S)-Hexadecanoylamino)-5-methyl-hexanoic acidIC507300.0 [1]
(4R)-4-[[(E)-Dec-3-enoyl]amino]-5-naphthalen-2-ylsulfanylpentanoic acidIC50100000.0 [1]
2-Phenoxy-6-hydroxyquinoline-4-acetamideIC5010000.0 [1]
2-(1-Benzyl-2,6-dimethyl-3-oxamoylindol-4-yl)oxyacetic acidIC502200.0 [1]
3-(2-Methyl-5-propan-2-ylthiophen-3-yl)-1H-pyrazole-5-carboxamideIC5051.29 [1]
3-(2-Methyl-1-benzothiophen-3-yl)-1H-pyrazole-5-carboxamideIC50173.78 [1]
3-(2-Methyl-5-phenylthiophen-3-yl)-1H-pyrazole-5-carboxamideIC50346.74 [1]
3-(2,5-Dichlorothiophen-3-yl)-1H-pyrazole-5-carboxamideIC50398.11 [1]
3-(2-Methylthiophen-3-yl)-1H-pyrazole-5-carboxamideIC50630.96 [1]
1-Methyl-5-(2-methyl-1-benzothiophen-3-yl)pyrazole-3-carboxamideIC50851.14 [1]
5-(2,5-Dimethylthiophen-3-yl)-1-methylpyrazole-3-carboxamideIC50851.14 [1]
1-Methyl-5-(2-methyl-5-phenylthiophen-3-yl)pyrazole-3-carboxamideIC501202.26 [1]
(3R)-3-[3-[2-Carbamoyl-6-(trifluoromethoxy)indol-1-yl]phenyl]butanoic acidIC50200.0 [1]
3-[4-(3-Phenylmethoxy-2-tetradecoxypropoxy)phenyl]-4H-1,2,4-oxadiazol-5-oneIC5014000.0 [1]
3-[4-(3-Decoxy-2-tetradecoxypropoxy)phenyl]-4H-1,2,4-oxadiazol-5-oneIC501000.0 [1]
3-[4-[3-(4-Phenylbutoxy)-2-tetradecoxypropoxy]phenyl]-4H-1,2,4-oxadiazol-5-oneIC5012000.0 [1]
3-[4-(3-Benzhydryloxy-2-tetradecoxypropoxy)phenyl]-4H-1,2,4-oxadiazol-5-oneIC505300.0 [1]
3-[4-(2-Tetradecoxy-3-trityloxypropoxy)phenyl]-4H-1,2,4-oxadiazol-5-oneIC501250.0 [1]
4-[[3-[4-[(5-Oxo-4H-1,2,4-oxadiazol-3-yl)methyl]phenoxy]-2-tetradecoxypropoxy]methyl]benzonitrileIC505000.0 [1]
4-[[2-Octadecoxy-3-[4-[(5-oxo-4H-1,2,4-oxadiazol-3-yl)methyl]phenoxy]propoxy]methyl]benzonitrileIC50900.0 [1]
3-[3-(2-Carbamoyl-6-methylindol-1-yl)phenyl]propanoic acidIC50230.0 [1]
3-[(2-Carbamoylindol-1-yl)methyl]benzoic acidIC5020700.0 [1]
1-[3-[3-(Methanesulfonamido)-3-oxopropyl]phenyl]indole-2-carboxamideIC504800.0 [1]
2-[[3-(2-Carbamoylindol-1-yl)benzoyl]amino]acetic acidIC507200.0 [1]
3-(2-Carbamoylindol-1-yl)benzoic acidIC5029100.0 [1]
3-[3-(2-Carbamoyl-5-methylindol-1-yl)phenyl]propanoic acidIC502700.0 [1]
3-[3-(2-Carbamoyl-7-methylindol-1-yl)phenyl]propanoic acidIC501900.0 [1]
(E)-3-[3-(2-Carbamoylindol-1-yl)phenyl]prop-2-enoic acidIC5023600.0 [1]
3-[3-[2-Carbamoyl-6-(hydroxymethyl)indol-1-yl]phenyl]propanoic acidIC502800.0 [1]
2-[3-(2-Carbamoylindol-1-yl)phenoxy]acetic acidIC5026900.0 [1]
1-[3-(3-Amino-3-oxopropyl)phenyl]indole-2-carboxamideIC5030000.0 [1]
3-[3-(2-Carbamoyl-6-methoxyindol-1-yl)phenyl]propanoic acidIC50620.0 [1]
3-[3-(2-Carbamoyl-6-fluoroindol-1-yl)phenyl]propanoic acidIC50260.0 [1]
3-[3-(2-Carbamoyl-4-methylindol-1-yl)phenyl]propanoic acidIC50830.0 [1]
3-[5-[2-Carbamoyl-6-(trifluoromethoxy)indol-1-yl]-2-oxopyridin-1-yl]propanoic acidIC504800.0 [1]
3-[3-[2-Carbamoyl-6-(trifluoromethoxy)indol-1-yl]pyrazol-1-yl]propanoic acidIC504800.0 [1]
3-[3-(2-Carbamoylindol-1-yl)phenyl]propanoic acidIC50990.0 [1]
3-[6-[2-Carbamoyl-6-(trifluoromethoxy)indol-1-yl]pyridin-2-yl]butanoic acidIC50500.0 [1]
2-[3-(2-Carbamoylindol-1-yl)phenyl]acetic acidIC5010300.0 [1]
3-[3-(2-Carbamoyl-6-ethylindol-1-yl)phenyl]propanoic acidIC50170.0 [1]
3-[4-[2-Carbamoyl-6-(trifluoromethoxy)indol-1-yl]pyrazol-1-yl]propanoic acidIC5010000.0 [1]
3-[3-[2-Carbamoyl-6-(trifluoromethoxy)indol-1-yl]phenyl]-2-methoxypropanoic acidIC50170.0 [1]
2-[[6-[2-Carbamoyl-6-(trifluoromethoxy)indol-1-yl]pyridin-2-yl]methyl]butanoic acidIC50940.0 [1]
3-[6-[2-Carbamoyl-6-(trifluoromethoxy)indol-1-yl]pyridin-2-yl]-2-methylpropanoic acidIC50570.0 [1]
3-[5-[2-Carbamoyl-6-(trifluoromethoxy)indol-1-yl]furan-2-yl]propanoic acidIC50430.0 [1]
3-[6-[2-Carbamoyl-6-(trifluoromethoxy)indol-1-yl]pyridin-2-yl]-2,2-dimethylpropanoic acidIC50320.0 [1]
Tert-butyl 2-[(7S)-7-benzyl-5-methyl-1-[2-[(2-methylpropan-2-yl)oxy]-2-oxoethyl]-2,6-dioxo-1,3,5-triazepan-3-yl]acetateIC5011000.0 [1]
2-[3-Biphenyl-2-ylmethyl-2-ethyl-8-(2-oxo-propoxy)-indolizin-1-yl]-2-oxo-acetamideIC501600.0 [1]
2-[4-[2-(Benzenesulfonamido)-2-oxoethoxy]-1-benzyl-2-ethylbenzo[g]indol-3-yl]-2-oxoacetamideIC5090.0 [1]
2-[4-[2-(Benzenesulfonamido)-2-oxoethoxy]-1-benzyl-2-(2-methylpropyl)benzo[g]indol-3-yl]-2-oxoacetamideIC5030.0 [1]
2-[1-Benzyl-2-(2-methylpropyl)-3-oxamoylbenzo[g]indol-4-yl]oxyacetic acidIC5010.0 [1]
N-(Benzenesulfonyl)-2-[1-benzyl-2-(2-methylpropyl)-3-oxamoylindol-4-yl]oxypropanamideIC5080.0 [1]
2-[1-Benzyl-4-[2-[(4-chlorophenyl)sulfonylamino]-2-oxoethoxy]-2-(2-methylpropyl)indol-3-yl]-2-oxoacetamideIC50540.0 [1]
2-[1-Benzyl-4-[2-[(3-chlorophenyl)sulfonylamino]-2-oxoethoxy]-2-(2-methylpropyl)indol-3-yl]-2-oxoacetamideIC50140.0 [1]
2-[1-Benzyl-4-[2-[(2-chlorophenyl)sulfonylamino]-2-oxoethoxy]-2-(2-methylpropyl)indol-3-yl]-2-oxoacetamideIC5014.0 [1]
2-[1-Benzyl-4-[2-[(4-methylphenyl)sulfonylamino]-2-oxoethoxy]-2-(2-methylpropyl)indol-3-yl]-2-oxoacetamideIC50320.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Group X secretory phospholipase A2 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/group-x-secretory-phospholipase-a2-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 9). Quest Database™ Group X secretory phospholipase A2 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/group-x-secretory-phospholipase-a2-inhibitors-ic50-ki.
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