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Heat shock protein HSP 90-alpha Inhibitors (IC50, Ki)

Structure
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Compound Name
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▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
GeldanamycinIC5027.0 [1]
TanespimycinIC50309.0 [1]
TanespimycinKi4.6 [1], 29.0 [2]
LuminespibIC500.4 [1], 7.8 [2], 12.0 [3], 22.0 [4], 25.0 [5]
LuminespibKi2.0 [1]
6-Chloro-9-((4-methoxy-3,5-dimethylpyridin-2-yl)methyl)-9H-purin-2-amineIC505.1 [1], 19.0 [2], 29.0 [3], 52.0 [4], 65.7 [5]
6-Chloro-9-((4-methoxy-3,5-dimethylpyridin-2-yl)methyl)-9H-purin-2-amineKi1.7 [1], 2.0 [2]
PU-H71IC5043.0 [1], 51.0 [2], 89.0 [3]
RadicicolIC5016.0 [1], 150.0 [2], 530.0 [3]
Snx-2112IC503.0 [1], 29.0 [2]
Snx-2112Ki4.0 [1]
5-(5-Chloro-2,4-dihydroxyphenyl)-N-ethyl-4-(4-methoxyphenyl)-1H-pyrazole-3-carboxamideIC5019.0 [1], 25.0 [2], 880.0 [3]
Methyl 2-[2-(1-benzyl-1H-imidazol-2-yl)ethyl]-3-chloro-4,6-dihydroxybenzoateIC5013100.0 [1], 13200.0 [2], 14000.0 [3]
(16S)-5,5,9,16-Tetramethyl-7-oxo-2,14,17-triazatetracyclo[16.3.1.02,10.03,8]docosa-1(22),3(8),9,18,20-pentaene-19-carboxamideIC50110.0 [1]
1-(2-Hydroxy-5-(trifluoromethyl)phenyl)-5-(trifluoromethyl)-1H-benzo[d]imidazol-2(3H)-oneIC503320.0 [1], 81000.0 [2]
5-[2-Amino-4-chloro-7-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]pyrrolo[2,3-d]pyrimidin-5-yl]-2-methylpent-4-yn-2-olIC501.1 [1]
5-[2-Amino-4-chloro-7-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]pyrrolo[2,3-d]pyrimidin-5-yl]-2-methylpent-4-yn-2-olKi0.2 [1]
(18S)-5,5,9-Trimethyl-7-oxo-2,14,20-triazapentacyclo[19.3.1.02,10.03,8.014,18]pentacosa-1(25),3(8),9,21,23-pentaene-22-carboxamideIC5096.0 [1], 1037.0 [2]
(16S)-5,5,9,16-Tetramethyl-7-oxo-2,13,17-triazatetracyclo[16.3.1.02,10.03,8]docosa-1(22),3(8),9,18,20-pentaene-19-carboxamideIC50210.0 [1]
3-(5-Chloro-2,4-dihydroxyphenyl)-1H-benzimidazol-2-oneIC5054.0 [1], 15200.0 [2]
1-(2,4-Dihydroxyphenyl)-1,3-Dihydro-2h-Benzimidazol-2-OneIC50220.0 [1], 85000.0 [2]
N-[[1-(5-Chloro-2,4-dihydroxyphenyl)-2-oxo-3H-benzimidazol-5-yl]methyl]naphthalene-1-sulfonamideIC5030.0 [1], 550.0 [2]
N-[[1-(5-Chloro-2,4-dihydroxyphenyl)-2-oxo-3H-benzimidazol-5-yl]methyl]acetamideIC5040.0 [1], 24800.0 [2]
N-[[1-(5-Chloro-2,4-dihydroxyphenyl)-2-oxo-3H-benzimidazol-5-yl]methyl]methanesulfonamideIC5050.0 [1], 25200.0 [2]
1-[[1-(5-Chloro-2,4-dihydroxyphenyl)-2-oxo-3H-benzimidazol-5-yl]methyl]-3-phenylureaIC5060.0 [1], 15400.0 [2]
3-(2,5-Dihydroxyphenyl)-1H-benzimidazol-2-oneIC5034900.0 [1], 200000.0 [2]
3-(4-Chloro-2,5-dihydroxyphenyl)-1H-benzimidazol-2-oneIC502530.0 [1], 200000.0 [2]
N-[[1-(5-Chloro-2,4-dihydroxyphenyl)-2-oxo-3H-benzimidazol-5-yl]methyl]benzamideIC5072.0 [1], 22900.0 [2]
N-[[1-(5-Chloro-2,4-dihydroxyphenyl)-2-oxo-3H-benzimidazol-5-yl]methyl]naphthalene-2-sulfonamideIC5047.0 [1], 1140.0 [2]
1-[[1-(5-Chloro-2,4-dihydroxyphenyl)-2-oxo-3H-benzimidazol-5-yl]methyl]-3-ethylureaIC5033.0 [1], 14200.0 [2]
N-[[1-(5-Chloro-2,4-dihydroxyphenyl)-2-oxo-3H-benzimidazol-5-yl]methyl]benzenesulfonamideIC5027.0 [1], 3420.0 [2]
3-[2-Hydroxy-5-(trifluoromethyl)phenyl]-1H-benzimidazol-2-oneIC502320.0 [1], 127000.0 [2]
2-(4-Hydroxycyclohexylamino)-4-(6-methoxyindol-1-yl)benzamideIC50100000.0 [1]
2-(4-Hydroxycyclohexylamino)-4-(4-methoxyindol-1-yl)benzamideIC50100000.0 [1]
3-Chloro-4-indol-1-ylbenzamideIC50100000.0 [1]
Adenosine-5'-triphosphateIC50861330.0 [1]
Adenosine-5'-diphosphateIC5059308.0 [1]
ThiamineIC5012500.0 [1]
VorinostatIC501000.0 [1]
2-ChloroadenosineIC501250000.0 [1]
AlvespimycinKi680.0 [1]
GanetespibIC505.0 [1]
OnalespibIC5013.6 [1]
4-[4-(2,3-Dihydro-1,4-benzodioxin-6-YL)-3-methyl-1H-pyrazol-5-YL]-6-ethylbenzene-1,3-diolIC50280.0 [1]
Nvp-hsp990(hsp990)IC5013.0 [1]
4-[4-(4-Methoxyphenyl)-5-methyl-1H-pyrazol-3-yl]benzene-1,3-diolIC504400.0 [1]
Debio 0932IC5033.0 [1]
CID 67495834Ki3.0 [1]
Tas-116IC50210.0 [1]
8-((6-Bromobenzo[d][1,3]dioxol-5-yl)thio)-9-(pent-4-yn-1-yl)-9H-purin-6-amineIC50300.0 [1]
8-((3,5-Dichlorophenyl)thio)-9-(3-(isopropylamino)propyl)-9H-purin-6-amineIC5027300.0 [1]
4-Chloro-6-[4-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-methyl-1H-pyrazol-3-yl]benzene-1,3-diolIC50210.0 [1]
4-Bromo-6-(6-hydroxy-1,2-benzisoxazol-3-yl)benzene-1,3-diolIC50190.0 [1]
CID 86280454Ki100000.0 [1]
9-(Pent-4-yn-1-yl)-8-((2,4,5-trichlorophenyl)thio)-9H-purin-6-amineIC50200000.0 [1]
8-((2,4-Dimethylphenyl)thio)-9-(pent-4-yn-1-yl)-9H-purin-6-amineIC50300000.0 [1]
8-((2,5-Dichlorophenyl)thio)-9-(pent-4-yn-1-yl)-9H-purin-6-amineIC5060400.0 [1]
8-((3,5-Dimethylphenyl)thio)-9-(pent-4-yn-1-yl)-9H-purin-6-amineIC50300000.0 [1]
8-((2,4-Dichlorophenyl)thio)-9-(pent-4-yn-1-yl)-9H-purin-6-amineIC50300000.0 [1]
8-((3,5-Dichlorophenyl)thio)-9-(pent-4-yn-1-yl)-9H-purin-6-amineIC50500000.0 [1]
8-((2,5-Dimethylphenyl)thio)-9-(pent-4-yn-1-yl)-9H-purin-6-amineIC50300000.0 [1]
4-Chloro-6-(6-hydroxy-1,2-benzoxazol-3-yl)benzene-1,3-diolIC5060.0 [1]
2-Chloro-9-methyl-9H-purin-6-amineIC501250000.0 [1]
4-(5-Chloro-1h,3h-Benzo[de]isochromen-6-Yl)-6-(Methylsulfanyl)-1,3,5-Triazin-2-AmineIC503000.0 [1]
4-(6-Hydroxy-benzo[D]isoxazol-3-YL)benzene-1,3-diolIC5015200.0 [1]
8-(2-Chloro-phenylsulfanyl)-9-pent-4-ynyl-9H-purin-6-ylamineIC50100000.0 [1]
8-(4-Methoxy-phenylsulfanyl)-9-pent-4-ynyl-9H-purin-6-ylamineIC50100000.0 [1]
[2-(6-Amino-9-pent-4-ynyl-9H-purin-8-ylsulfanyl)-phenyl]-methanolIC50100000.0 [1]
8-[2-Chloro-5-(trifluoromethyl)phenyl]sulfanyl-9-pent-4-ynylpurin-6-amineIC50100000.0 [1]
8-(4-Chloro-phenylsulfanyl)-9-pent-4-ynyl-9H-purin-6-ylamineIC50100000.0 [1]
9-Pent-4-ynyl-8-(2-trifluoromethoxy-phenylsulfanyl)-9H-purin-6-ylamineIC50100000.0 [1]
8-(2-Methoxy-phenylsulfanyl)-9-pent-4-ynyl-9H-purin-6-ylamineIC50100000.0 [1]
8-(2,4-Dimethoxy-phenylsulfanyl)-9-pent-4-ynyl-9H-purin-6-ylamineIC5050000.0 [1]
4-(Methylsulfanyl)-6-phenyl-1,3,5-triazin-2-amineIC5031000.0 [1]
3-(5-Chloro-2,4-dihydroxyphenyl)-4-(4-methoxyphenyl)-5-methyl-1H-pyrazoleIC50150.0 [1]
4-Chloro-6-{5-[(2-morpholin-4-ylethyl)amino]-1,2-benzisoxazol-3-yl}benzene-1,3-diolIC5030.0 [1]
8-[(2,4-Dimethylphenyl)sulfanyl]-3-Pent-4-Yn-1-Yl-3h-Purin-6-AmineIC50250000.0 [1]
4-(2-Morpholinoethylthio)-6-(methylthio)-1,3,5-triazine-2-amineIC5033000.0 [1]
4-(2-Methoxy-phenyl)-6-methyl-pyrimidin-2-yl-amineKi8300.0 [1]
4-Chloro-6-(2-Methoxyphenyl)pyrimidin-2-AmineKi1200.0 [1]
(16S)-13-Acetyl-5,5,9,16-tetramethyl-7-oxo-2,13,17-triazatetracyclo[16.3.1.02,10.03,8]docosa-1(22),3(8),9,18,20-pentaene-19-carboxamideIC50110.0 [1]
(16S)-5,5,9,16-Tetramethyl-7,15-dioxo-2,14,17-triazatetracyclo[16.3.1.02,10.03,8]docosa-1(22),3(8),9,18,20-pentaene-19-carboxamideIC5082.0 [1]
(16S)-13-[(2S)-2-Aminopropanoyl]-5,5,9,16-tetramethyl-7-oxo-2,13,17-triazatetracyclo[16.3.1.02,10.03,8]docosa-1(22),3(8),9,18,20-pentaene-19-carboxamideIC50145.0 [1]
1-(2,4-Dihydroxy-5-propan-2-ylphenyl)-N-ethyl-5-[4-(imidazol-1-ylmethyl)phenyl]triazole-4-carboxamideIC5023.0 [1]
1-(2,4-Dihydroxy-5-propan-2-ylphenyl)-N-ethyl-5-[4-(morpholin-4-ylmethyl)phenyl]triazole-4-carboxamideIC505.0 [1]
8-(Mesitylthio)-9-(pent-4-yn-1-yl)-9H-purin-6-amineIC50500000.0 [1]
2-[(2,4-Dihydroxyphenyl)sulfonyl]-2,3-Dihydro-1h-Isoindole-4,6-DiolIC5047000.0 [1]
4-[4-(2,3-Dihydro-1,4-benzodioxin-6-yl)-5-methyl-1H-pyrazol-3-yl]benzene-1,3-diolIC504730.0 [1]
5-(2,4-Dihydroxy-5-propan-2-ylbenzoyl)-N-ethyl-6,7-dihydro-4H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamideIC5029.0 [1]
Ethyl 5-(2,4-dihydroxy-5-propan-2-ylbenzoyl)-6,7-dihydro-4H-[1,2]oxazolo[4,5-c]pyridine-3-carboxylateIC50100.0 [1]
8-(2,4-Dichlorophenyl)sulfonyl-9-pent-4-ynylpurin-6-amineIC5025000.0 [1]
9-But-3-ynyl-8-(3,5-dichlorophenyl)sulfanylpurin-6-amineIC5050000.0 [1]
8-(2,4-Dichlorophenoxy)-9-pent-4-ynylpurin-6-amineIC50100000.0 [1]
8-(2,4-Dichlorophenyl)sulfanyl-9-pentan-2-ylpurin-6-amineIC50100000.0 [1]
8-(2,4-Dichlorophenyl)sulfinyl-9-pent-4-ynylpurin-6-amineIC5024900.0 [1]
8-[(2,4-Dichlorophenyl)methyl]-9-pent-4-ynylpurin-6-amineIC50100000.0 [1]
9-Benzyl-8-(3,5-dichlorophenyl)sulfanylpurin-6-amineIC5050000.0 [1]
8-(3,5-Dichlorophenyl)sulfanyl-9-(6,6,6-trifluorohexyl)purin-6-amineIC5050000.0 [1]
9-Pent-4-ynyl-8-(2,3,4-trichlorophenyl)sulfanylpurin-6-amineIC5015970.0 [1]
8-(3,5-Dichlorophenyl)sulfanyl-9-(2-phenylethyl)purin-6-amineIC5050000.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Heat shock protein HSP 90-alpha Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 10 May. 2024, https://www.aatbio.com/data-sets/heat-shock-protein-hsp-90-alpha-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 10). Quest Database™ Heat shock protein HSP 90-alpha Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/heat-shock-protein-hsp-90-alpha-inhibitors-ic50-ki.
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