 | Terfenadine | IC50 | 128.82 [1] |
| Terfenadine | Ki | 56.0 [1], 320.0 [2] |
 | Cisapride | IC50 | 39.81 [1] |
| Cisapride | Ki | 139.4 [1] |
 | Astemizole | IC50 | 8.0 [1] |
| Astemizole | Ki | 2.9 [1], 12.8 [2], 20.0 [3] |
 | Dofetilide | IC50 | 10.0 [1] |
| Dofetilide | Ki | 6.4 [1], 7.7 [2] |
 | Mibefradil | IC50 | 1400.0 [1] |
| Mibefradil | Ki | 190.0 [1], 353.0 [2] |
 | Risperidone | IC50 | 162.18 [1] |
| Risperidone | Ki | 920.0 [1], 3432.8 [2] |
 | Haloperidol | IC50 | 30.2 [1] |
| Haloperidol | Ki | 120.0 [1], 512.0 [2] |
 | Clozapine | IC50 | 323.59 [1] |
| Clozapine | Ki | 3080.0 [1], 4060.0 [2], 8660.6 [3], 17000.0 [4] |
 | Pimozide | IC50 | 20.0 [1] |
| Pimozide | Ki | 42.0 [1] |
 | Sparfloxacin | IC50 | 26302.68 [1] |
| Sparfloxacin | Ki | 38619.4 [1] |
 | Sertindole | IC50 | 10.0 [1] |
 | Thioridazine | IC50 | 95.5 [1] |
| Thioridazine | Ki | 869.0 [1], 1301.0 [2] |
 | Bepridil | IC50 | 549.54 [1] |
| Bepridil | Ki | 184.0 [1], 291.0 [2], 444.0 [3] |
 | Verapamil | IC50 | 141.25 [1] |
 | Levofloxacin | IC50 | 1100000.0 [1] |
| Levofloxacin | Ki | 150000.0 [1] |
 | Moxifloxacin | IC50 | 128824.96 [1] |
 | Fexofenadine | IC50 | 23000.0 [1] |
| Fexofenadine | Ki | 23000.0 [1] |
 | Halofantrine | IC50 | 199.53 [1] |
| Halofantrine | Ki | 7500.0 [1] |
 | N-(4-((1-(2-(6-Methyl-2-pyridinyl)ethyl)-4-piperidinyl)carbonyl)phenyl)methanesulfonamide | IC50 | 19.95 [1] |
 | 1-(2-(6-Methyl-2-pyridyl)ethyl)-4-(4-methylsulfonylaminobenzoyl)piperidine dihydrochloride | IC50 | 89.0 [1] |
| 1-(2-(6-Methyl-2-pyridyl)ethyl)-4-(4-methylsulfonylaminobenzoyl)piperidine dihydrochloride | Ki | 18.7 [1], 19.4 [2] |
 | Sildenafil | IC50 | 3311.31 [1] |
 | Amitriptyline | IC50 | 10000.0 [1] |
| Amitriptyline | Ki | 14410.6 [1] |
 | Grepafloxacin | IC50 | 50118.72 [1] |
 | Chlorpromazine | IC50 | 1479.11 [1] |
| Chlorpromazine | Ki | 4774.3 [1] |
 | Droperidol | IC50 | 32.36 [1] |
| Droperidol | Ki | 759.6 [1] |
 | Mizolastine | IC50 | 436.52 [1] |
| Mizolastine | Ki | 7258.0 [1] |
 | N-[4-[2-(6-Cyano-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]cyclohexyl]quinoline-4-carboxamide | IC50 | 630.96 [1], 676.08 [2], 1995.26 [3] |
| N-[4-[2-(6-Cyano-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]cyclohexyl]quinoline-4-carboxamide | Ki | 630.96 [1] |
 | Olanzapine | IC50 | 181.97 [1] |
| Olanzapine | Ki | 36000.0 [1] |
 | Imipramine | IC50 | 3388.44 [1] |
 | Ziprasidone | IC50 | 125.89 [1] |
 | Gatifloxacin | IC50 | 128824.96 [1] |
 | Ciprofloxacin | IC50 | 954992.59 [1] |
| Ciprofloxacin | Ki | 100000.0 [1] |
 | Fluoxetine | IC50 | 10.0 [1], 457.09 [2], 1513.56 [3] |
| Fluoxetine | Ki | 10066.0 [1] |
 | Diltiazem | IC50 | 17378.01 [1] |
 | Desipramine | IC50 | 1380.38 [1] |
| Desipramine | Ki | 22816.6 [1] |
 | Aripiprazole | IC50 | 630.96 [1], 1000.0 [2], 3860.0 [3] |
| Aripiprazole | Ki | 598.0 [1], 1020.0 [2] |
 | Loratadine | IC50 | 169.82 [1], 173.78 [2] |
| Loratadine | Ki | 32022.8 [1] |
 | Azimilide | IC50 | 562.34 [1] |
 | CID 56927659 | IC50 | 1700.0 [1], 1740.0 [2], 3400.0 [3] |
| CID 56927659 | Ki | 1701.0 [1] |
 | Cocaine | IC50 | 5754.4 [1], 7244.36 [2] |
 | Nifedipine | IC50 | 50118.72 [1] |
 | Chloroquine | IC50 | 2500.0 [1], 2511.89 [2] |
| Chloroquine | Ki | 3162.28 [1], 7500.0 [2] |
 | Citalopram | IC50 | 10.0 [1], 3981.07 [2] |
| Citalopram | Ki | 13661.8 [1] |
 | Quinidine | IC50 | 323.59 [1] |
 | Diphenhydramine | IC50 | 2570.4 [1], 5200.0 [2], 26915.35 [3] |
| Diphenhydramine | Ki | 26101.3 [1] |
 | Carvedilol | IC50 | 350.0 [1], 10471.29 [2], 12589.25 [3] |
| Carvedilol | Ki | 3374.9 [1] |
 | Domperidone | IC50 | 57.54 [1], 162.18 [2] |
 | Cetirizine | IC50 | 30199.52 [1] |
 | Perhexiline | IC50 | 7762.47 [1] |
 | Dolasetron | IC50 | 6025.6 [1], 12022.64 [2] |
 | Tecastemizole | IC50 | 27.54 [1], 28.18 [2] |
 | 6-[[[1-[(1S)-2-(3-Fluoro-6-methoxy-1,5-naphthyridin-4-yl)-1-hydroxyethyl]-2-oxabicyclo[2.2.2]octan-4-yl]amino]methyl]-4H-pyrido[3,2-b][1,4]oxazin-3-one | IC50 | 18000.0 [1] |
 | Nicotine | IC50 | 244299.74 [1], 245470.89 [2] |
 | Amiodarone | IC50 | 30.0 [1], 1000.0 [2], 10000.0 [3] |
 | Bupivacaine hydrochloride | IC50 | 22000.0 [1], 32000.0 [2], 95000.0 [3], 265000.0 [4], 866000.0 [5] |
 | Clarithromycin | IC50 | 33113.11 [1], 46000.0 [2], 58884.37 [3] |
 | Ofloxacin | IC50 | 1412537.54 [1], 1420000.0 [2] |
 | Ketoconazole | IC50 | 1900.0 [1], 1905.46 [2] |
 | Sunitinib | IC50 | 251.19 [1], 500.0 [2], 7943.28 [3], 10000.0 [4] |
 | Ondansetron | IC50 | 400.0 [1], 812.83 [2] |
 | Nitrendipine | IC50 | 10000.0 [1] |
 | Chlorpheniramine | IC50 | 1100.0 [1], 20892.96 [2] |
 | Disopyramide | IC50 | 12000.0 [1], 91201.08 [2] |
 | Granisetron | IC50 | 3715.35 [1], 3730.0 [2], 3801.89 [3] |
 | Paliperidone | IC50 | 1000.0 [1], 1258.93 [2], 1288.25 [3], 1300.0 [4] |
 | Levobupivacaine hydrochloride | IC50 | 13000.0 [1], 83000.0 [2], 278000.0 [3], 1013000.0 [4] |
 | Alosetron | IC50 | 2300.0 [1], 3200.0 [2], 3235.94 [3] |
 | Ibutilide | IC50 | 10.0 [1], 15.14 [2], 20.0 [3] |
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