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HERG Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
TerfenadineIC50128.82 [1]
TerfenadineKi56.0 [1], 320.0 [2]
CisaprideIC5039.81 [1]
CisaprideKi139.4 [1]
AstemizoleIC508.0 [1]

References
This online resource may be cited as follows
MLA
"Quest DatabaseHERG Inhibitors (IC50, Ki)." AAT Bioquest, Inc.4 Apr2026https://www.aatbio.com/data-sets/herg-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2026April 4). Quest DatabaseHERG Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/herg-inhibitors-ic50-ki.
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