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Histamine H1 receptor Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
PyrilamineIC501.3 [1], 1.8 [2], 3.0 [3], 12.59 [4], 46.77 [5]
PyrilamineKi5.01e+17 [1]
HistamineIC50158.49 [1], 1000.0 [2]
HistamineKi15848900000000.0 [1]
CetirizineKi14.0 [1]

References
This online resource may be cited as follows
MLA
"Quest DatabaseHistamine H1 receptor Inhibitors (IC50, Ki)." AAT Bioquest, Inc.15 Dec2025https://www.aatbio.com/data-sets/histamine-h1-receptor-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 15). Quest DatabaseHistamine H1 receptor Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/histamine-h1-receptor-inhibitors-ic50-ki.
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