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Histamine H2 receptor Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
CimetidineIC50140.0 [1], 270.0 [2], 781.0 [3], 1000.0 [4]
CimetidineKi70.0 [1], 170.0 [2], 490.0 [3], 5431.0 [4]
HistamineKi5000.0 [1], 50118.72 [2], 25118900000000.0 [3]
BurimamideKi3981.07 [1]
ImmepipKi1000.0 [1], 10000.0 [2]

References
This online resource may be cited as follows
MLA
"Quest DatabaseHistamine H2 receptor Inhibitors (IC50, Ki)." AAT Bioquest, Inc.2 Jan2026https://www.aatbio.com/data-sets/histamine-h2-receptor-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2026January 2). Quest DatabaseHistamine H2 receptor Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/histamine-h2-receptor-inhibitors-ic50-ki.
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