Name: Histamine H3 receptor Inhibitors (IC50, Ki)
Creator: AAT Bioquest
License: https://www.aatbio.com/tou.html

Histamine H3 receptor Inhibitors (IC50, Ki)

Structure	Compound Name	Standard Type	Standard Values (in nM)
	Thioperamide	IC50	16.0 ^[1], 120.0 ^[2], 517.5 ^[3]
	1-[4-(3-Piperidinopropoxy)benzyl]piperidine	IC50	0.53 ^[1]
	(R)-4-(2-(2-(2-Methylpyrrolidin-1-yl)ethyl)benzofuran-5-yl)benzonitrile	IC50	0.63 ^[1]
	Pitolisant	IC50	12.0 ^[1]
	Pitolisant	Ki	0.3 ^[1]
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References

This online resource may be cited as follows

MLA	"Quest Database™ Histamine H3 receptor Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 28 Dec. 2025, https://www.aatbio.com/data-sets/histamine-h3-receptor-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2025, December 28). Quest Database™ Histamine H3 receptor Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/histamine-h3-receptor-inhibitors-ic50-ki.
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