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Histamine H4 receptor Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
1-[(5-Chloro-1H-indol-2-yl)carbonyl]-4-methylpiperazineIC5086.0 [1]
1-[(5-Chloro-1H-indol-2-yl)carbonyl]-4-methylpiperazineKi46.0 [1]
ThioperamideIC50667.0 [1], 680.0 [2], 977.0 [3]
HistamineKi14.45 [1]
(5-Chloro-1H-benzimidazol-2-yl)(4-methylpiperazin-1-yl)methanoneIC50138.0 [1], 530.0 [2]

References
This online resource may be cited as follows
MLA
"Quest DatabaseHistamine H4 receptor Inhibitors (IC50, Ki)." AAT Bioquest, Inc.28 Dec2025https://www.aatbio.com/data-sets/histamine-h4-receptor-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 28). Quest DatabaseHistamine H4 receptor Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/histamine-h4-receptor-inhibitors-ic50-ki.
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