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Histone acetyltransferase GCN5 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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▼
(2R,3S)-4-Methylidene-5-oxo-2-propyloxolane-3-carboxylic acidIC50100000.0 [1]
2-(4-Fluorophenyl)isothiazolo[5,4-b]pyridin-3(2H)-oneIC508390.0 [1], 8400.0 [2]
Butyrolactone 3IC50100000.0 [1]
2-[(4-Chlorophenyl)methyl]-[1,2]thiazolo[5,4-b]pyridin-3-oneIC5089900.0 [1], 89910.0 [2]
4-[(2s,4r)-1-Acetyl-4-[(4-Chlorophenyl)amino]-2-Methyl-1,2,3,4-Tetrahydroquinolin-6-Yl]benzoic AcidIC50316.23 [1]
2-(4-Methylpyrimidin-2-yl)-1,2-benzothiazol-3-oneIC5019900.0 [1]
3-[7-(Difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-N-methyl-1-(oxan-4-yl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-5-carboxamideIC5020000.0 [1]
2-(4-Pyrrolidin-1-ylsulfonylphenyl)-1,2-benzothiazol-3-oneIC506270.0 [1]
2-(1,3-Thiazol-2-yl)-1,2-benzothiazol-3-oneIC507870.0 [1]
Ethyl 4-(3-oxo-1,2-benzisothiazol-2(3H)-yl)benzoateIC508530.0 [1]
2-(1,3-Benzothiazol-2-yl)-1,2-benzothiazol-3-oneIC5023300.0 [1]
4,6-Dimethyl-2-(thiophene-2-carbonyl)-[1,2]thiazolo[5,4-b]pyridin-3-oneIC506130.0 [1]
2-(4-Chlorophenyl)isothiazolo[5,4-b]pyridin-3(2H)-oneIC5015470.0 [1]
CID 118021718IC5080000.0 [1]
4-Bromo-2-methyl-5-[[(3R,5R)-1-methyl-5-phenylpiperidin-3-yl]amino]pyridazin-3-oneKi1.4 [1]
[(3,5-Dimethyl-4-oxocyclohexa-2,5-dien-1-ylidene)amino] 4-methoxybenzenesulfonateIC5033900.0 [1]
Ethyl 2-(4,6-dimethyl-3-oxoisothiazolo[5,4-b]pyridin-2(3H)-yl)acetateIC508370.0 [1]
N-[3-(3-Methyl-4-Oxo-4,5,6,7-Tetrahydro-2h-Isoindol-1-Yl)-4-Phenoxyphenyl]methanesulfonamideIC501000.0 [1]
1-(3-Phenylazanyl-1,4,6,7-Tetrahydropyrazolo[4,3-C]pyridin-5-Yl)ethanoneIC5020000.0 [1]
PRMT5 Inhibitor C17IC50100000.0 [1]
1-[3-[7-(Difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-1-(oxan-4-yl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-5-yl]ethanoneIC5020000.0 [1]
1-[3-[2-Fluoro-4-(1-methylpyrazol-4-yl)anilino]-1-[(3R)-oxolan-3-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-5-yl]ethanoneIC5020000.0 [1]
(2R,3R)-4-Methylidene-5-oxo-3-propyloxolane-2-carboxylic acidIC50100000.0 [1]
5-Nitro-2-(4-phenoxyphenyl)isothiazolo[5,4-b]pyridin-3-oneIC502040.0 [1]
2-(4-Butylphenyl)-5-phenylisothiazolo[5,4-b]pyridin-3(2H)-oneIC508650.0 [1]
2-(3-Oxo-1,2-benzothiazol-2(3H)-yl)-N-(1,3-thiazol-2-yl)acetamideIC5021700.0 [1]
1,2-Benzisothiazole-2(3H)-butanoic acid, 3-oxo-IC5066700.0 [1]
2-[[4-(Trifluoromethyl)phenyl]methyl]-[1,2]thiazolo[5,4-b]pyridin-3-oneIC5087360.0 [1]
2-[(3,4-Dichlorophenyl)methyl]-[1,2]thiazolo[5,4-b]pyridin-3-oneIC5023700.0 [1]
3-[2-(2,4-Difluorophenoxy)-5-methylsulfonylphenyl]-1-methyl-6H-pyrrolo[2,3-c]pyridin-7-oneIC501000.0 [1]
6-[(5Z)-5-[1-[(4-Methylphenyl)methyl]-2-oxoindol-3-ylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]hexanoic acidIC5047000.0 [1]
6-[(5Z)-5-[1-[(4-Fluorophenyl)methyl]-2-oxoindol-3-ylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]hexanoic acidIC50209600.0 [1]
2-(3-Oxo-1,2-benzothiazol-2(3H)-yl)-N-(pyridin-2-ylmethyl)acetamideIC5011200.0 [1]
2-(4-Methyl-1,3-thiazol-2-yl)-1,2-benzothiazol-3-oneIC507110.0 [1]
N-(2-Methoxyethyl)-2-(3-oxo-1,2-benzothiazol-2(3H)-yl)acetamideIC5015500.0 [1]
N-(2-Methylpropyl)-3-(3-oxo-1,2-benzothiazol-2(3H)-yl)propanamideIC5034900.0 [1]
N-(2-Methylpropyl)-2-(3-oxo-1,2-benzothiazol-2(3H)-yl)acetamideIC5020800.0 [1]
6-[(5Z)-5-[1-[(4-Methoxyphenyl)methyl]-2-oxoindol-3-ylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]hexanoic acidIC5054700.0 [1]
6-[(5Z)-5-[1-[(4-Nitrophenyl)methyl]-2-oxoindol-3-ylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]hexanoic acidIC5069600.0 [1]
8-[(5Z)-5-[1-[(4-Methylphenyl)methyl]-2-oxoindol-3-ylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]octanoic acidIC5063500.0 [1]
4-[[(5Z)-5-[1-[(4-Methylphenyl)methyl]-2-oxoindol-3-ylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]methyl]cyclohexane-1-carboxylic acidIC5046400.0 [1]
Items per page: 1 - 10 of 41
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References

This online tool may be cited as follows

MLA

"Quest Database™ Histone acetyltransferase GCN5 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/histone-acetyltransferase-gcn5-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 9). Quest Database™ Histone acetyltransferase GCN5 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/histone-acetyltransferase-gcn5-inhibitors-ic50-ki.
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