logo
AAT Bioquest

Histone acetyltransferase KAT8 Inhibitors (IC50, Ki)

Structure
Compound Name
Standard Type
Standard Values (in nM)
4-Amino-1-naphtholIC501100.0 [1], 1600.0 [2], 1800.0 [3], 9700.0 [4]
4-Amino-1-naphtholKi17.0 [1], 2600.0 [2]
2-(4-Heptylphenethyl)-6-hydroxybenzoic acidIC5015000.0 [1], 27000.0 [2], 47000.0 [3]
PhenylhydrazineIC501000000.0 [1]
1-NaphthylamineIC50181000.0 [1]
Phenylhydrazine hydrochlorideIC501000000.0 [1]
4-AminophenolIC50500000.0 [1]
4-ChloroanilineIC501000000.0 [1]
Anacardic acidIC5043000.0 [1]
4-HydroxyquinolineIC50500000.0 [1]
1-NitronaphthaleneIC501000000.0 [1]
4-FluoroanilineIC501000000.0 [1]
2-Hydroxy-6-((8Z,11Z)-pentadeca-8,11,14-trienyl)benzoic acidIC5043000.0 [1]
4-FluorobenzylamineIC501000000.0 [1]
8-Amino-2-naphthalenesulfonic acidIC50940000.0 [1]
4-Nitro-1-naphtholIC50141000.0 [1]
(4-Fluorophenyl)hydrazineIC50310000.0 [1]
2,8-Bis(5-methyl-2-furyl)pyrido[3,2-g]quinoline-4,6-dicarboxylic acidIC5017000.0 [1]
2-(1-Naphthyl)-N-(2-{[2-oxo-2-(1-pyrrolidinyl)ethyl]sulfanyl}-1,3-benzothiazol-6-yl)acetamideIC5014000.0 [1]
4-[2-(1,3-Benzothiazol-2-yl)vinyl]-N,N-diethylbenzenesulfonamideIC506000.0 [1]
(4-Aminonaphthalen-1-yl)methanolIC50500000.0 [1]
4-(Dimethylamino)naphthalen-1-ol hydrochlorideIC5023000.0 [1]
8-Aminoisoquinolin-5-olIC507600.0 [1]
4-(Aminomethyl)naphthalen-1-ol;hydrochlorideIC50500000.0 [1]
4-Amino-3-methoxynaphthalen-1-olIC50177000.0 [1]
N-(4-Hydroxynaphthalen-1-yl)decanamideIC50250000.0 [1]
N-(4-Hydroxynaphthalen-1-yl)-2-phenylacetamideIC50365000.0 [1]
4-[(E)-2-(5-Chloro-1,3-benzothiazol-2-yl)ethenyl]-N,N-diethylbenzenesulfonamideIC5030000.0 [1]
4-[(E)-2-(5,6-Dimethyl-1,3-benzothiazol-2-yl)ethenyl]-N,N-diethylbenzenesulfonamideIC507700.0 [1]
N,N-Diethyl-4-[(E)-2-(5-fluoro-1,3-benzothiazol-2-yl)ethenyl]benzenesulfonamideIC5040000.0 [1]
N,N-Diethyl-4-[(E)-2-(6-fluoro-1,3-benzothiazol-2-yl)ethenyl]benzenesulfonamideIC506600.0 [1]
4-[(E)-2-(5-Bromo-1,3-benzothiazol-2-yl)ethenyl]-N,N-diethylbenzenesulfonamideIC5030000.0 [1]
N-(5-Ethyl-1,3,4-thiadiazol-2-yl)-3-[3-[(5-ethyl-1,3,4-thiadiazol-2-yl)amino]-3-oxopropyl]sulfanylpropanamideIC5018000.0 [1]
4-Hydroxynaphthalene-1-carboxamideIC50500000.0 [1]
4-Methoxynaphthalen-1-amine hydrochlorideIC5089000.0 [1]
4-(Benzyloxy)naphthalen-1-amineIC50500000.0 [1]
N-(4-Hydroxynaphthalen-1-yl)acetamideIC50500000.0 [1]
N-(4-Hydroxynaphthalen-1-yl)propanamideIC50500000.0 [1]
4-Methoxyphenylhydrazine hydrochlorideIC50680000.0 [1]
2,4-Dichlorophenylhydrazine hydrochlorideIC501000000.0 [1]
2-(7-Methyl-4-oxo-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]triazin-3-yl)-N-naphthalen-1-ylacetamideIC5025000.0 [1]
3-(1-Benzofuran-2-carbonyl)-1-(furan-2-ylmethyl)-4-hydroxy-2-(4-methylphenyl)-2H-pyrrol-5-oneIC5029000.0 [1]
4-Amino-1-naphthalenecarbonitrileIC50500000.0 [1]
7,9-Di(thiophen-2-yl)thieno[2,3-b:4,5-b']dipyridine-2,4-diolIC5023000.0 [1]
Chembl4172065IC5066000.0 [1]
N-(4-Hydroxynaphthalen-1-yl)-4-methylbenzenesulfonamideIC5037000.0 [1]
[({[3-Cyano-4-phenyl-6-(2-thienyl)-2-pyridinyl]sulfanyl}acetyl)amino]acetic acidIC5074000.0 [1]
4-Aminonaphthalen-1-yl acetateIC50500000.0 [1]



References

This online tool may be cited as follows

MLA

"Quest Database™ Histone acetyltransferase KAT8 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.9 May2024https://www.aatbio.com/data-sets/histone-acetyltransferase-kat8-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024May 9). Quest Database™ Histone acetyltransferase KAT8 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/histone-acetyltransferase-kat8-inhibitors-ic50-ki.
BibTeXEndNoteRefMan