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Histone acetyltransferase p300 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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CID 1285941IC506800.0 [1]
CID 1285941Ki400.0 [1]
[[(3R)-4-[[3-[2-[2-[[(5S)-5-Acetamido-6-amino-6-oxohexyl]amino]-2-oxoethyl]sulfanylethylamino]-3-oxopropyl]amino]-3-hydroxy-2,2-dimethyl-4-oxobutoxy]-hydroxyphosphoryl] [(2R,3S,4R,5R)-5-(6-aminopurin-9-yl)-4-hydroxy-3-phosphonooxyoxolan-2-yl]methyl hydrogen phosphateIC503.2 [1], 50.0 [2], 500.0 [3], 980.0 [4]
[[(3R)-4-[[3-[2-[2-[[(5S)-5-Acetamido-6-amino-6-oxohexyl]amino]-2-oxoethyl]sulfanylethylamino]-3-oxopropyl]amino]-3-hydroxy-2,2-dimethyl-4-oxobutoxy]-hydroxyphosphoryl] [(2R,3S,4R,5R)-5-(6-aminopurin-9-yl)-4-hydroxy-3-phosphonooxyoxolan-2-yl]methyl hydrogen phosphateKi19.0 [1]
Anacardic acidIC504150.0 [1], 8500.0 [2]
GarcinolIC501700.0 [1], 6000.0 [2], 7000.0 [3]
GarcinolKi4900.0 [1]
4-[(4E)-4-[[5-(4,5-Dimethyl-2-nitrophenyl)furan-2-yl]methylidene]-3-methyl-5-oxopyrazol-1-yl]benzoic acidIC50320.0 [1], 1600.0 [2], 2400.0 [3]
4-[(4E)-4-[[5-(4,5-Dimethyl-2-nitrophenyl)furan-2-yl]methylidene]-3-methyl-5-oxopyrazol-1-yl]benzoic acidKi400.0 [1]
PlumbaginIC502000.0 [1], 20000.0 [2]
(1E,4Z,6E)-5-Hydroxy-1,7-bis(4-hydroxy-3-methoxyphenyl)hepta-1,4,6-trien-3-oneIC506500.0 [1], 40000.0 [2], 400000.0 [3]
2-Hydroxy-6-((8Z,11Z)-pentadeca-8,11,14-trienyl)benzoic acidIC505000.0 [1], 1000000.0 [2]
Guttiferone EIC50500.0 [1], 7000.0 [2]
[(3,5-Dimethyl-4-oxocyclohexa-2,5-dien-1-ylidene)amino] 4-methoxybenzenesulfonateIC501980.0 [1], 128000.0 [2]
CurcuminIC506500.0 [1], 25000.0 [2]
2-(4-Fluorophenyl)isothiazolo[5,4-b]pyridin-3(2H)-oneIC505350.0 [1], 5400.0 [2]
(-)-Epigallocatechin gallateIC5030000.0 [1]
Coenzyme AIC5045940.0 [1]
4-AminophenolIC50500000.0 [1]
1-(4-(7-(Diethylamino)-4-methyl-2-oxo-2H-chromen-3-yl)phenyl)-1H-pyrrole-2,5-dioneIC50260.0 [1]
CyqualonIC50111000.0 [1]
Sgc-cbp30IC50230.0 [1]
2-[4-[(4-Bromophenyl)sulfonylamino]-1-hydroxynaphthalen-2-yl]sulfanylacetic acidIC50330.0 [1]
CamboginKi3900.0 [1]
4-[(2s,4r)-1-Acetyl-4-[(4-Chlorophenyl)amino]-2-Methyl-1,2,3,4-Tetrahydroquinolin-6-Yl]benzoic AcidIC5031622.78 [1]
J Acid ureaIC50118500.0 [1]
4-Amino-1-naphtholIC501400.0 [1]
2,6-Bis(3,4-dihydroxybenzylidene)cyclohexanoneIC50233000.0 [1]
C.I. Direct Red 23IC5013700.0 [1]
1,7-Bis(3,4-dihydroxyphenyl)-5-hydroxy-1,4,6-heptatriene-3-oneIC5046000.0 [1]
1,1-Dioxido-1-benzothien-3-yl 5-phenyl-1,3,4-oxadiazol-2-yl sulfideIC5011000.0 [1]
CID 72201043IC5058000.0 [1]
CID 12005893IC501800.0 [1]
CID 12006282IC502000.0 [1]
2-(4-Methylpyrimidin-2-yl)-1,2-benzothiazol-3-oneIC5024700.0 [1]
(4R)-4-Methyl-6-[1-methyl-3-(1-methylpyrazol-4-yl)indazol-5-yl]-1,3,4,5-tetrahydro-1,5-benzodiazepin-2-oneIC5051.0 [1]
3-[7-(Difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-N-methyl-1-(oxan-4-yl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-5-carboxamideIC501.2 [1]
4-[({3-[(Carboxymethyl)thio]-4-hydroxy-1-naphthyl}amino)sulfonyl]benzoic acidIC50660.0 [1]
2-(4-Pyrrolidin-1-ylsulfonylphenyl)-1,2-benzothiazol-3-oneIC508030.0 [1]
2-(1,3-Thiazol-2-yl)-1,2-benzothiazol-3-oneIC509350.0 [1]
Ethyl 4-(3-oxo-1,2-benzisothiazol-2(3H)-yl)benzoateIC5012900.0 [1]
N-[4-Hydroxy-3-(1H-1,2,4-triazol-5-ylsulfanyl)naphthalen-1-yl]naphthalene-2-sulfonamideIC50510.0 [1]
CtpbIC50275000.0 [1]
4,6-Dimethyl-2-(thiophene-2-carbonyl)-[1,2]thiazolo[5,4-b]pyridin-3-oneIC506740.0 [1]
4-Nitro-1-naphtholIC50106000.0 [1]
5-[(1,1-Dioxido-1-benzothiophen-3-yl)sulfanyl]-1-phenyl-1H-tetrazoleIC506200.0 [1]
(2S,5S,7R,9R,13R,14R)-13-[(2R,5R)-5,6-Dimethylheptan-2-yl]-5-hydroxy-2,14-dimethyl-6-methylidenetetracyclo[7.7.1.02,7.014,17]heptadec-1(17)-en-10-oneIC503300.0 [1]
2-(4-Chlorophenyl)isothiazolo[5,4-b]pyridin-3(2H)-oneIC505710.0 [1]
2-Phenylisothiazol-3(2H)-oneIC5023000.0 [1]
N-[(4-Fluorophenyl)methyl]-2-[(3R)-6-(methylcarbamoylamino)-2',4'-dioxospiro[1,2-dihydroindene-3,5'-1,3-oxazolidine]-3'-yl]-N-[(2S)-1,1,1-trifluoropropan-2-yl]acetamideIC5060.0 [1]
N-{4-Hydroxy-3-[(1-phenyl-1H-tetrazol-5-yl)sulfanyl]naphthalen-1-yl}benzenesulfonamideIC503100.0 [1]
6-Hydroxy-5-[(Z)-indol-3-ylidenemethyl]-1-methyl-2-sulfanylidenepyrimidin-4-oneIC5050000.0 [1]
1,7-Bis(3-bromo-4-hydroxyphenyl)-5-hydroxy-1,4,6-heptatriene-3-oneIC5033000.0 [1]
Histone Acetyltransferase Inhibitor IIIC505000.0 [1]
4-Bromo-N-[4-hydroxy-3-(1H-1,2,4-triazol-5-ylsulfanyl)naphthalen-1-yl]benzenesulfonamideIC501100.0 [1]
6-[(7-Bromo-5-nitro-2,1,3-benzothiadiazol-4-yl)thio]-9H-purineIC502200.0 [1]
3-[(5-Pyridin-4-yl-1,3,4-oxadiazol-2-yl)sulfanyl]-1-benzothiophene 1,1-dioxideIC506200.0 [1]
2-(2-Pyridyl)-isothiazol-3(2H)-oneIC5028000.0 [1]
(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[2-[[2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-2-Acetamidopropanoyl]amino]-5-carbamimidamidopentanoyl]amino]-3-hydroxybutanoyl]amino]-6-aminohexanoyl]amino]-5-amino-5-oxopentanoyl]amino]-3-hydroxybutanoyl]amino]propanoyl]amino]-5-carbamimidamidopentanoyl]amino]-6-aminohexanoyl]amino]-3-hydroxypropanoyl]amino]-3-hydroxybutanoyl]amino]acetyl]amino]acetyl]amino]-6-[[2-[2-[3-[[(2R)-4-[[[(2R,3S,4R,5R)-5-(6-aminopurin-9-yl)-4-hydroxy-3-phosphonooxyoxolan-2-yl]methoxy-hydroxyphosphoryl]oxy-hydroxyphosphoryl]oxy-2-hydroxy-3,3-dimethylbutanoyl]amino]propanoylamino]ethylsulfanyl]acetyl]amino]hexanoyl]amino]propanoyl]pyrrolidine-2-carbonyl]amino]-5-carbamimidamidopentanoyl]amino]-6-aminohexanoyl]amino]-5-amino-5-oxopentanoyl]amino]-4-methylpentanoic acidIC507540.0 [1]
(1S,3S,9R,11R)-7-(4-Hydroxy-3-methoxybenzoyl)-4,4,10,10-tetramethyl-3,9,11-tris(3-methylbut-2-enyl)-5-oxatricyclo[7.3.1.01,6]tridec-6-ene-8,13-dioneIC505000.0 [1]
1-(4-Methylphenyl)-3-[(4-phenyl-1,2,4-triazol-3-yl)sulfanyl]pyrrolidine-2,5-dioneIC509800.0 [1]
1,3-Dibenzyl-5-[(4-hydroxyphenyl)methylidene]-1,3-diazinane-2,4,6-trioneIC502100.0 [1]
1,3-Dibenzyl-5-[(3,4-dihydroxyphenyl)methylidene]-1,3-diazinane-2,4,6-trioneIC501600.0 [1]
1,3-Dibenzyl-5-[(3-hydroxy-4-methoxyphenyl)methylidene]-1,3-diazinane-2,4,6-trioneIC505900.0 [1]
1,3-Dibenzyl-5-[(4-hydroxy-3-methoxyphenyl)methylidene]-1,3-diazinane-2,4,6-trioneIC501500.0 [1]
1,3-Dibenzyl-5-[(3,4-dimethoxyphenyl)methylidene]-1,3-diazinane-2,4,6-trioneIC5011400.0 [1]
1,3-Dibenzyl-5-[(4-methoxyphenyl)methylidene]-1,3-diazinane-2,4,6-trioneIC508000.0 [1]
5-[(4-Hydroxyphenyl)methylidene]-1,3-bis(2-methylpropyl)-1,3-diazinane-2,4,6-trioneIC508500.0 [1]
5-[(3,4-Dihydroxyphenyl)methylidene]-1,3-bis(2-methylpropyl)-1,3-diazinane-2,4,6-trioneIC505400.0 [1]
5-[(3-Hydroxy-4-methoxyphenyl)methylidene]-1,3-bis(2-methylpropyl)-1,3-diazinane-2,4,6-trioneIC5031400.0 [1]
5-[(4-Hydroxy-3-methoxyphenyl)methylidene]-1,3-bis(2-methylpropyl)-1,3-diazinane-2,4,6-trioneIC504200.0 [1]
5-[(4-Hydroxy-3-methoxyphenyl)methylidene]-1,3-bis(prop-2-enyl)-1,3-diazinane-2,4,6-trioneIC5026400.0 [1]
4-[(4Z)-4-[2-[5-[(4,5-Dimethyl-2-nitrophenyl)methyl]furan-2-yl]ethylidene]-3-methyl-5-oxopyrazol-1-yl]benzoic acidIC501600.0 [1]
1-[3-[7-(Difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-1-(oxan-4-yl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-5-yl]ethanoneIC501.3 [1]
1-[3-[2-Fluoro-4-(1-methylpyrazol-4-yl)anilino]-1-[(3R)-oxolan-3-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-5-yl]ethanoneIC5030.0 [1]
(5E)-5-Benzylidene-1-methyl-2-sulfanylidene-1,3-diazinane-4,6-dioneIC5045000.0 [1]
4-(Dimethylamino)naphthalen-1-ol hydrochlorideIC503700.0 [1]
(1S,3E,5R,7S)-3-[(3,4-Dihydroxyphenyl)-hydroxymethylidene]-6,6-dimethyl-7-[(Z)-3-methylbut-1-enyl]-5-(3-methylbut-2-enyl)-1-[(E,2R)-5-methyl-2-prop-1-en-2-ylhex-3-enyl]bicyclo[3.3.1]nonane-2,4,9-trioneIC507000.0 [1]
(1S,3S,9R,11S)-7-(3-Hydroxy-4-methoxybenzoyl)-4,4,10,10-tetramethyl-11-[(Z)-3-methylbut-1-enyl]-3,9-bis(3-methylbut-2-enyl)-5-oxatricyclo[7.3.1.01,6]tridec-6-ene-8,13-dioneIC505000.0 [1]
(2S)-2-[2-[[(1S)-1-Carboxy-3-[5-[(Z)-[(5S)-5-[3-(diaminomethylideneamino)propyl]-3,6-dioxopiperazin-2-ylidene]methyl]-2-hydroxyphenoxy]propyl]amino]-2-oxoethyl]-2-hydroxybutanedioic acidIC5022.0 [1]
4-[(4Z)-4-[[5-(4,5-Dimethyl-2-nitrophenyl)furan-2-yl]methylidene]-3-methyl-5-oxopyrazol-1-yl]-N-prop-2-ynylbenzamideIC5014100.0 [1]
2-[(4-Chlorophenyl)methyl]-[1,2]thiazolo[5,4-b]pyridin-3-oneIC505740.0 [1]
8-Aminoisoquinolin-5-olIC501100.0 [1]
4-Bromo-N-(3-chloro-4-hydroxynaphthalen-1-yl)benzenesulfonamideIC501800.0 [1]
N-Methyl-2,3-diphenyl-1,2,4-thiadiazol-2-ium-5-amine;chlorideIC501900.0 [1]
3-[(1-Acetyl-5-methoxyindole-3-carbonyl)amino]-5-(furan-2-yl)benzoic acidIC501780.0 [1]
3-[(1-Acetyl-5-methoxyindole-3-carbonyl)amino]-4-fluoro-5-(1-methylpyrazol-4-yl)benzoic acidIC5049.0 [1]
CID 145948689IC50200000.0 [1]
3-[(1-Acetylindole-3-carbonyl)amino]-4-fluorobenzoic acidIC504450.0 [1]
3-[(1-Acetylindole-3-carbonyl)amino]benzoic acidIC505550.0 [1]
(1S,2S,5S,7S,9R,13R,14R,18S)-13-[(2R,5R)-5,6-Dimethylheptan-2-yl]-5-hydroxy-2,14-dimethyl-6-methylidene-17-oxapentacyclo[7.7.2.01,18.02,7.014,18]octadecan-10-oneIC508800.0 [1]
3-[(1-Acetylindole-3-carbonyl)amino]-5-(oxan-2-yloxymethyl)benzoic acidIC502510.0 [1]
4-Amino-3-methoxynaphthalen-1-olIC5052000.0 [1]
(1R,2R,5S,7R,13R,14R)-13-[(2R,5R)-5,6-Dimethylheptan-2-yl]-5-hydroxy-2,14-dimethyl-6-methylidenetetracyclo[7.7.1.02,7.014,17]heptadec-9(17)-en-10-oneIC5010000.0 [1]
(1S,2S,5S,7S,9R,13R,14R,18R)-13-[(2R,5R)-5,6-Dimethylheptan-2-yl]-5,9-dihydroxy-2,14-dimethyl-6-methylidene-17-oxapentacyclo[7.7.2.01,18.02,7.014,18]octadecan-10-oneIC5010000.0 [1]
N-(4-Hydroxynaphthalen-1-yl)decanamideIC5060000.0 [1]
3-[(1-Acetyl-5-methoxyindole-3-carbonyl)amino]-5-(1-methylpyrazol-4-yl)benzoic acidIC50510.0 [1]
N-(4-Hydroxynaphthalen-1-yl)-2-phenylacetamideIC50250000.0 [1]
3-[(1-Acetylindole-3-carbonyl)amino]-5-(furan-2-yl)benzoic acidIC50970.0 [1]
(1S,2R,5R,6S,9S,11R,13R,17S)-17-[(2R,5R)-5,6-Dimethylheptan-2-yl]-9-hydroxy-2,6-dimethyl-10-methylidene-18-oxapentacyclo[11.5.0.01,5.02,17.06,11]octadecan-14-oneIC5010000.0 [1]
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References

This online tool may be cited as follows

MLA

"Quest Database™ Histone acetyltransferase p300 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/histone-acetyltransferase-p300-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 9). Quest Database™ Histone acetyltransferase p300 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/histone-acetyltransferase-p300-inhibitors-ic50-ki.
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