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Histone acetyltransferase PCAF Inhibitors (IC50, Ki)

Structure
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▼
Compound Name
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▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
Anacardic acidIC505000.0 [1], 33900.0 [2]
N-(3-Aminopropyl)-4-methyl-2-nitrobenzenamineIC501600.0 [1]
2-(4-Fluorophenyl)isothiazolo[5,4-b]pyridin-3(2H)-oneIC50720.0 [1], 1640.0 [2], 9700.0 [3], 9740.0 [4]
2-Hydroxy-6-((8Z,11Z)-pentadeca-8,11,14-trienyl)benzoic acidIC508500.0 [1], 667050.0 [2], 1000000.0 [3]
4-Bromo-2-methyl-5-[[(3R,5R)-1-methyl-5-phenylpiperidin-3-yl]amino]pyridazin-3-oneIC5039.81 [1], 60.0 [2]
4-Bromo-2-methyl-5-[[(3R,5R)-1-methyl-5-phenylpiperidin-3-yl]amino]pyridazin-3-oneKi1.4 [1]
2-[[4-(Trifluoromethyl)phenyl]methyl]-[1,2]thiazolo[5,4-b]pyridin-3-oneIC5025500.0 [1], 130000.0 [2]
GarcinolIC505000.0 [1], 6000.0 [2]
2-Phenyl-isothiazolo[5,4-b]pyridin-3-oneIC506100.0 [1], 7850.0 [2]
[[(3R)-4-[[3-[2-[2-[[(5S)-5-Acetamido-6-amino-6-oxohexyl]amino]-2-oxoethyl]sulfanylethylamino]-3-oxopropyl]amino]-3-hydroxy-2,2-dimethyl-4-oxobutoxy]-hydroxyphosphoryl] [(2R,3S,4R,5R)-5-(6-aminopurin-9-yl)-4-hydroxy-3-phosphonooxyoxolan-2-yl]methyl hydrogen phosphateIC50108300.0 [1], 200000.0 [2]
5-Chloro-2-ethylisothiazol-3(2H)-oneIC503000.0 [1]
2-(4-Chlorophenyl)isothiazolo[5,4-b]pyridin-3(2H)-oneIC503530.0 [1]
4-Bromo-2-methyl-5-[[(3S,5S)-1-methyl-5-phenylpiperidin-3-yl]amino]pyridazin-3-oneIC5010000.0 [1], 12589.25 [2]
2-(4-Nitrophenyl)isothiazolo[5,4-b]pyridin-3-oneIC502990.0 [1], 4100.0 [2]
Methyl 3-(5-chloro-3-oxoisothiazol-2(3H)-yl)propanoateIC501800.0 [1]
Methyl 3-(5-chloro-1-oxido-3-oxoisothiazol-2(3H)-yl)propanoateIC505600.0 [1]
(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[2-[[2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-2-Acetamidopropanoyl]amino]-5-carbamimidamidopentanoyl]amino]-3-hydroxybutanoyl]amino]-6-aminohexanoyl]amino]-5-amino-5-oxopentanoyl]amino]-3-hydroxybutanoyl]amino]propanoyl]amino]-5-carbamimidamidopentanoyl]amino]-6-aminohexanoyl]amino]-3-hydroxypropanoyl]amino]-3-hydroxybutanoyl]amino]acetyl]amino]acetyl]amino]-6-[[2-[2-[3-[[(2R)-4-[[[(2R,3S,4R,5R)-5-(6-aminopurin-9-yl)-4-hydroxy-3-phosphonooxyoxolan-2-yl]methoxy-hydroxyphosphoryl]oxy-hydroxyphosphoryl]oxy-2-hydroxy-3,3-dimethylbutanoyl]amino]propanoylamino]ethylsulfanyl]acetyl]amino]hexanoyl]amino]propanoyl]pyrrolidine-2-carbonyl]amino]-5-carbamimidamidopentanoyl]amino]-6-aminohexanoyl]amino]-5-amino-5-oxopentanoyl]amino]-4-methylpentanoic acidIC50300.0 [1], 2270.0 [2]
4-Chloro-2-methyl-5-[[(3R,5S)-1-methyl-5-(2-methylpropyl)piperidin-3-yl]amino]pyridazin-3-oneIC5013.0 [1]
2-[(4-Chlorophenyl)methyl]-[1,2]thiazolo[5,4-b]pyridin-3-oneIC5017450.0 [1], 17500.0 [2]
6-[[(1S,2S)-1-[4-(Benzenesulfonyl)phenyl]-1-(dimethylamino)propan-2-yl]amino]-2,4-dimethyl-1,2,4-triazine-3,5-dioneIC5070.0 [1]
N-(3-Aminopropyl)-2-nitrobenzenamineIC505000.0 [1], 5600.0 [2]
2-(4-Bromophenyl)-5-nitro-isothiazolo[5,4-b]pyridin-3-oneIC50860.0 [1], 4910.0 [2]
5-Nitro-2-(4-nitrophenyl)isothiazolo[5,4-b]pyridin-3-oneIC5011800.0 [1], 15800.0 [2]
2-(4-Methoxyphenyl)-5-nitro-isothiazolo[5,4-b]pyridin-3-oneIC501830.0 [1], 3420.0 [2]
2-(4-Nitrophenyl)-5-methylisothiazolo[5,4-b]pyridin-3(2H)-oneIC502720.0 [1], 15300.0 [2]
2-[(3,4-Dichlorophenyl)methyl]-[1,2]thiazolo[5,4-b]pyridin-3-oneIC506940.0 [1]
2-Benzyl-6-nitro-1,2-benzothiazol-3-oneIC507660.0 [1], 51300.0 [2]
N'-[[6-(3-Aminopropylimino)-1-hydroxypyridin-3-yl]methyl]propane-1,3-diamineIC50900.0 [1], 930.0 [2]
[[(3S)-4-[[3-[2-[[1-[(5S)-5-[[2-[[2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-Acetamidopropanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-6-aminohexanoyl]amino]-3-phosphonooxypropanoyl]amino]-3-hydroxybutanoyl]amino]acetyl]amino]acetyl]amino]-6-[[(2S)-1-[(2S)-2-[[(2S)-5-(diaminomethylideneamino)-1-[[(2S)-1,6-diamino-1-oxohexan-2-yl]amino]-1-oxopentan-2-yl]carbamoyl]pyrrolidin-1-yl]-1-oxopropan-2-yl]amino]-6-oxohexyl]triazol-4-yl]methylsulfanyl]ethylamino]-3-oxopropyl]amino]-3-hydroxy-2,2-dimethyl-4-oxobutoxy]-hydroxyphosphoryl] [(2R,3S,4R,5R)-5-(6-aminopurin-9-yl)-4-hydroxy-3-phosphonooxyoxolan-2-yl]methyl hydrogen phosphateIC501700.0 [1], 33000.0 [2]
[[(3S)-4-[[3-[2-[[1-[(5S)-5-[[2-[[2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-Acetamidopropanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-6-aminohexanoyl]amino]-3-hydroxypropanoyl]amino]-3-hydroxybutanoyl]amino]acetyl]amino]acetyl]amino]-6-[[(2S)-1-[(2S)-2-[[(2S)-5-(diaminomethylideneamino)-1-[[(2S)-1,6-diamino-1-oxohexan-2-yl]amino]-1-oxopentan-2-yl]carbamoyl]pyrrolidin-1-yl]-1-oxopropan-2-yl]amino]-6-oxohexyl]triazol-4-yl]methylsulfanyl]ethylamino]-3-oxopropyl]amino]-3-hydroxy-2,2-dimethyl-4-oxobutoxy]-hydroxyphosphoryl] [(2R,3S,4R,5R)-5-(6-aminopurin-9-yl)-4-hydroxy-3-phosphonooxyoxolan-2-yl]methyl hydrogen phosphateIC502800.0 [1], 117000.0 [2]
(-)-Epigallocatechin gallateIC5060000.0 [1]
Coenzyme AIC5041910.0 [1]
PlumbaginIC5050000.0 [1]
4-AminophenolIC50500000.0 [1]
EmbelinIC507200.0 [1]
1-Methyl-2-quinoloneIC5070000.0 [1]
Sgc-cbp30IC5020000.0 [1]
4-[(2s,4r)-1-Acetyl-4-[(4-Chlorophenyl)amino]-2-Methyl-1,2,3,4-Tetrahydroquinolin-6-Yl]benzoic AcidIC507943.28 [1]
Guttiferone EIC505000.0 [1]
4-Amino-1-naphtholIC503600.0 [1]
CID 72201043IC5035000.0 [1]
4-[(2-Amino-4-hydroxy-5-methylphenyl)diazenyl]-N-pyridin-2-ylbenzenesulfonamideKi5520.0 [1]
2-(4-Methylpyrimidin-2-yl)-1,2-benzothiazol-3-oneIC5013600.0 [1]
3-[7-(Difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-N-methyl-1-(oxan-4-yl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-5-carboxamideIC5020000.0 [1]
2-(4-Pyrrolidin-1-ylsulfonylphenyl)-1,2-benzothiazol-3-oneIC506190.0 [1]
2-(1,3-Thiazol-2-yl)-1,2-benzothiazol-3-oneIC505770.0 [1]
Ethyl 4-(3-oxo-1,2-benzisothiazol-2(3H)-yl)benzoateIC506950.0 [1]
2-(1,3-Benzothiazol-2-yl)-1,2-benzothiazol-3-oneIC504550.0 [1]
4,6-Dimethyl-2-(thiophene-2-carbonyl)-[1,2]thiazolo[5,4-b]pyridin-3-oneIC509300.0 [1]
4-Nitro-1-naphtholIC50221000.0 [1]
2-(3-Chloro-4-fluorophenyl)-3(2H)-isothiazoloneIC504200.0 [1]
2-(3-Chloro-2-fluorophenyl)-3(2H)-isothiazoloneIC505400.0 [1]
2-(3-Methoxyphenyl)isothiazolo[5,4-b]pyridin-3(2H)-oneIC505030.0 [1]
2-Phenylisothiazol-3(2H)-oneIC5028000.0 [1]
4-[(2-Amino-3-chloro-4-hydroxy-5-methylphenyl)diazenyl]-N-pyridin-2-ylbenzenesulfonamideKi3340.0 [1]
4-Cyano-N-(1,3-diethyl-2-oxoquinolin-6-yl)benzenesulfonamideIC50100000.0 [1]
[(3,5-Dimethyl-4-oxocyclohexa-2,5-dien-1-ylidene)amino] 4-methoxybenzenesulfonateIC5034700.0 [1]
2-(4-Bromophenyl)isothiazolo[5,4-b]pyridin-3(2H)-oneIC504430.0 [1]
2-(4-Methoxyphenyl)isothiazolo[5,4-b]pyridin-3(2H)-oneIC505710.0 [1]
2-(2-Pyridyl)-isothiazol-3(2H)-oneIC5019000.0 [1]
Ethyl 2-(4,6-dimethyl-3-oxoisothiazolo[5,4-b]pyridin-2(3H)-yl)acetateIC5013600.0 [1]
(Z)-2-Hydroxy-6-(4-(pentyloxy)styryl)benzoic acidIC50662000.0 [1]
Isothiazolo[5,4-b]pyridin-3(2H)-one, 2-(phenylmethyl)-IC5022960.0 [1]
N-[3-(3-Methyl-4-Oxo-4,5,6,7-Tetrahydro-2h-Isoindol-1-Yl)-4-Phenoxyphenyl]methanesulfonamideIC501000.0 [1]
1-(3-Phenylazanyl-1,4,6,7-Tetrahydropyrazolo[4,3-C]pyridin-5-Yl)ethanoneIC5020000.0 [1]
2-Ethylisothiazol-3(2H)-oneIC5010000.0 [1]
4-Chloro-2-methyl-5-(methylamino)pyridazin-3(2H)-oneIC5019952.62 [1]
2-[4-(Dimethylamino)phenyl]-1,2-thiazol-3-oneIC505400.0 [1]
4-Chloro-2-methyl-5-[(1-methylpiperidin-4-yl)amino]pyridazin-3-oneIC5015848.93 [1]
4-Chloro-2-methyl-5-[(4-methyl-1,3-thiazol-5-yl)methylamino]pyridazin-3-oneIC507943.28 [1]
4-Chloro-2-methyl-5-(propan-2-ylamino)pyridazin-3-oneIC5031622.78 [1]
4-Chloro-2-methyl-5-[(1-methylpiperidin-3-yl)amino]pyridazin-3-oneIC501258.93 [1]
4-Chloro-2-methyl-5-[(1-methylpyrrolidin-3-yl)amino]pyridazin-3-oneIC5015848.93 [1]
8-[[(1R,2R)-1-(Dimethylamino)-1-phenylpropan-2-yl]amino]-6-methylpyrido[2,3-d]pyridazin-5-oneIC5019.0 [1]
1-[3-[7-(Difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-1-(oxan-4-yl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-5-yl]ethanoneIC5020000.0 [1]
1-[3-[2-Fluoro-4-(1-methylpyrazol-4-yl)anilino]-1-[(3R)-oxolan-3-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-5-yl]ethanoneIC5020000.0 [1]
4-Chloro-2-methyl-5-[[(3S)-1-methylpiperidin-3-yl]amino]pyridazin-3-oneIC506309.57 [1]
4-Chloro-2-methyl-5-[[(3R)-1-methylpiperidin-3-yl]amino]pyridazin-3-oneIC50501.19 [1]
4-(Dimethylamino)naphthalen-1-ol hydrochlorideIC504200.0 [1]
(1S,3E,5R,7S)-3-[(3,4-Dihydroxyphenyl)-hydroxymethylidene]-6,6-dimethyl-7-[(Z)-3-methylbut-1-enyl]-5-(3-methylbut-2-enyl)-1-[(E,2R)-5-methyl-2-prop-1-en-2-ylhex-3-enyl]bicyclo[3.3.1]nonane-2,4,9-trioneIC505000.0 [1]
4,5-Dichloro-2-ethylisothiazol-3(2H)-oneIC502400.0 [1]
Methyl 3-(3-Oxo-2-isothiazolyl)propanoateIC5010000.0 [1]
2-Pentylisothiazol-3(2H)-oneIC5010000.0 [1]
5-(N-Benzylamino)-4-chloro-2-methyl-3(2H)-pyridazinoneIC5012589.25 [1]
4-Chloro-2-methyl-5-[(2-methyl-3,4-dihydro-1H-isoquinolin-5-yl)amino]pyridazin-3-oneIC50316.23 [1]
8-Aminoisoquinolin-5-olIC507100.0 [1]
2-p-Tolylisothiazolo[5,4-b]pyridine-3(2H)-oneIC504630.0 [1]
4-[(E)-(2-Amino-4-Hydroxy-3,5-Dimethylphenyl)diazenyl]-N-(Pyridin-2-Yl)benzenesulfonamideKi3340.0 [1]
5-Anilino-4-chloro-2-methylpyridazin-3-oneIC5010000.0 [1]
4-Chloro-2-methyl-5-[[(3S,5S)-1-methyl-5-phenylpiperidin-3-yl]amino]pyridazin-3-oneIC5025118.86 [1]
4-Chloro-2-methyl-5-[[(3R,5R)-1-methyl-5-phenylpiperidin-3-yl]amino]pyridazin-3-oneIC5079.43 [1]
4-Chloro-2-methyl-5-[[(3R,5S)-1-methyl-5-phenylpiperidin-3-yl]amino]pyridazin-3-oneIC5039810.72 [1]
4-Chloro-2-methyl-5-(3-methylanilino)pyridazin-3-oneIC506309.57 [1]
5-[2-(Aminomethyl)anilino]-4-chloro-2-methylpyridazin-3-oneIC501000.0 [1]
3-[(1-Acetyl-5-methoxyindole-3-carbonyl)amino]-5-(furan-2-yl)benzoic acidIC5020000.0 [1]
3-[(1-Acetyl-5-methoxyindole-3-carbonyl)amino]-4-fluoro-5-(1-methylpyrazol-4-yl)benzoic acidIC5020000.0 [1]
CID 145948689IC50300.0 [1]
3-[(1-Acetylindole-3-carbonyl)amino]-4-fluorobenzoic acidIC5020000.0 [1]
3-[(1-Acetylindole-3-carbonyl)amino]benzoic acidIC5020000.0 [1]
3-[(1-Acetylindole-3-carbonyl)amino]-5-(oxan-2-yloxymethyl)benzoic acidIC5020000.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Histone acetyltransferase PCAF Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/histone-acetyltransferase-pcaf-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 9). Quest Database™ Histone acetyltransferase PCAF Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/histone-acetyltransferase-pcaf-inhibitors-ic50-ki.
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