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Histone acetyltransferase PCAF Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
Anacardic acidIC505000.0 [1], 33900.0 [2]
N-(3-Aminopropyl)-4-methyl-2-nitrobenzenamineIC501600.0 [1]
2-(4-Fluorophenyl)isothiazolo[5,4-b]pyridin-3(2H)-oneIC50720.0 [1], 1640.0 [2], 9700.0 [3], 9740.0 [4]
2-Hydroxy-6-((8Z,11Z)-pentadeca-8,11,14-trienyl)benzoic acidIC508500.0 [1], 667050.0 [2], 1000000.0 [3]
4-Bromo-2-methyl-5-[[(3R,5R)-1-methyl-5-phenylpiperidin-3-yl]amino]pyridazin-3-oneIC5039.81 [1], 60.0 [2]

References
This online resource may be cited as follows
MLA
"Quest DatabaseHistone acetyltransferase PCAF Inhibitors (IC50, Ki)." AAT Bioquest, Inc.15 Dec2025https://www.aatbio.com/data-sets/histone-acetyltransferase-pcaf-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 15). Quest DatabaseHistone acetyltransferase PCAF Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/histone-acetyltransferase-pcaf-inhibitors-ic50-ki.
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