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Histone-arginine methyltransferase CARM1 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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2-{4-[3-Fluoro-2-(2-Methoxyphenyl)-1h-Indol-5-Yl] Piperidin-1-Yl}-N-MethylethanamineIC5030.0 [1]
S-Adenosyl-L-homocysteineKi400.0 [1], 860.0 [2]
N,N,N'-TrimethylethylenediamineIC503000.0 [1]
(2S)-2-Amino-4-[[(2S,3S,4R,5R)-3,4-dihydroxy-5-[6-(methylamino)purin-9-yl]oxolan-2-yl]methylsulfanyl]butanoic acidKi20000.0 [1], 100000.0 [2]
5'-[(3-{[(4-Tert-Butylphenyl)carbamoyl]amino}propyl)(Propan-2-Yl)amino]-5'-DeoxyadenosineKi50000.0 [1], 100000.0 [2]
BMS pyrazole inhibitor 7fIC500.04 [1], 40.0 [2]
2-[3-[[[(2S)-2-Aminopropanoyl]amino]methyl]phenyl]-N-benzyl-5-(trifluoromethyl)pyrazole-3-carboxamideIC5080.0 [1]
2-(4-Benzylpiperidin-1-yl)ethanamineIC501000.0 [1]
N-Methyl-2-(4-methylpiperidin-1-yl)ethanamineIC50200.0 [1]
2-[3-[[(2-Aminoacetyl)amino]methyl]phenyl]-N-[4-(2-methylsulfonylphenyl)phenyl]-5-(trifluoromethyl)pyrazole-3-carboxamideIC501800.0 [1]
(2R)-2-Amino-N-ethylpropanamideIC50105000.0 [1]
Ellagic acidIC5025000.0 [1]
StilbamidineIC50400000.0 [1]
FuramidineIC50400000.0 [1]
CID 71268957IC50128000.0 [1]
5-[5-(4-Carbamimidoylphenyl)furan-2-yl]pyridine-2-carboximidamideIC50400000.0 [1]
Carm1-IN-1IC508600.0 [1]
Benzo[d]imidazole inhibitors of PRMT4 from BMSIC500.07 [1]
CID 53868701IC5034.0 [1]
(2S)-2-Amino-5-[[(2R,3S,4R,5R)-3,4-dihydroxy-5-[6-(methylamino)purin-9-yl]oxolan-2-yl]methyl-(2-iodoethyl)amino]pentanoic acidIC50100000.0 [1]
1-(4-Tert-butylphenyl)-3-[3-[[(2R,3S,4R,5R)-3,4-dihydroxy-5-[6-(methylamino)purin-9-yl]oxolan-2-yl]methyl-propan-2-ylamino]propyl]ureaKi100000.0 [1]
1-[3-[[(3R,4S,5R)-3-(6-Aminopurin-9-yl)-4,5-dihydroxycyclopenten-1-yl]methyl-propan-2-ylamino]propyl]-3-(4-tert-butylphenyl)ureaKi50000.0 [1]
1-[3-[[(1R,2R,3S,4R)-4-(6-Aminopurin-9-yl)-2,3-dihydroxycyclopentyl]methyl-propan-2-ylamino]propyl]-3-(4-tert-butylphenyl)ureaKi50000.0 [1]
1-[3-[[(1S,2R,3S,4R)-4-(6-Aminopurin-9-yl)-2,3-dihydroxycyclopentyl]methyl-propan-2-ylamino]propyl]-3-(4-tert-butylphenyl)ureaKi50000.0 [1]
MS023IC504.0 [1]
PRMT5 Inhibitor C17IC50100000.0 [1]
2-(4-(2-(2-Methoxypyridin-3-yl)-1H-benzo[d]imidazol-5-yl)piperidin-1-yl)-N-methylethanamineIC501.2 [1]
2-Hydroxy-5-{[4-(4-methoxy-3-methylphenyl)-1,3-thiazol-2-yl]amino}benzoic acidIC50100000.0 [1]
4-[[6-(4-Cyanoanilino)-5-nitropyrimidin-4-yl]amino]benzenecarboximidamideIC5010000.0 [1]
(2R)-2-Amino-N-[[3-[5-[5-(1H-indol-4-yl)-1,3,4-oxadiazol-2-yl]-3-(trifluoromethyl)pyrazol-1-yl]phenyl]methyl]propanamideIC5027.0 [1]
N-Methyl-2-(4-phenoxypiperidin-1-yl)ethanamineIC50149.0 [1]
N-Methyl-2-(4-phenylsulfanylpiperidin-1-yl)ethanamineIC503680.0 [1]
[1-[2-(Methylamino)ethyl]piperidin-4-yl] benzoateIC50177.0 [1]
N-Methyl-2-[4-[[4-(2-methylbutan-2-yl)phenyl]methoxy]piperidin-1-yl]ethanamineIC5016.0 [1]
2-[4-[(2-Bromophenyl)methoxy]piperidin-1-yl]-N-methylethanamineIC5014.0 [1]
1-[2-(Methylamino)ethyl]-N-phenylpiperidine-4-carboxamideIC501540.0 [1]
N-Methyl-2-[4-[[4-(2-methylpropyl)phenyl]methoxy]piperidin-1-yl]ethanamineIC5085.0 [1]
N-Methyl-2-[4-(2-phenylethyl)piperidin-1-yl]ethanamineIC50108.0 [1]
N-Methyl-2-[4-[[4-(trifluoromethyl)phenyl]methoxy]piperidin-1-yl]ethanamineIC5062.0 [1]
N-Methyl-2-[4-[[4-(trifluoromethoxy)phenyl]methoxy]piperidin-1-yl]ethanamineIC5028.0 [1]
N-Methyl-2-[4-[[4-(2,2,2-trifluoroethoxy)phenyl]methoxy]piperidin-1-yl]ethanamineIC5053.0 [1]
2-[4-[(2-Fluorophenyl)methoxy]piperidin-1-yl]-N-methylethanamineIC5035.0 [1]
2-(3-Benzylpiperidin-1-yl)-N-methylethanamineIC50120.0 [1]
2-[4-[(4-Fluorophenyl)methoxy]piperidin-1-yl]-N-methylethanamineIC5019.0 [1]
1-[2-(Methylamino)ethyl]-N-phenylpiperidin-4-amineIC50616.0 [1]
N-Methyl-2-[4-[[2-(trifluoromethyl)phenyl]methoxy]piperidin-1-yl]ethanamineIC5023.0 [1]
2-[4-[(3-Chlorophenyl)methoxy]piperidin-1-yl]-N-methylethanamineIC5033.0 [1]
2-[4-[(2-Chlorophenyl)methoxy]piperidin-1-yl]-N-methylethanamineIC5018.0 [1]
2-[4-[(3-Fluorophenyl)methoxy]piperidin-1-yl]-N-methylethanamineIC5041.0 [1]
2-[4-[[4-(3,5-Dimethylpyrazol-1-yl)phenyl]methoxy]piperidin-1-yl]-N-methylethanamineIC5015.0 [1]
2-[4-[(4-Chlorophenyl)methoxy]piperidin-1-yl]-N-methylethanamineIC5018.0 [1]
N-Methyl-2-[4-[(2-phenylphenyl)methoxy]piperidin-1-yl]ethanamineIC5041.0 [1]
2-[4-[(4-Bromophenyl)methoxy]piperidin-1-yl]-N-methylethanamineIC5015.0 [1]
2-[4-[(4-Cyclohexylphenyl)methoxy]piperidin-1-yl]-N-methylethanamineIC5042.0 [1]
N-[[1-[2-(Methylamino)ethyl]piperidin-4-yl]methyl]anilineIC50103.0 [1]
[1-[2-(Methylamino)ethyl]piperidin-4-yl]methyl benzoateIC501070.0 [1]
N-Methyl-2-[4-[(3-phenylphenyl)methoxy]piperidin-1-yl]ethanamineIC5027.0 [1]
N-[1-[2-(Methylamino)ethyl]piperidin-4-yl]benzamideIC50231.0 [1]
N-Methyl-2-[4-[(4-phenylphenyl)methoxy]piperidin-1-yl]ethanamineIC5017.0 [1]
N-Methyl-2-[4-[[3-(trifluoromethyl)phenyl]methoxy]piperidin-1-yl]ethanamineIC5028.0 [1]
2-[4-[[4-(2,3-Dichlorophenoxy)phenyl]methoxy]piperidin-1-yl]-N-methylethanamineIC5022.0 [1]
2-[4-[(3-Bromophenyl)methoxy]piperidin-1-yl]-N-methylethanamineIC5017.0 [1]
N'-[[2-(2-Chlorophenyl)sulfanylphenyl]methyl]-N'-methylethane-1,2-diamineIC5063.0 [1]
[1-[2-(Methylamino)ethyl]piperidin-4-yl]-phenylmethanolIC501637.0 [1]
N-Methyl-2-[4-(phenoxymethyl)piperidin-1-yl]ethanamineIC5098.0 [1]
2-(4-Benzylpiperidin-1-yl)-N-methylethanamineIC50890.0 [1]
1-(4-Benzylpiperidin-1-yl)-3-(methylamino)propan-2-olIC501220.0 [1]
(2S)-2-Amino-N-[[3-[5-(5-phenyl-1,3,4-oxadiazol-2-yl)-3-(trifluoromethyl)pyrazol-1-yl]phenyl]methyl]propanamideIC5060.0 [1]
(2S)-2-Amino-N-[[3-[5-(3-phenyl-1,2,4-oxadiazol-5-yl)-3-(trifluoromethyl)pyrazol-1-yl]phenyl]methyl]propanamideIC50210.0 [1]
(2S)-2-Amino-N-[[3-[5-(5-benzyl-1,3,4-oxadiazol-2-yl)-3-(trifluoromethyl)pyrazol-1-yl]phenyl]methyl]propanamideIC50310.0 [1]
(2S)-2-Amino-N-[[3-[5-(5-pyridin-4-yl-1,3,4-oxadiazol-2-yl)-3-(trifluoromethyl)pyrazol-1-yl]phenyl]methyl]propanamideIC501540.0 [1]
(2S)-2-Amino-N-[[3-[5-[5-(2-methoxyphenyl)-1,3,4-oxadiazol-2-yl]-3-(trifluoromethyl)pyrazol-1-yl]phenyl]methyl]propanamideIC5050.0 [1]
(2S)-2-Amino-N-[[3-[5-[5-(3-methoxyphenyl)-1,3,4-oxadiazol-2-yl]-3-(trifluoromethyl)pyrazol-1-yl]phenyl]methyl]propanamideIC50160.0 [1]
(2S)-2-Amino-N-[[3-[5-[5-(2-chlorophenyl)-1,3,4-oxadiazol-2-yl]-3-(trifluoromethyl)pyrazol-1-yl]phenyl]methyl]propanamideIC5050.0 [1]
(2S)-2-Amino-N-[[3-[5-[5-(2-methoxyanilino)-1,3,4-oxadiazol-2-yl]-3-(trifluoromethyl)pyrazol-1-yl]phenyl]methyl]propanamideIC5050.0 [1]
(2S)-2-Amino-N-[[3-[3-methyl-5-(5-phenyl-1,3,4-oxadiazol-2-yl)pyrazol-1-yl]phenyl]methyl]propanamideIC50130.0 [1]
(S)-2-Amino-N-(3-(1-methyl-4-(5-phenyl-1,3,4-oxadiazol-2-yl)-1H-pyrazol-5-yl)benzyl)propanamideIC502200.0 [1]
(2S)-2-Amino-N-[[3-[1-methyl-4-(5-phenyl-1,3,4-oxadiazol-2-yl)pyrazol-3-yl]phenyl]methyl]propanamideIC50400.0 [1]
(S)-2-Amino-N-(3-(4-(5-phenyl-1,3,4-oxadiazol-2-yl)oxazol-5-yl)benzyl)propanamideIC50360.0 [1]
(2S)-2-Amino-N-[[3-[5-(5-phenyl-1,3,4-oxadiazol-2-yl)imidazol-1-yl]phenyl]methyl]propanamideIC502100.0 [1]
(2S)-2-Amino-N-methyl-N-[[3-[5-(5-phenyl-1,3,4-oxadiazol-2-yl)-3-(trifluoromethyl)pyrazol-1-yl]phenyl]methyl]propanamideIC5010000.0 [1]
(2S)-1-N-[[3-[5-(5-Phenyl-1,3,4-oxadiazol-2-yl)-3-(trifluoromethyl)pyrazol-1-yl]phenyl]methyl]propane-1,2-diamineIC5010000.0 [1]
2-[3-[[(2-Aminoacetyl)amino]methyl]phenyl]-N-methyl-5-(trifluoromethyl)pyrazole-3-carboxamideIC5010600.0 [1]
2-[3-[[(2-Aminoacetyl)amino]methyl]phenyl]-N,N-dimethyl-5-(trifluoromethyl)pyrazole-3-carboxamideIC5029800.0 [1]
2-[3-[[(2-Aminoacetyl)amino]methyl]phenyl]-N-phenyl-5-(trifluoromethyl)pyrazole-3-carboxamideIC507700.0 [1]
2-[3-[[(2-Aminoacetyl)amino]methyl]phenyl]-N-(3-methylsulfonylphenyl)-5-(trifluoromethyl)pyrazole-3-carboxamideIC50230.0 [1]
2-[3-[[(2-Aminoacetyl)amino]methyl]phenyl]-N-(4-phenylphenyl)-5-(trifluoromethyl)pyrazole-3-carboxamideIC501420.0 [1]
2-[3-[(3-Aminopropanoylamino)methyl]phenyl]-N-[2-fluoro-4-(2-methylsulfonylphenyl)phenyl]-5-(trifluoromethyl)pyrazole-3-carboxamideIC5016900.0 [1]
2-[3-[[[(2S)-2-Aminopropanoyl]amino]methyl]phenyl]-N-[2-fluoro-4-(2-methylsulfonylphenyl)phenyl]-5-(trifluoromethyl)pyrazole-3-carboxamideIC50160.0 [1]
2-[3-[[[(2R)-2-Aminopropanoyl]amino]methyl]phenyl]-N-[2-fluoro-4-(2-methylsulfonylphenyl)phenyl]-5-(trifluoromethyl)pyrazole-3-carboxamideIC5020100.0 [1]
2-[3-[[(2-Amino-2-methylpropanoyl)amino]methyl]phenyl]-N-[2-fluoro-4-(2-methylsulfonylphenyl)phenyl]-5-(trifluoromethyl)pyrazole-3-carboxamideIC5030000.0 [1]
2-[3-[[(2-Amino-3,3,3-trifluoropropanoyl)amino]methyl]phenyl]-N-[2-fluoro-4-(2-methylsulfonylphenyl)phenyl]-5-(trifluoromethyl)pyrazole-3-carboxamideIC5030000.0 [1]
N-[2-Fluoro-4-(2-methylsulfonylphenyl)phenyl]-2-[3-[[[2-(methylamino)acetyl]amino]methyl]phenyl]-5-(trifluoromethyl)pyrazole-3-carboxamideIC5030000.0 [1]
1-(3-(((S)-2-Aminopropanamido)methyl)phenyl)-N-phenyl-3-(trifluoromethyl)-1H-pyrazole-5-carboxamideIC501320.0 [1]
2-[3-[[[(2S)-2-Aminopropanoyl]amino]methyl]phenyl]-N-benzyl-N-methyl-5-(trifluoromethyl)pyrazole-3-carboxamideIC503400.0 [1]
2-[3-[[[(2S)-2-Aminopropanoyl]amino]methyl]phenyl]-N-[(1S)-1-phenylethyl]-5-(trifluoromethyl)pyrazole-3-carboxamideIC507100.0 [1]
2-[3-[[[(2S)-2-Aminopropanoyl]amino]methyl]phenyl]-N-[(1R)-1-phenylethyl]-5-(trifluoromethyl)pyrazole-3-carboxamideIC50180.0 [1]
2-[3-[[[(2S)-2-Aminopropanoyl]amino]methyl]phenyl]-N-(2-phenylethyl)-5-(trifluoromethyl)pyrazole-3-carboxamideIC501100.0 [1]
2-[3-[[[(2S)-2-Aminopropanoyl]amino]methyl]phenyl]-N-cyclohexyl-5-(trifluoromethyl)pyrazole-3-carboxamideIC504300.0 [1]
2-[4-[[[(2S)-2-Aminopropanoyl]amino]methyl]phenyl]-N-benzyl-5-(trifluoromethyl)pyrazole-3-carboxamideIC5050000.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Histone-arginine methyltransferase CARM1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/histone-arginine-methyltransferase-carm1-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 9). Quest Database™ Histone-arginine methyltransferase CARM1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/histone-arginine-methyltransferase-carm1-inhibitors-ic50-ki.
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