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Histone deacetylase 3 Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
VorinostatIC5090.1 [1]
VorinostatKi5.0 [1], 12.0 [2], 29.0 [3], 36.0 [4]
Trichostatin AIC5010.32 [1]
Trichostatin AKi0.5 [1], 0.58 [2]
EntinostatIC50501.0 [1]
EntinostatKi360.0 [1]
PanobinostatIC502.1 [1]
PanobinostatKi1.1 [1], 2.3 [2], 2.4 [3]
MocetinostatIC501165.0 [1]
MocetinostatKi265.0 [1]
Tubastatin AIC5030000.0 [1]
ApicidinIC500.6 [1], 2.5 [2], 9.7 [3], 29.0 [4]
ApicidinKi0.26 [1]
DacinostatIC500.4 [1], 3.6 [2], 9.0 [3], 10.5 [4]
DacinostatKi4.2 [1]
LargazoleIC50604.0 [1]
4-Acetamido-N-(2-amino-5-thiophen-2-ylphenyl)benzamideIC50398.0 [1], 10000.0 [2], 20000.0 [3]
4-Acetamido-N-(2-amino-5-thiophen-2-ylphenyl)benzamideKi500.0 [1]
TubacinIC50630.0 [1], 1270.0 [2]
TubacinKi275.0 [1], 544.3 [2]
BelinostatIC5046.0 [1]
BelinostatKi1.5 [1], 19.0 [2]
RomidepsinIC501.3 [1], 62.0 [2]
RomidepsinKi0.15 [1]
TacedinalineIC501200.0 [1], 100000.0 [2]
TacedinalineKi550.0 [1]
RicolinostatIC5051.0 [1], 135.0 [2]
N-Hydroxy-1-(4-methoxybenzyl)-1H-indole-6-carboxamideIC5030000.0 [1], 50000.0 [2]
Largazole ThiolIC500.7 [1], 3.4 [2]
CID 25023797IC50560.0 [1], 1200.0 [2]
CID 25023798IC509400.0 [1]
N-[5-(Hydroxyamino)-5-oxopentyl]-5-(2-methylpropyl)-2-(1,3-thiazol-2-yl)-1,3-thiazole-4-carboxamideIC50100.0 [1], 102.0 [2], 175.05 [3]
5-Cyclopropyl-N-[5-(hydroxyamino)-5-oxopentyl]-2-(1,3-thiazol-2-yl)-1,3-thiazole-4-carboxamideIC50108.24 [1], 260.0 [2], 262.0 [3]
ScriptaidIC50100.0 [1]
ScriptaidKi4.1 [1]
AbexinostatKi8.2 [1], 10.0 [2]
QuisinostatKi2.1 [1], 4.3 [2]
n,n'-DihydroxyoctanediamideIC5062600.0 [1]
n,n'-DihydroxyoctanediamideKi125.0 [1]
GivinostatKi3.0 [1]
HDAC6 InhibitorIC500.42 [1], 190.0 [2]
N-Hydroxy-4-phenylbutanamideIC502000.0 [1]
N-Hydroxy-4-phenylbutanamideKi1650.0 [1]
N-(6-(2-Aminophenylamino)-6-oxohexyl)-4-methylbenzamideIC5060.0 [1], 300.0 [2]
4-[2-[2-Hydroxyethyl(Phenyl)amino]-2-Oxidanylidene-Ethyl]-~{n}-Oxidanyl-BenzamideIC501700.0 [1]
N-(2-Aminophenyl)-4-[1-[2-(3-thienyl)ethyl]-1H-1,2,3-triazol-4-yl]benzamideIC50240.0 [1], 3940.0 [2]
N'-Hydroxy-N-[3-(1-phenyltriazol-4-yl)phenyl]octanediamideIC507.2 [1]
CID 24853793IC50120.0 [1], 122.0 [2]
CID 24857909IC50670.0 [1]
N-Hydroxy-6-[(2S,5S,8S,11S)-8-(1H-indol-3-ylmethyl)-2-methyl-11-(2-methylpropyl)-3,6,9,13-tetraoxo-1,4,7,10-tetrazacyclotridec-5-yl]hexanamideIC508.0 [1], 18.0 [2]
N-(4-Hydroxybiphenyl-3-yl)benzamideIC5050000.0 [1]
6-[(2S,5S,8S,11S)-2-Benzyl-8-(1H-indol-3-ylmethyl)-11-(2-methylpropyl)-3,6,9,13-tetraoxo-1,4,7,10-tetrazacyclotridec-5-yl]-N-hydroxyhexanamideIC5031.0 [1]
6-[(2S,5S,8S,11S)-2-Methyl-11-(2-methylpropyl)-8-(naphthalen-1-ylmethyl)-3,6,9,13-tetraoxo-1,4,7,10-tetrazacyclotridec-5-yl]hexanoic acidIC50990.0 [1]
(E)-N-Hydroxy-3-[2-(2-phenylethyl)-1-(2-pyrrolidin-1-ylethyl)benzimidazol-5-yl]prop-2-enamideKi12.0 [1], 12.5 [2]
(2R)-5-Oxo-N-[(2S)-1-oxo-7-sulfanyl-1-[3-(trifluoromethyl)anilino]heptan-2-yl]pyrrolidine-2-carboxamideIC5011.0 [1]
CID 15984018IC50230.0 [1]
(S)-Benzyl 4-(5-(2-aminophenylcarbamoyl)pyridin-2-yl)-2-methylpiperazine-1-carboxylateIC50939.0 [1], 942.0 [2]
N-(2-Amino-5-thiophen-2-ylphenyl)-4-methoxybenzamideIC5020000.0 [1]
(5R,8S,11S)-5-Methyl-8-propan-2-yl-11-[(E)-4-sulfanylbut-1-enyl]-10-oxa-3,17-dithia-7,14,19,20-tetrazatricyclo[14.2.1.12,5]icosa-1(18),2(20),16(19)-triene-6,9,13-trioneIC500.7 [1], 2.78 [2]
1-[5-(2,3-Dihydro-1H-indol-1-ylcarbonyl)thiophen-2-yl]-2,2,2-trifluoroethan-1-oneIC501400.0 [1], 1700.0 [2]
(E)-3-(1'-Benzyl-4-oxospiro[3H-chromene-2,4'-piperidine]-6-yl)-N-hydroxyprop-2-enamideIC509.4 [1], 65.0 [2]
1-[5-[3-[4-(1,3,4-Oxadiazole-2-yl)phenoxymethyl]-1,2,4-oxadiazole-5-yl]-2-thienyl]trifluoroethanoneIC50380.0 [1], 1000.0 [2]
6-[(2S,5S,8S,11S)-2-(4-Aminobutyl)-11-(2-methylpropyl)-8-(naphthalen-1-ylmethyl)-3,6,9,13-tetraoxo-1,4,7,10-tetrazacyclotridec-5-yl]hexanoic acidIC50240.0 [1], 242.0 [2]
N-Hydroxy-2-(1-methylpyrrole-2-carbonyl)-3,4-dihydro-1H-isoquinoline-6-carboxamideIC5046000.0 [1]
(E)-3-[1'-[(4-Fluorophenyl)methyl]-4-oxospiro[3H-chromene-2,4'-piperidine]-6-yl]-N-hydroxyprop-2-enamideIC5090.0 [1], 92.0 [2]
(E)-N-Hydroxy-3-[4-oxo-1'-(2-phenylethyl)spiro[3H-chromene-2,4'-piperidine]-6-yl]prop-2-enamideIC50130.0 [1]
N-[(2S)-1-[4-[(E)-3-(Hydroxyamino)-3-oxoprop-1-enyl]-2-methoxyphenoxy]-3-(1H-indol-3-yl)propan-2-yl]-2-propylpentanamideIC507.5 [1], 280.0 [2]
N-[[4-(Hydroxycarbamoyl)phenyl]methyl]-1-methylpyrrole-2-carboxamideIC504500.0 [1]
(1R,5S)-N-[2-Amino-5-(4-fluorophenyl)phenyl]-8-oxabicyclo[3.2.1]octane-3-carboxamideIC502280.0 [1], 13700.0 [2]
[(E)-5-Sulfanylpent-2-enyl] (2S)-3-methyl-2-[[2-(1,3-thiazol-4-yl)-1,3-thiazole-4-carbonyl]amino]butanoateIC5058.0 [1], 60.0 [2]
[(E)-5-Sulfanylpent-2-enyl] (2S)-3-methyl-2-[[2-(2-methyl-1,3-thiazol-4-yl)-1,3-thiazole-4-carbonyl]amino]butanoateIC50106.0 [1], 110.0 [2]
[(E)-5-Octanoylsulfanylpent-2-enyl] (2S)-3-methyl-2-[[2-(1,3-thiazol-4-yl)-1,3-thiazole-4-carbonyl]amino]butanoateIC502830.0 [1], 2831.0 [2]
[(E)-5-Octanoylsulfanylpent-2-enyl] (2S)-3-methyl-2-[[2-(2-methyl-1,3-thiazol-4-yl)-1,3-thiazole-4-carbonyl]amino]butanoateIC503558.0 [1], 3560.0 [2]
N-[5-(Hydroxyamino)-5-oxopentyl]-2-(1,3-thiazol-2-yl)-1,3-thiazole-4-carboxamideIC50107.0 [1], 110.0 [2]
N-[5-(Hydroxyamino)-5-oxopentyl]-5-methyl-2-(1,3-thiazol-2-yl)-1,3-thiazole-4-carboxamideIC50620.0 [1], 691.0 [2]
5-Ethyl-N-[5-(hydroxyamino)-5-oxopentyl]-2-(1,3-thiazol-2-yl)-1,3-thiazole-4-carboxamideIC50256.0 [1], 260.0 [2]
N-[5-(Hydroxyamino)-5-oxopentyl]-5-propan-2-yl-2-(1,3-thiazol-2-yl)-1,3-thiazole-4-carboxamideIC50358.0 [1], 360.0 [2]
5-Butyl-N-[5-(hydroxyamino)-5-oxopentyl]-2-(1,3-thiazol-2-yl)-1,3-thiazole-4-carboxamideIC50188.0 [1], 190.0 [2]
5-Ethenyl-N-[5-(hydroxyamino)-5-oxopentyl]-2-(1,3-thiazol-2-yl)-1,3-thiazole-4-carboxamideIC50380.0 [1], 384.0 [2]
N-[5-(Hydroxyamino)-5-oxopentyl]-5-[(E)-3-methylbut-1-enyl]-2-(1,3-thiazol-2-yl)-1,3-thiazole-4-carboxamideIC50140.0 [1], 142.0 [2]
N-[5-(Hydroxyamino)-5-oxopentyl]-5-[(E)-prop-1-enyl]-2-(1,3-thiazol-2-yl)-1,3-thiazole-4-carboxamideIC50106.0 [1], 110.0 [2]
N-[5-(Hydroxyamino)-5-oxopentyl]-5-(2-hydroxy-2-methylpropyl)-2-(1,3-thiazol-2-yl)-1,3-thiazole-4-carboxamideIC502203.0 [1], 2590.0 [2]
5-Cyclohexyl-N-[5-(hydroxyamino)-5-oxopentyl]-2-(1,3-thiazol-2-yl)-1,3-thiazole-4-carboxamideIC50325.0 [1], 330.0 [2]
N-[5-(Hydroxyamino)-5-oxopentyl]-5-(2-propan-2-ylcyclopropyl)-2-(1,3-thiazol-2-yl)-1,3-thiazole-4-carboxamideIC50276.0 [1], 280.0 [2]
N-[5-(Hydroxyamino)-5-oxopentyl]-5-phenyl-2-(1,3-thiazol-2-yl)-1,3-thiazole-4-carboxamideIC50377.0 [1], 380.0 [2]
5-(4-Fluorophenyl)-N-[5-(hydroxyamino)-5-oxopentyl]-2-(1,3-thiazol-2-yl)-1,3-thiazole-4-carboxamideIC50310.0 [1], 314.0 [2]
5-(2-Chlorophenyl)-N-[5-(hydroxyamino)-5-oxopentyl]-2-(1,3-thiazol-2-yl)-1,3-thiazole-4-carboxamideIC50450.0 [1], 453.0 [2]
5-(2-Chloro-4-fluorophenyl)-N-[5-(hydroxyamino)-5-oxopentyl]-2-(1,3-thiazol-2-yl)-1,3-thiazole-4-carboxamideIC50587.0 [1], 590.0 [2]
N-[5-(Hydroxyamino)-5-oxopentyl]-5-(4-nitrophenyl)-2-(1,3-thiazol-2-yl)-1,3-thiazole-4-carboxamideIC50200.0 [1], 201.0 [2]
5-Benzyl-N-[5-(hydroxyamino)-5-oxopentyl]-2-(1,3-thiazol-2-yl)-1,3-thiazole-4-carboxamideIC5079.0 [1], 80.0 [2]
N-[5-(Hydroxyamino)-5-oxopentyl]-5-(2-phenylmethoxyethyl)-2-(1,3-thiazol-2-yl)-1,3-thiazole-4-carboxamideIC50158.0 [1], 160.0 [2]
N-[(2S)-1-[[4-(Hydroxyamino)-4-oxobutyl]amino]-3-methyl-1-oxobutan-2-yl]-2-(1,3-thiazol-4-yl)-1,3-thiazole-4-carboxamideIC501638.0 [1], 1640.0 [2]
N-[(2S)-1-[[3-(Hydroxyamino)-3-oxopropyl]amino]-3-methyl-1-oxobutan-2-yl]-2-(1,3-thiazol-4-yl)-1,3-thiazole-4-carboxamideIC503136.0 [1], 3170.0 [2]
N-[(2S)-1-[[3-(Hydroxyamino)-3-oxopropyl]amino]-3-methyl-1-oxobutan-2-yl]-2-(2-methyl-1,3-thiazol-4-yl)-1,3-thiazole-4-carboxamideIC502218.0 [1], 2220.0 [2]
N-[(2S)-1-[[4-(Hydroxyamino)-4-oxobutyl]amino]-3-methyl-1-oxobutan-2-yl]-2-(2-methyl-1,3-thiazol-4-yl)-1,3-thiazole-4-carboxamideIC501577.0 [1], 1580.0 [2]
N-[5-(Hydroxyamino)-5-oxopentyl]-2-(1,3-thiazol-4-yl)-1,3-thiazole-4-carboxamideIC50193.0 [1], 270.0 [2]
N-[5-(Hydroxyamino)-5-oxopentyl]-2-(2-methyl-1,3-thiazol-4-yl)-1,3-thiazole-4-carboxamideIC50150.0 [1], 615.0 [2]
N-[[4-[(E)-3-(Hydroxyamino)-3-oxoprop-1-enyl]cyclohexyl]methyl]-4,4-dimethyl-2-oxo-1,3-dihydroquinoline-6-carboxamideIC5015.0 [1], 370.0 [2]
N-[[4-[3-(Hydroxyamino)-3-oxopropyl]cyclohexyl]methyl]-4,4-dimethyl-2-oxo-1,3-dihydroquinoline-6-carboxamideIC5087.0 [1], 89.0 [2]
Valproic acidIC50161000.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Histone deacetylase 3 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/histone-deacetylase-3-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 9). Quest Database™ Histone deacetylase 3 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/histone-deacetylase-3-inhibitors-ic50-ki.
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