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Histone-lysine N-methyltransferase, H3 lysine-9 specific 5 Inhibitors (IC50, Ki)

Structure
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▼
Compound Name
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▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
N-(1-Benzylpiperidin-4-yl)-6,7-dimethoxy-2-(4-methyl-1,4-diazepan-1-yl)quinazolin-4-amineIC50700.0 [1]
CID 44251522IC5020.0 [1], 50.0 [2], 58.0 [3]
Unc-0638IC5019.0 [1]
SodiumIC5081000.0 [1], 100000.0 [2]
SinefunginIC50100.0 [1], 513000.0 [2]
CID 46901937IC5015.0 [1], 23.0 [2]
GlutathioneIC50100000.0 [1]
OxiglutationeIC50100000.0 [1]
CysteamineIC50100000.0 [1]
DisulfiramIC501600.0 [1]
S-Adenosyl-L-homocysteineIC50230.0 [1]
AnthraquinoneIC50100000.0 [1]
Cystamine dihydrochlorideIC50100000.0 [1]
NinhydrinIC50100000.0 [1]
1,4-NaphthoquinoneIC5014000.0 [1]
EbselenIC50730.0 [1]
ThiramIC501100.0 [1]
Diphenyl diselenideIC50860.0 [1]
2,2'-DithiodipyridineIC502700.0 [1]
AzodicarbonamideIC501700.0 [1]
N-(4-((2-Amino-6-methylpyrimidin-4-yl)amino)phenyl)-4-(quinolin-4-ylamino)benzamideIC5065000.0 [1]
CID 53315878IC502.5 [1]
CID 76285486IC5038.0 [1]
Benzeneseleninic acidIC504900.0 [1]
CID 53315882IC5015.0 [1]
6,7-Dimethoxy-2-(pyrrolidin-1-yl)-N-(5-(pyrrolidin-1-yl)pentyl)quinazolin-4-amineIC50100000.0 [1]
CID 44604812IC504.0 [1]
6,7-Dimethoxy-N-(1-methylpiperidin-4-yl)-2-(piperidin-1-yl)quinazolin-4-amineIC5012.0 [1]
6,7-Dimethoxy-N-(1-Methylpiperidin-4-Yl)-2-(Morpholin-4-Yl)quinazolin-4-AmineIC5013.0 [1]
N2,N2-Diethyl-6,7-dimethoxy-N4-(1-methylpiperidin-4-yl)quinazoline-2,4-diamineIC5023.0 [1]
6,7-Dimethoxy-N2,N2-dimethyl-N4-(1-methylpiperidin-4-yl)quinazoline-2,4-diamineIC5011.0 [1]
BromoselenobenzeneIC501500.0 [1]
Phenylselenenyl chlorideIC501100.0 [1]
7-(5-Aminopentoxy)-4-N-[1-(5-aminopentyl)piperidin-4-yl]-2-N-[3-(dimethylamino)propyl]-6-methoxyquinazoline-2,4-diamineIC50100.0 [1]
N-(Phenylseleno)phthalimideIC501000.0 [1]
N-[3-[(2-Amino-6-methylpyrimidin-4-yl)amino]phenyl]-4-(quinolin-4-ylamino)benzamideIC50600000.0 [1]
N-[3-[(2-Amino-6-methylpyrimidin-4-yl)amino]phenyl]-3-(quinolin-4-ylamino)benzamideIC50100000.0 [1]
2-Cyclohexyl-6-methoxy-N-(1-propan-2-ylpiperidin-4-yl)-7-(3-pyrrolidin-1-ylpropoxy)quinolin-4-amineIC50180.0 [1]
N-(1-Cyclopropylpiperidin-4-yl)-6-methoxy-2-(5-methylfuran-2-yl)-7-(3-pyrrolidin-1-ylpropoxy)quinolin-4-amineIC5020000.0 [1]
(2S)-2-Amino-4-[[(2S,3S,4R,5R)-5-(6-aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methylsulfanyl]-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]butanamideIC5030000.0 [1]
6,7-Dimethoxy-2-N-methyl-4-N-(1-methylpiperidin-4-yl)-2-N-propylquinazoline-2,4-diamineIC505.0 [1]
2-N-Cyclopentyl-6,7-dimethoxy-2-N-methyl-4-N-(1-methylpiperidin-4-yl)quinazoline-2,4-diamineIC504.0 [1]
6-Methoxy-7-[(2-methyl-2-azaspiro[3.3]heptan-6-yl)oxy]-2-(5-methylfuran-2-yl)-N-(1-methylpiperidin-4-yl)quinolin-4-amineIC5020000.0 [1]
2-(5-Ethylfuran-2-yl)-6-methoxy-N-[(1-methylpiperidin-4-yl)methyl]-7-(3-pyrrolidin-1-ylpropoxy)quinolin-4-amineIC5020000.0 [1]
6,7-Dimethoxy-2-N-methyl-4-N-(1-methylpiperidin-4-yl)-2-N-propan-2-ylquinazoline-2,4-diamineIC5018.0 [1]
2-N-Cyclohexyl-6,7-dimethoxy-2-N-methyl-4-N-(1-methylpiperidin-4-yl)quinazoline-2,4-diamineIC506.0 [1]
2-N-Hexyl-6,7-dimethoxy-4-N-(1-methylpiperidin-4-yl)quinazoline-2,4-diamineIC507.0 [1]
6,7-Dimethoxy-N-(1-methylpiperidin-4-yl)-2-morpholin-4-ylquinolin-4-amineIC506.0 [1]
2-N-Heptyl-6,7-dimethoxy-4-N-(1-methylpiperidin-4-yl)quinazoline-2,4-diamineIC5044.0 [1]
2-N-(Cyclohexylmethyl)-6,7-dimethoxy-2-N-methyl-4-N-(1-methylpiperidin-4-yl)quinazoline-2,4-diamineIC5020.0 [1]
6-Ethoxy-7-methoxy-N-(1-methylpiperidin-4-yl)-2-morpholin-4-ylquinazolin-4-amineIC505000.0 [1]
2-Cyclohexyl-6,7-dimethoxy-N-(1-methylpiperidin-4-yl)quinazolin-4-amineIC5034.0 [1]
7-Methoxy-6-methyl-N-(1-methylpiperidin-4-yl)-2-morpholin-4-ylquinazolin-4-amineIC50808.0 [1]
6,7-Dimethoxy-N-(1-methylpiperidin-4-yl)-2-pyrrolidin-1-ylquinazolin-4-amineIC5012.0 [1]
2-N-Ethyl-6,7-dimethoxy-4-N-(1-methylpiperidin-4-yl)-2-N-propylquinazoline-2,4-diamineIC5020.0 [1]
N-(1-Ethylpiperidin-4-yl)-6,7-dimethoxy-2-morpholin-4-ylquinazolin-4-amineIC5026.0 [1]
6,7-Dimethoxy-2-N-methyl-4-N-(1-methylpiperidin-4-yl)-2-N-(2-methylpropyl)quinazoline-2,4-diamineIC5028.0 [1]
6,7-Dimethoxy-2-morpholin-4-yl-N-(1-propan-2-ylpiperidin-4-yl)quinazolin-4-amineIC5015.0 [1]
7-Fluoro-6-methoxy-N-(1-methylpiperidin-4-yl)-2-morpholin-4-ylquinazolin-4-amineIC505000.0 [1]
3-[[6,7-Dimethoxy-4-[(1-methylpiperidin-4-yl)amino]quinazolin-2-yl]-methylamino]propan-1-olIC5073.0 [1]
2-[[6,7-Dimethoxy-4-[(1-methylpiperidin-4-yl)amino]quinazolin-2-yl]-methylamino]ethanolIC5020.0 [1]
2-N-Cyclobutyl-6,7-dimethoxy-2-N-methyl-4-N-(1-methylpiperidin-4-yl)quinazoline-2,4-diamineIC5017.0 [1]
6,7-Dimethoxy-2-N-methyl-4-N-(1-methylpiperidin-4-yl)-2-N-(oxan-4-yl)quinazoline-2,4-diamineIC50159.0 [1]
2-N-Benzyl-6,7-dimethoxy-2-N-methyl-4-N-(1-methylpiperidin-4-yl)quinazoline-2,4-diamineIC5046.0 [1]
7-Methoxy-N-(1-methylpiperidin-4-yl)-2-morpholin-4-yl-6-propan-2-yloxyquinazolin-4-amineIC506000.0 [1]
6-Fluoro-7-methoxy-N-(1-methylpiperidin-4-yl)-2-morpholin-4-ylquinazolin-4-amineIC501230.0 [1]
2-N-Hexyl-6,7-dimethoxy-4-N-(1-methylpiperidin-4-yl)quinoline-2,4-diamineIC5011.0 [1]
6-[[6,7-Dimethoxy-4-[(1-methylpiperidin-4-yl)amino]quinazolin-2-yl]amino]hexan-1-olIC5059.0 [1]
6,7-Dimethoxy-2-morpholin-4-yl-N-(1-propylpiperidin-4-yl)quinazolin-4-amineIC5011.0 [1]
2-N-Hexyl-6,7-dimethoxy-2-N-methyl-4-N-(1-methylpiperidin-4-yl)quinazoline-2,4-diamineIC5018.0 [1]
6,7-Dimethoxy-2-N-(2-methoxyethyl)-2-N-methyl-4-N-(1-methylpiperidin-4-yl)quinazoline-2,4-diamineIC5058.0 [1]
7-Ethoxy-6-methoxy-N-(1-methylpiperidin-4-yl)-2-morpholin-4-ylquinazolin-4-amineIC501000.0 [1]
2-N-Cyclohexyl-6,7-dimethoxy-4-N-(1-methylpiperidin-4-yl)quinazoline-2,4-diamineIC5077.0 [1]
6,7-Dimethoxy-2-N-(2-methoxyethyl)-4-N-(1-methylpiperidin-4-yl)quinazoline-2,4-diamineIC50135.0 [1]
2-N-Butyl-6,7-dimethoxy-4-N-(1-methylpiperidin-4-yl)quinazoline-2,4-diamineIC5035.0 [1]
2-N-[2-(Dimethylamino)ethyl]-6,7-dimethoxy-2-N-methyl-4-N-(1-methylpiperidin-4-yl)quinazoline-2,4-diamineIC5024.0 [1]
2-(4,4-Difluoropiperidin-1-yl)-6,7-dimethoxy-N-(1-methylpiperidin-4-yl)quinazolin-4-amineIC5097.0 [1]
6-Methoxy-7-methyl-N-(1-methylpiperidin-4-yl)-2-morpholin-4-ylquinazolin-4-amineIC5029.0 [1]
N-(1-Cyclopropylpiperidin-4-yl)-6,7-dimethoxy-2-morpholin-4-ylquinazolin-4-amineIC5012.0 [1]
6,7-Dimethoxy-N-(1-methylpiperidin-4-yl)-2-(oxan-4-yl)quinazolin-4-amineIC50341.0 [1]
2-N-(2,2-Dimethylpropyl)-6,7-dimethoxy-2-N-methyl-4-N-(1-methylpiperidin-4-yl)quinazoline-2,4-diamineIC5050.0 [1]
2-N-Ethyl-6,7-dimethoxy-2-N-methyl-4-N-(1-methylpiperidin-4-yl)quinazoline-2,4-diamineIC5018.0 [1]
6,7-Dimethoxy-2-N-methyl-4-N-(1-methylpiperidin-4-yl)-2-N-phenylquinazoline-2,4-diamineIC5043.0 [1]
2-N-(2,2-Dimethylpropyl)-6,7-dimethoxy-4-N-(1-methylpiperidin-4-yl)quinazoline-2,4-diamineIC5024.0 [1]
2-N-Butyl-6,7-dimethoxy-2-N-methyl-4-N-(1-methylpiperidin-4-yl)quinazoline-2,4-diamineIC5035.0 [1]
2-N-Butyl-2-N-ethyl-6,7-dimethoxy-4-N-(1-methylpiperidin-4-yl)quinazoline-2,4-diamineIC5023.0 [1]
6,7-Dimethoxy-2-N-(5-methylhexyl)-4-N-(1-methylpiperidin-4-yl)quinazoline-2,4-diamineIC5027.0 [1]
6,7-Dimethoxy-4-N-(1-methylpiperidin-4-yl)-2-N-pentylquinazoline-2,4-diamineIC5063.0 [1]
2-(Azepan-1-yl)-6,7-dimethoxy-N-(1-methylpiperidin-4-yl)quinazolin-4-amineIC5016.0 [1]
6-Methoxy-N-(1-methylpiperidin-4-yl)-2-morpholin-4-yl-7-propan-2-yloxyquinazolin-4-amineIC505000.0 [1]
2-N-Butyl-6,7-dimethoxy-4-N-(1-methylpiperidin-4-yl)-2-N-propylquinazoline-2,4-diamineIC5036.0 [1]
6,7-Dimethoxy-2-N-methyl-4-N-(1-methylpiperidin-4-yl)-2-N-pentylquinazoline-2,4-diamineIC5028.0 [1]
2-N-Cyclopropyl-6,7-dimethoxy-2-N-methyl-4-N-(1-methylpiperidin-4-yl)quinazoline-2,4-diamineIC5030.0 [1]
1-(1,2,3-Benzothiadiazol-6-Yl)-3-(2-Oxo-2-Phenylethyl)ureaIC5025000.0 [1]
N-[4-[(2-Amino-6-methylpyrimidin-4-yl)amino]phenyl]-3-(quinolin-4-ylamino)benzamideIC50100000.0 [1]
N-[2-[(2-Amino-6-methylpyrimidin-4-yl)amino]phenyl]-3-(quinolin-4-ylamino)benzamideIC50500000.0 [1]
N-[2-[(2-Amino-6-methylpyrimidin-4-yl)amino]phenyl]-4-(quinolin-4-ylamino)benzamideIC50400000.0 [1]
(2R,3R,4S,5R)-2-(6-Aminopurin-9-yl)-5-pentyloxolane-3,4-diolIC5087000.0 [1]
(2R,3S,4R,5R)-2-(2-Amino-3-cyclohexylpropyl)-5-(6-aminopurin-9-yl)oxolane-3,4-diolIC501500.0 [1]
(2R,3R,4S,5R)-2-(6-Aminopurin-9-yl)-5-(3-phenylpropyl)oxolane-3,4-diolIC50235000.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Histone-lysine N-methyltransferase, H3 lysine-9 specific 5 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/histone-lysine-n-methyltransferase-h3-lysine-9-specific-5-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 9). Quest Database™ Histone-lysine N-methyltransferase, H3 lysine-9 specific 5 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/histone-lysine-n-methyltransferase-h3-lysine-9-specific-5-inhibitors-ic50-ki.
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