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Histone-lysine N-methyltransferase SETD7 Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
3-[3-[4-[4-(Trifluoromethyl)phenyl]-1H-indole-1-yl]benzylamino]benzoic acidIC509930.0 [1], 19000.0 [2], 19500.0 [3], 22500.0 [4]
CyproheptadineIC501000.0 [1], 3400.0 [2], 20000.0 [3]
CyproheptadineKi15000.0 [1]
S-Adenosyl-L-homocysteineIC5030000.0 [1]
SinefunginIC502500.0 [1]

References
This online resource may be cited as follows
MLA
"Quest DatabaseHistone-lysine N-methyltransferase SETD7 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.16 Dec2025https://www.aatbio.com/data-sets/histone-lysine-n-methyltransferase-setd7-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 16). Quest DatabaseHistone-lysine N-methyltransferase SETD7 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/histone-lysine-n-methyltransferase-setd7-inhibitors-ic50-ki.
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