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Histone-lysine N-methyltransferase SUV39H1 Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
ChaetocinIC50800.0 [1]
S-Adenosyl-L-homocysteineIC501200.0 [1]
S-Adenosyl-L-homocysteineKi4900.0 [1]
(2S)-2-Amino-4-[[(2S,3S,4R,5R)-3,4-dihydroxy-5-[6-(methylamino)purin-9-yl]oxolan-2-yl]methylsulfanyl]butanoic acidKi20000.0 [1], 100000.0 [2]
5'-[(3-{[(4-Tert-Butylphenyl)carbamoyl]amino}propyl)(Propan-2-Yl)amino]-5'-DeoxyadenosineKi50000.0 [1], 100000.0 [2]

References
This online resource may be cited as follows
MLA
"Quest DatabaseHistone-lysine N-methyltransferase SUV39H1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.22 Dec2025https://www.aatbio.com/data-sets/histone-lysine-n-methyltransferase-suv39h1-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 22). Quest DatabaseHistone-lysine N-methyltransferase SUV39H1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/histone-lysine-n-methyltransferase-suv39h1-inhibitors-ic50-ki.
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