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HMG-CoA reductase Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
LovastatinIC5037.0 [1]
SimvastatinIC5039.81 [1]
SimvastatinKi2.6 [1], 68000.0 [2]
RosuvastatinIC503.1 [1], 4.0 [2], 5.0 [3], 5.4 [4]
RosuvastatinKi0.9 [1], 71000.0 [2]

References
This online resource may be cited as follows
MLA
"Quest DatabaseHMG-CoA reductase Inhibitors (IC50, Ki)." AAT Bioquest, Inc.6 Dec2025https://www.aatbio.com/data-sets/hmg-coa-reductase-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 6). Quest DatabaseHMG-CoA reductase Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/hmg-coa-reductase-inhibitors-ic50-ki.
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