Homeodomain-interacting protein kinase 1 Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	Staurosporine	IC50	2639.0 [1]
	Doramapimod	IC50	30000.0 [1]
	Bisindolylmaleimide IX mesylate	IC50	0.37 [1]
	N-(Pyridin-4-yl)-3-[1-(4-chlorobenzyl)indol-3-yl]-propanamide	IC50	100000.0 [1]
	1-[5-Amino-4-(3,4-dichlorophenyl)-3-methylpyrazol-1-yl]ethanone	IC50	100000.0 [1]
	3-[1-[(4-Chlorophenyl)methyl]indol-3-yl]-N-(4-nitrophenyl)propanamide	IC50	100000.0 [1]
	1-[5-Tert-butyl-3-[4-[2-(dimethylamino)ethyl]-5-oxo-1,4-diazepane-1-carbonyl]thiophen-2-yl]-3-(2,3-dichlorophenyl)urea	IC50	30000.0 [1]
	N-[2-[2-Aminoethyl(methyl)amino]-5-[[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]phenyl]acetamide	IC50	40.0 [1]
	6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-one	IC50	10000.0 [1]
	Tilfrinib	IC50	10000.0 [1]
	1-Tert-butyl-3-[7-(4-hydroxy-3-methoxyphenyl)-1,5-naphthyridin-2-yl]urea	IC50	100000.0 [1]
	4-(2-Chloro-4-fluorophenyl)-8-(2,6-dichlorophenyl)-7-oxido-1,7-naphthyridin-7-ium	IC50	10000.0 [1]
	N-[(4-Methoxyphenyl)methyl]-[1]benzofuro[2,3-b]pyridin-4-amine	Ki	1000000.0 [1]
	1-Benzyl-3-[7-(1-methylpyrazol-4-yl)-1,5-naphthyridin-2-yl]urea	IC50	100000.0 [1]
	1-Tert-butyl-3-[7-(1-methylpyrazol-4-yl)-1,5-naphthyridin-2-yl]urea	IC50	100000.0 [1]
	1-[7-(1-Methylpyrazol-4-yl)-1,5-naphthyridin-2-yl]-3-phenylurea	IC50	100000.0 [1]
	1-Ethyl-3-[7-(4-methoxyphenyl)-1,5-naphthyridin-2-yl]urea	IC50	100000.0 [1]
	1-[7-(3,4-Dimethoxyphenyl)-1,5-naphthyridin-2-yl]-3-ethylurea	IC50	13600.0 [1]
	1-Tert-butyl-3-[7-(3,4-dimethoxyphenyl)-1,5-naphthyridin-2-yl]urea	IC50	100000.0 [1]
	1-[7-(1-Methylpyrazol-4-yl)-1,5-naphthyridin-2-yl]-3-(2-phenylethyl)urea	IC50	100000.0 [1]
	1-(4-Methoxyphenyl)-3-(3-phenylpyrido[3,4-b]pyrazin-8-yl)urea	IC50	20430.0 [1]
	N-(3-Chloro-4-fluorophenyl)-3-phenylpyrido[3,4-b]pyrazin-8-amine	IC50	100000.0 [1]
	3-Phenyl-N-(4-piperidin-1-ylphenyl)pyrido[3,4-b]pyrazin-8-amine	IC50	2730.0 [1]
	N-Phenyl-3-(4-piperidin-1-ylphenyl)pyrido[3,4-b]pyrazin-8-amine	IC50	100000.0 [1]
	N-(3-Methoxyphenyl)-3-(4-piperidin-1-ylphenyl)pyrido[3,4-b]pyrazin-8-amine	IC50	100000.0 [1]
	1-(3-Methoxyphenyl)-3-(2-phenylpyrido[3,4-b]pyrazin-5-yl)urea	IC50	100000.0 [1]
	1-Ethyl-3-(2-phenylpyrido[3,4-b]pyrazin-5-yl)urea	IC50	100000.0 [1]
	N-(3-Ethynylphenyl)-2-phenylpyrido[3,4-b]pyrazin-5-amine	IC50	100000.0 [1]
	3-Phenyl-N-(4-piperidin-1-ylphenyl)pyrido[3,4-b]pyrazin-7-amine	IC50	100000.0 [1]
	N-(2-Methoxyphenyl)-2-phenylpyrido[3,4-b]pyrazin-5-amine	IC50	100000.0 [1]
	N-(4-Methoxyphenyl)-2-phenylpyrido[3,4-b]pyrazin-5-amine	IC50	100000.0 [1]
	2-Phenyl-N-(4-piperidin-1-ylphenyl)pyrido[3,4-b]pyrazin-5-amine	IC50	922.0 [1]
	N-(4-Morpholin-4-ylphenyl)-2-phenylpyrido[3,4-b]pyrazin-5-amine	IC50	100000.0 [1]
	2-(4-Methoxyphenyl)-N-(4-piperidin-1-ylphenyl)pyrido[3,4-b]pyrazin-5-amine	IC50	7250.0 [1]
	2-(4-Methoxyphenyl)-N-(4-morpholin-4-ylphenyl)pyrido[3,4-b]pyrazin-5-amine	IC50	100000.0 [1]
	2-Phenyl-N-(4-piperidin-1-ylphenyl)pyrido[3,4-b]pyrazin-7-amine	IC50	30510.0 [1]
	N-(4-Morpholin-4-ylphenyl)-2-phenylpyrido[3,4-b]pyrazin-7-amine	IC50	100000.0 [1]
	1-(3-Phenylpyrido[3,4-b]pyrazin-8-yl)-3-prop-2-enylurea	IC50	100000.0 [1]
	N-(3-Methoxyphenyl)-2-phenylpyrido[3,4-b]pyrazin-7-amine	IC50	100000.0 [1]
	N-(3-Methoxyphenyl)-2-phenylpyrido[3,4-b]pyrazin-5-amine	IC50	100000.0 [1]
	1-(3-Methoxyphenyl)-3-(3-phenylpyrido[3,4-b]pyrazin-8-yl)urea	IC50	100000.0 [1]
	2-Phenyl-N-(4-piperidin-1-ylphenyl)pyrido[3,4-b]pyrazin-8-amine	IC50	2590.0 [1]
	N-(4-Morpholin-4-ylphenyl)-2-phenylpyrido[3,4-b]pyrazin-8-amine	IC50	8150.0 [1]
	2-(4-Methoxyphenyl)-N-(4-piperidin-1-ylphenyl)pyrido[3,4-b]pyrazin-8-amine	IC50	3210.0 [1]
	2-(4-Methoxyphenyl)-N-(4-morpholin-4-ylphenyl)pyrido[3,4-b]pyrazin-8-amine	IC50	4020.0 [1]
	N-(2,5-Dimethoxyphenyl)-2-(4-methoxyphenyl)pyrido[3,4-b]pyrazin-8-amine	IC50	13100.0 [1]
	N-Phenyl-2-(4-piperidin-1-ylphenyl)pyrido[3,4-b]pyrazin-8-amine	IC50	11850.0 [1]
	N-(3-Methoxyphenyl)-2-(4-piperidin-1-ylphenyl)pyrido[3,4-b]pyrazin-8-amine	IC50	12650.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 48 ⟨⟩

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References

This online tool may be cited as follows

MLA	"Quest Database™ Homeodomain-interacting protein kinase 1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/homeodomain-interacting-protein-kinase-1-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, May 9). Quest Database™ Homeodomain-interacting protein kinase 1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/homeodomain-interacting-protein-kinase-1-inhibitors-ic50-ki.
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