 | Gossypol | IC50 | 170.0 [1], 4800.0 [2] |
| Gossypol | Ki | 200.0 [1] |
 | Abt-737 | IC50 | 1000.0 [1] |
| Abt-737 | Ki | 20000.0 [1] |
 | 4-[8-Chloro-11-[3-(4-chloro-3,5-dimethylphenoxy)propyl]-1-oxo-7-(1,3,5-trimethylpyrazol-4-yl)-4,5-dihydro-3H-[1,4]diazepino[1,2-a]indol-2-yl]-1-methylindole-6-carboxylic acid | Ki | 1.4 [1] |
 | 8-Oxo-3-thiomorpholino-8H-acenaphtho[1,2-b]pyrrole-9-carbonitrile | IC50 | 35.0 [1], 46.0 [2], 95.0 [3] |
| 8-Oxo-3-thiomorpholino-8H-acenaphtho[1,2-b]pyrrole-9-carbonitrile | Ki | 58.0 [1], 62.0 [2] |
 | (2S)-N-(4-Methylphenyl)sulfonyl-2-[(5Z)-4-oxo-5-[(4-phenylphenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-3-yl]-3-phenylpropanamide | Ki | 250.0 [1], 290.0 [2], 440.0 [3], 470.0 [4] |
 | Venetoclax | Ki | 444.0 [1], 780.0 [2] |
 | 2-[4-[(4-Bromophenyl)sulfonylamino]-1-hydroxynaphthalen-2-yl]sulfanylacetic acid | IC50 | 2400.0 [1] |
| 2-[4-[(4-Bromophenyl)sulfonylamino]-1-hydroxynaphthalen-2-yl]sulfanylacetic acid | Ki | 490.0 [1], 1870.0 [2] |
 | 3-[8-Chloro-11-[3-(4-chloro-3,5-dimethylphenoxy)propyl]-1-oxo-7-(1,3,5-trimethylpyrazol-4-yl)-4,5-dihydro-3H-[1,4]diazepino[1,2-a]indol-2-yl]benzoic acid | Ki | 2.1 [1], 7.0 [2], 8.4 [3], 50.0 [4] |
 | 2-[[[3-[3-(4-Chloro-3,5-dimethylphenoxy)propyl]-7-(1,3,5-trimethylpyrazol-4-yl)-1H-indole-2-carbonyl]amino]methyl]pyridine-4-carboxylic acid | Ki | 7.0 [1], 41.0 [2], 50.0 [3], 165.0 [4] |
 | 7-[8-Chloro-11-[3-(4-chloro-3,5-dimethylphenoxy)propyl]-1-oxo-7-(1,3,5-trimethylpyrazol-4-yl)-4,5-dihydro-3H-[1,4]diazepino[1,2-a]indol-2-yl]-1,3-benzodioxole-5-carboxylic acid | Ki | 0.77 [1], 1.0 [2], 3.3 [3], 5.8 [4] |
 | 5-[8-Chloro-11-[3-(4-chloro-3,5-dimethylphenoxy)propyl]-1-oxo-7-(1,3,5-trimethylpyrazol-4-yl)-4,5-dihydro-3H-[1,4]diazepino[1,2-a]indol-2-yl]naphthalene-1-carboxylic acid | Ki | 0.31 [1], 1.0 [2], 1.2 [3], 2.7 [4] |
 | 7-[8-Chloro-11-[3-(4-chloro-3,5-dimethylphenoxy)propyl]-1-oxo-7-(1,3,5-trimethylpyrazol-4-yl)-4,5-dihydro-3H-[1,4]diazepino[1,2-a]indol-2-yl]-1-methylindole-5-carboxylic acid | Ki | 1.8 [1], 3.4 [2], 6.4 [3], 8.8 [4] |
 | 6-[8-Chloro-11-[3-(4-chloro-3,5-dimethylphenoxy)propyl]-1-oxo-7-(1,3,5-trimethylpyrazol-4-yl)-4,5-dihydro-3H-[1,4]diazepino[1,2-a]indol-2-yl]-1-methylindole-4-carboxylic acid | Ki | 0.7 [1], 1.0 [2], 2.3 [3], 2.8 [4] |
 | 8-[8-Chloro-11-[3-(4-chloro-3,5-dimethylphenoxy)propyl]-1-oxo-7-(1,3,5-trimethylpyrazol-4-yl)-4,5-dihydro-3H-[1,4]diazepino[1,2-a]indol-2-yl]quinoline-5-carboxylic acid | Ki | 1.0 [1], 1.4 [2], 4.4 [3], 5.0 [4] |
 | 7-[8-Chloro-11-[3-(4-chloro-3,5-dimethylphenoxy)propyl]-1-oxo-7-(1,3,5-trimethylpyrazol-4-yl)-4,5-dihydro-3H-[1,4]diazepino[1,2-a]indol-2-yl]-1-methylindole-3-carboxylic acid | Ki | 0.65 [1], 1.0 [2], 1.6 [3], 5.2 [4] |
 | 3-[8-Chloro-11-[3-(4-chloro-3,5-dimethylphenoxy)propyl]-1-oxo-7-(1,3,5-trimethylpyrazol-4-yl)-4,5-dihydro-3H-[1,4]diazepino[1,2-a]indol-2-yl]-1-methylindole-5-carboxylic acid | Ki | 0.11 [1], 0.37 [2], 1.0 [3] |
 | 3-[8-Chloro-11-[3-(4-chloro-3,5-dimethylphenoxy)propyl]-1-oxo-7-(1,3,5-trimethylpyrazol-4-yl)-4,5-dihydro-3H-[1,4]diazepino[1,2-a]indol-2-yl]-1-methylindole-7-carboxylic acid | Ki | 0.46 [1], 1.0 [2], 1.4 [3], 2.1 [4] |
 | 3-[8-Chloro-11-[3-(4-chloro-3,5-dimethylphenoxy)propyl]-1-oxo-7-(1,3,5-trimethylpyrazol-4-yl)-4,5-dihydro-3H-[1,4]diazepino[1,2-a]indol-2-yl]-1-methylindole-6-carboxylic acid | Ki | 0.24 [1], 0.63 [2], 1.0 [3] |
 | 7-[8-Chloro-11-[3-(4-chloro-3,5-dimethylphenoxy)propyl]-1-oxo-7-(1,3,5-trimethylpyrazol-4-yl)-4,5-dihydro-3H-[1,4]diazepino[1,2-a]indol-2-yl]-1-methylindole-4-carboxylic acid | Ki | 2.4 [1], 3.6 [2], 8.0 [3], 11.0 [4] |
 | 7-(2-Methylphenyl)-1-(2-morpholin-4-ylethyl)-3-(3-naphthalen-1-yloxypropyl)indole-2-carboxylic acid | Ki | 9.0 [1], 21.0 [2], 470.0 [3], 1230.0 [4] |
 | 1-(2-Morpholin-4-ylethyl)-3-(3-naphthalen-1-yloxypropyl)-7-(1,3,5-trimethylpyrazol-4-yl)indole-2-carboxylic acid | Ki | 1.5 [1], 4.0 [2], 10.0 [3], 35.0 [4] |
 | Navitoclax | IC50 | 500.0 [1], 30000.0 [2] |
| Navitoclax | Ki | 550.0 [1] |
 | (2Z)-2-[(5Z)-5-[(3,5-Dimethyl-1H-pyrrol-2-yl)methylidene]-4-methoxypyrrol-2-ylidene]indole | IC50 | 2900.0 [1] |
| (2Z)-2-[(5Z)-5-[(3,5-Dimethyl-1H-pyrrol-2-yl)methylidene]-4-methoxypyrrol-2-ylidene]indole | Ki | 1000.0 [1] |
 | 2-(1-Hydroxy-4-(thiophene-2-sulfonamido)naphthalen-2-ylthio)acetic acid | IC50 | 7120.0 [1] |
| 2-(1-Hydroxy-4-(thiophene-2-sulfonamido)naphthalen-2-ylthio)acetic acid | Ki | 1550.0 [1] |
 | 3-(3-(Naphthalen-1-yloxy)propyl)-1H-indole-2-carboxylic acid | Ki | 330.0 [1], 340.0 [2], 7300.0 [3] |
 | Isopropyl-3-(4-isopropylphenoxy)-8-oxo-8H-acenaphtho[1,2-b]pyrrole-9-carbonitrile | IC50 | 321.0 [1] |
| Isopropyl-3-(4-isopropylphenoxy)-8-oxo-8H-acenaphtho[1,2-b]pyrrole-9-carbonitrile | Ki | 99.0 [1] |
 | 5-Benzyl-2-(5-benzyl-1,4,6,7-tetrahydroxy-3-methylnaphthalen-2-yl)-3-methylnaphthalene-1,4,6,7-tetrone | IC50 | 25.0 [1], 240.0 [2] |
| 5-Benzyl-2-(5-benzyl-1,4,6,7-tetrahydroxy-3-methylnaphthalen-2-yl)-3-methylnaphthalene-1,4,6,7-tetrone | Ki | 160.0 [1] |
 | 2-[1-Hydroxy-4-[[(4-phenoxyphenyl)sulfonyl]amino]-2-naphthylthio]acetic acid | IC50 | 180.0 [1], 1450.0 [2] |
| 2-[1-Hydroxy-4-[[(4-phenoxyphenyl)sulfonyl]amino]-2-naphthylthio]acetic acid | Ki | 180.0 [1] |
 | N-(Benzenesulfonyl)-6-chloro-3-[3-(4-chloro-3,5-dimethylphenoxy)propyl]-7-(1,3,5-trimethylpyrazol-4-yl)-1H-indole-2-carboxamide | Ki | 10.0 [1], 17.0 [2], 64.0 [3] |
 | N-(Benzenesulfonyl)-6-chloro-3-[3-(4-chloro-3,5-dimethylphenoxy)propyl]-7-(2-methylpyridin-3-yl)-1H-indole-2-carboxamide | Ki | 10.0 [1], 18.0 [2], 146.0 [3] |
 | 6-Chloro-3-[3-(4-chloro-3,5-dimethylphenoxy)propyl]-N-[3-[(3-methylbutanoylamino)methyl]phenyl]sulfonyl-7-(1,3,5-trimethylpyrazol-4-yl)-1H-indole-2-carboxamide | Ki | 5.6 [1], 10.0 [2], 92.0 [3] |
 | N-[5-(Benzylcarbamoyl)furan-2-yl]sulfonyl-6-chloro-3-[3-(4-chloro-3,5-dimethylphenoxy)propyl]-7-(1,3,5-trimethylpyrazol-4-yl)-1H-indole-2-carboxamide | Ki | 2.4 [1], 10.0 [2], 84.0 [3] |
 | 6-Chloro-3-[3-(4-chloro-3,5-dimethylphenoxy)propyl]-N-[5-(pyridin-4-ylmethylcarbamoyl)furan-2-yl]sulfonyl-7-(1,3,5-trimethylpyrazol-4-yl)-1H-indole-2-carboxamide | Ki | 8.5 [1], 10.0 [2], 20.0 [3] |
 | 6-Chloro-3-[3-(4-chloro-3,5-dimethylphenoxy)propyl]-N-[2-(3-methylbutylamino)pyridin-4-yl]sulfonyl-7-(1,3,5-trimethylpyrazol-4-yl)-1H-indole-2-carboxamide | Ki | 5.6 [1], 10.0 [2], 179.0 [3] |
 | 6-Chloro-3-[3-(4-chloro-3,5-dimethylphenoxy)propyl]-N-[2-(2-phenylethylamino)pyridin-4-yl]sulfonyl-7-(1,3,5-trimethylpyrazol-4-yl)-1H-indole-2-carboxamide | Ki | 1.2 [1], 10.0 [2], 78.0 [3] |
 | 6-Chloro-3-[3-(4-chloro-3,5-dimethylphenoxy)propyl]-N-[2-[methyl(2-phenylethyl)amino]pyridin-4-yl]sulfonyl-7-(1,3,5-trimethylpyrazol-4-yl)-1H-indole-2-carboxamide | Ki | 2.5 [1], 10.0 [2], 226.0 [3] |
 | 6-Chloro-3-[3-(4-chloro-3,5-dimethylphenoxy)propyl]-N-[2-(2,3-dihydro-1H-inden-2-ylamino)pyridin-4-yl]sulfonyl-7-(1,3,5-trimethylpyrazol-4-yl)-1H-indole-2-carboxamide | Ki | 1.0 [1], 10.0 [2], 61.0 [3] |
 | 6-Chloro-3-[3-(4-chloro-3,5-dimethylphenoxy)propyl]-N-[3-[[[2-(trifluoromethyl)benzoyl]amino]methyl]phenyl]sulfonyl-7-(1,3,5-trimethylpyrazol-4-yl)-1H-indole-2-carboxamide | Ki | 5.0 [1], 10.0 [2], 80.0 [3] |
 | 6-Chloro-3-[3-(4-chloro-3,5-dimethylphenoxy)propyl]-N-[3-[[[3-(trifluoromethyl)benzoyl]amino]methyl]phenyl]sulfonyl-7-(1,3,5-trimethylpyrazol-4-yl)-1H-indole-2-carboxamide | Ki | 7.0 [1], 10.0 [2], 78.0 [3] |
 | 6-Chloro-3-[3-(4-chloro-3,5-dimethylphenoxy)propyl]-N-[3-[[(1-methylpyrrole-2-carbonyl)amino]methyl]phenyl]sulfonyl-7-(1,3,5-trimethylpyrazol-4-yl)-1H-indole-2-carboxamide | Ki | 10.0 [1], 91.0 [2] |
 | 6-Chloro-3-[3-(4-chloro-3,5-dimethylphenoxy)propyl]-N-[3-[(furan-3-carbonylamino)methyl]phenyl]sulfonyl-7-(1,3,5-trimethylpyrazol-4-yl)-1H-indole-2-carboxamide | Ki | 2.9 [1], 10.0 [2], 69.0 [3] |
 | N-[3-(Acetamidomethyl)phenyl]sulfonyl-6-chloro-3-[3-(4-chloro-3,5-dimethylphenoxy)propyl]-7-(1,3,5-trimethylpyrazol-4-yl)-1H-indole-2-carboxamide | Ki | 10.0 [1], 11.1 [2], 42.0 [3] |
 | 6-Chloro-3-[3-(4-chloro-3,5-dimethylphenoxy)propyl]-N-[3-[(2-methylpropanoylamino)methyl]phenyl]sulfonyl-7-(1,3,5-trimethylpyrazol-4-yl)-1H-indole-2-carboxamide | Ki | 10.0 [1], 16.0 [2], 54.0 [3] |
 | 2-[4-[[4-(4-Chlorophenyl)phenyl]sulfonylamino]-1-hydroxynaphthalen-2-yl]sulfanylacetic acid | IC50 | 170.0 [1], 880.0 [2] |
| 2-[4-[[4-(4-Chlorophenyl)phenyl]sulfonylamino]-1-hydroxynaphthalen-2-yl]sulfanylacetic acid | Ki | 170.0 [1] |
 | 2-[4-[[4-(4-Fluorophenoxy)phenyl]sulfonylamino]-1-hydroxynaphthalen-2-yl]sulfanylacetic acid | IC50 | 170.0 [1], 900.0 [2] |
| 2-[4-[[4-(4-Fluorophenoxy)phenyl]sulfonylamino]-1-hydroxynaphthalen-2-yl]sulfanylacetic acid | Ki | 290.0 [1] |
 | 2-[4-[[4-(2,4-Difluorophenyl)phenyl]sulfonylamino]-1-hydroxynaphthalen-2-yl]sulfanylacetic acid | IC50 | 170.0 [1], 920.0 [2] |
| 2-[4-[[4-(2,4-Difluorophenyl)phenyl]sulfonylamino]-1-hydroxynaphthalen-2-yl]sulfanylacetic acid | Ki | 240.0 [1] |
 | Indole-2-carboxylic acid | Ki | 1000000.0 [1] |
 | Apogossypolone | IC50 | 540.0 [1] |
| Apogossypolone | Ki | 430.0 [1] |
 | Apogossypol | IC50 | 2600.0 [1] |
| Apogossypol | Ki | 2600.0 [1] |
 | 7-[5-[[4-[4-(Dimethylsulfamoyl)piperazin-1-yl]phenoxy]methyl]-1,3-dimethylpyrazol-4-yl]-1-(2-morpholin-4-ylethyl)-3-(3-naphthalen-1-yloxypropyl)indole-2-carboxylic acid | Ki | 0.45 [1], 7.9 [2] |
 | 2,3,5-Trihydroxy-7-methyl-N-(2-phenylpropyl)-6-[1,6,7-trihydroxy-3-methyl-5-(2-phenylpropylcarbamoyl)naphthalen-2-yl]naphthalene-1-carboxamide | IC50 | 280.0 [1], 330.0 [2] |
 | Nvp-cgm097 | IC50 | 50000.0 [1] |
 | Anthragallol | Ki | 270.0 [1], 1211.0 [2] |
 | [(4-{[(4-Chlorophenyl)sulfonyl]amino}-1-hydroxy-2-naphthyl)thio]acetic acid | IC50 | 2700.0 [1] |
| [(4-{[(4-Chlorophenyl)sulfonyl]amino}-1-hydroxy-2-naphthyl)thio]acetic acid | Ki | 820.0 [1] |
 | N-[4-(2-Tert-Butylphenylsulfonyl)phenyl]-2,3,4-trihydroxy-5-(2-isopropylbenzyl)benzamide | IC50 | 1030.0 [1] |
| N-[4-(2-Tert-Butylphenylsulfonyl)phenyl]-2,3,4-trihydroxy-5-(2-isopropylbenzyl)benzamide | Ki | 300.0 [1] |
 | [(1-Hydroxy-4-{[(4-methoxyphenyl)sulfonyl]amino}-2-naphthyl)thio]acetic acid | IC50 | 7170.0 [1] |
| [(1-Hydroxy-4-{[(4-methoxyphenyl)sulfonyl]amino}-2-naphthyl)thio]acetic acid | Ki | 9310.0 [1] |
 | 7-[3-[[4-(4-Acetylpiperazin-1-yl)phenoxy]methyl]-1,5-dimethylpyrazol-4-yl]-3-(3-naphthalen-1-yloxypropyl)-1-(pyridin-3-ylmethyl)indole-2-carboxylic acid | Ki | 1.8 [1], 98.0 [2] |
 | [(4-{[(4-Ethylphenyl)sulfonyl]amino}-1-hydroxy-2-naphthyl)thio]acetic acid | IC50 | 8680.0 [1] |
| [(4-{[(4-Ethylphenyl)sulfonyl]amino}-1-hydroxy-2-naphthyl)thio]acetic acid | Ki | 1550.0 [1] |
 | 4-[(E)-(2-Cyclohexylimino-4-methyl-1,3-thiazol-3-yl)iminomethyl]benzene-1,2,3-triol | IC50 | 4700.0 [1], 4720.0 [2] |
 | 2-({1-Hydroxy-4-[4-(propan-2-yl)benzenesulfonamido]naphthalen-2-yl}sulfanyl)acetic acid | IC50 | 4000.0 [1] |
| 2-({1-Hydroxy-4-[4-(propan-2-yl)benzenesulfonamido]naphthalen-2-yl}sulfanyl)acetic acid | Ki | 1060.0 [1] |
 | (4-Phenoxyphenyl)-(2,3,4-trihydroxy-5-propan-2-ylphenyl)methanone | Ki | 380.0 [1] |
 | 4-(4-Chlorophenyl)-1-[(3S)-3,4-dihydroxybutyl]-N-[3-(4-methylpiperazin-1-yl)propyl]-3-phenylpyrrole-2-carboxamide | IC50 | 100000.0 [1] |
 | N-(4-Hydroxynaphthalen-1-yl)benzenesulfonamide | IC50 | 100000.0 [1] |
| N-(4-Hydroxynaphthalen-1-yl)benzenesulfonamide | Ki | 27000.0 [1] |
 | [(1-Hydroxy-4-{[(4-methylphenyl)sulfonyl]amino}-2-naphthyl)thio]acetic acid | IC50 | 11570.0 [1] |
| [(1-Hydroxy-4-{[(4-methylphenyl)sulfonyl]amino}-2-naphthyl)thio]acetic acid | Ki | 3130.0 [1] |
 | [(4-{[(4-Fluorophenyl)sulfonyl]amino}-1-hydroxynaphthalen-2-yl)sulfanyl]acetic acid | IC50 | 5010.0 [1] |
| [(4-{[(4-Fluorophenyl)sulfonyl]amino}-1-hydroxynaphthalen-2-yl)sulfanyl]acetic acid | Ki | 4230.0 [1] |
 | ({1-Hydroxy-4-[(2-naphthylsulfonyl)amino]-2-naphthyl}sulfanyl)acetic acid | IC50 | 2760.0 [1] |
| ({1-Hydroxy-4-[(2-naphthylsulfonyl)amino]-2-naphthyl}sulfanyl)acetic acid | Ki | 730.0 [1] |
 | 2-Methyl-3-phenyl-5,6,7-trihydroxy-8-isobutylchromone | Ki | 400.0 [1] |
 | Benzo[d]thiazol-2-yl(2,3,4-trihydroxy-5-(4-phenoxybenzoyl)phenyl)methanone | Ki | 37.0 [1] |
 | 1,4-Bis(5,6,7-trihydroxy-8-isobutyl-2-methyl-4-oxo-4H-chromen-3-yl)benzene | Ki | 18.0 [1] |
 | 5,6,7-Trihydroxy-8-isobutyl-2-methyl-4H-chromen-4-one | Ki | 1690.0 [1] |
 | Phenyl-(2,3,4-trihydroxy-5-propan-2-ylphenyl)methanone | Ki | 4600.0 [1] |
 | 2-Methyl-1-[2,3,4-trihydroxy-5-(4-phenoxybenzoyl)phenyl]propan-1-one | Ki | 340.0 [1] |
 | 3-(p-Tolyloxy)-8-oxo-8H-acenaphtho[1,2-b]pyrrole-9-carbonitrile | Ki | 174.0 [1], 1915.0 [2] |
 | 3-(Biphenyl-4-yloxy)-8-oxo-8H-acenaphtho[1,2-b]pyrrole-9-carbonitrile | Ki | 1281.0 [1] |
 | 3-(4-Methoxyphenoxy)-8-oxo-8H-acenaphtho[1,2-b]pyrrole-9-carbonitrile | Ki | 122.0 [1], 258.0 [2] |
 | 3-(4-Methoxyphenylthio)-8-oxo-8H-acenaphtho[1,2-b]pyrrole-9-carbonitrile | IC50 | 388.0 [1] |
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