Structure | Compound Name | Standard Type | Standard Values (in nM) |
|---|---|---|---|
| IKK Inhibitor VII | IC50 | 300.0 [1] | |
| [4-[[4-[5-(3-Hydroxy-3-methylbutyl)thiophen-2-yl]pyrimidin-2-yl]amino]phenyl]-(4-pyrrolidin-1-ylpiperidin-1-yl)methanone | IC50 | 50.0 [1], 450.0 [2], 500.0 [3], 600.0 [4], 2000.0 [5] | |
| [4-[[4-[5-(4-Hydroxybutyl)thiophen-2-yl]pyrimidin-2-yl]amino]phenyl]-(4-pyrrolidin-1-ylpiperidin-1-yl)methanone | IC50 | 40.0 [1], 200.0 [2], 2000.0 [3] | |
| 4-(4-(Benzo[b]thiophen-2-yl)pyrimidin-2-ylamino)-N-(2-(dimethylamino)ethyl)benzamide | IC50 | 300.0 [1], 500.0 [2], 5000.0 [3] | |
| [4-[[4-(1-Benzothiophen-2-yl)pyrimidin-2-yl]amino]phenyl]-[4-(dimethylamino)piperidin-1-yl]methanone | IC50 | 80.0 [1], 300.0 [2], 400.0 [3], 2000.0 [4] | |
MLA | "Quest Database™ Inhibitor of NF-kappa-B kinase (IKK) Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 4 Dec. 2025, https://www.aatbio.com/data-sets/inhibitor-of-nf-kappa-b-kinase-ikk-inhibitors-ic50-ki. | |
APA | AAT Bioquest, Inc. (2025, December 4). Quest Database™ Inhibitor of NF-kappa-B kinase (IKK) Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/inhibitor-of-nf-kappa-b-kinase-ikk-inhibitors-ic50-ki. | |
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