Inosine-5'-monophosphate dehydrogenase 1 Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	Mycophenolic acid	IC50	19.0 [1], 20.0 [2], 32.0 [3], 55.0 [4], 260.0 [5]
	Mycophenolic acid	Ki	40.0 [1]
	C2-Mycophenolic adenine dinucleotide	Ki	330.0 [1]
	[[(2R,3S,4R,5R)-5-(6-Aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] [(2S,3R,4S,5S)-5-(4-carbamoyl-1,3-thiazol-2-yl)-3,4-dihydroxyoxolan-2-yl]methyl hydrogen phosphate	Ki	110.0 [1], 470.0 [2], 710.0 [3]
	[(2R,3S,4R,5R)-5-(6-Amino-2-ethylpurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-[[hydroxy-[2-(4-hydroxy-6-methoxy-7-methyl-3-oxo-1H-2-benzofuran-5-yl)ethoxy]phosphoryl]methyl]phosphinic acid	Ki	16.0 [1], 20.0 [2]
	Tiazofurin adenine dinucleotide	Ki	100.0 [1], 110.0 [2]
	[(2R,3S,4R,5R)-5-(6-Amino-2-phenylpurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-[[hydroxy-[2-(4-hydroxy-6-methoxy-7-methyl-3-oxo-1H-2-benzofuran-5-yl)ethoxy]phosphoryl]methyl]phosphinic acid	Ki	66.0 [1], 70.0 [2]
	Mycophenolic hydroxamic acid	IC50	350.0 [1]
	Mycophenolic hydroxamic acid	Ki	70.0 [1]
	[(2S,3R,4S,5S)-5-(6-Aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-[[hydroxy-[(E)-4-(4-hydroxy-6-methoxy-7-methyl-3-oxo-1H-2-benzofuran-5-yl)-2-methylbut-2-enoxy]phosphoryl]methyl]phosphinic acid	Ki	520.0 [1]
	Selenazole-4-carboxyamide-adenine dinucleotide	Ki	33.0 [1], 62.0 [2]
	[[(2R,3S,4R,5R)-5-(6-Aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] [(2R,3S,4R,5R)-5-(4-carbamoylselenophen-2-yl)-3,4-dihydroxyoxolan-2-yl]methyl hydrogen phosphate	Ki	260.0 [1], 580.0 [2]
	[[(2R,3S,4R,5R)-5-(6-Aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] [(2R,3S,4R,5R)-5-(4-carbamoylthiophen-2-yl)-3,4-dihydroxyoxolan-2-yl]methyl hydrogen phosphate	Ki	340.0 [1], 370.0 [2]
	[[(2R,3S,4R,5R)-5-(6-Aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] [(2R,3S,4R,5R)-5-(4-carbamoylfuran-2-yl)-3,4-dihydroxyoxolan-2-yl]methyl hydrogen phosphate	Ki	37970.0 [1], 135120.0 [2]
	Adenosine	Ki	100000.0 [1]
	1,1-Dioxido-1-benzothien-3-yl 5-phenyl-1,3,4-oxadiazol-2-yl sulfide	IC50	5600.0 [1]
	1-(3-Methoxy-4-oxazol-5-yl-phenyl)-3-m-tolyl-urea	IC50	55.0 [1]
	[(2S,3R,4S,5S)-5-(6-Aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-[[[(2R,3S,4R,5R)-5-(4-carbamoyl-1,3-thiazol-2-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl]methyl]phosphinic acid	Ki	110.0 [1]
	[(2R,3S,4R,5R)-5-(6-Aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-[[hydroxy-[(E)-4-(4-hydroxy-6-methoxy-7-methyl-3-oxo-1H-2-benzofuran-5-yl)-2-methylbut-2-enoxy]phosphoryl]methyl]phosphinic acid	Ki	520.0 [1]
	[(2S,3R,4S,5S)-5-(6-Aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-[[[(2R,3S,4R,5R)-5-(4-carbamoyl-1,3-thiazol-2-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl]-difluoromethyl]phosphinic acid	Ki	300.0 [1]
	O-Desmethyl Mycophenolic Acid	IC50	150.0 [1]
	Methyl mycophenolate	IC50	1500.0 [1]
	7-Hydroxy-6-[(E)-6-hydroxy-3-methylhex-2-enyl]-5-methoxy-4-methyl-3H-2-benzofuran-1-one	IC50	770.0 [1]
	7-Methoxy-6-oxazol-5-yl-2-phenyl-1H-quinolin-4-one	IC50	99.0 [1]
	3-[[5-(4-Chlorophenyl)-1,3,4-oxadiazol-2-yl]sulfanyl]-1-benzothiophene 1,1-dioxide	IC50	11100.0 [1]
	3-[[5-(4-Methoxyphenyl)-1,3,4-oxadiazol-2-yl]sulfanyl]-1-benzothiophene 1,1-dioxide	IC50	30000.0 [1]
	(E)-6-(4-Hydroxy-6-methoxy-7-methyl-3-oxo-1H-2-benzofuran-5-yl)hex-4-enoic acid	IC50	1800.0 [1]
	6-(4-Acetoxy-6-methoxy-7-methyl-3-oxo-1,3-dihydroisobenzofuran-5-yl)-4-methylhex-4-enoic acid	IC50	4100.0 [1]
	[[(2R,3S,4R,5R)-5-(6-Amino-2-iodopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] [(2R,3S,4R,5R)-5-(4-carbamoyl-1,3-thiazol-2-yl)-3,4-dihydroxyoxolan-2-yl]methyl hydrogen phosphate	Ki	19.0 [1]
	[[(2R,3S,4R,5R)-5-(6-Amino-2-ethynylpurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] [(2R,3S,4R,5R)-5-(4-carbamoyl-1,3-thiazol-2-yl)-3,4-dihydroxyoxolan-2-yl]methyl hydrogen phosphate	Ki	10.0 [1]
	[[(2R,3S,4R,5R)-5-(6-Amino-2-ethylpurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] [(2R,3S,4R,5R)-5-(4-carbamoyl-1,3-thiazol-2-yl)-3,4-dihydroxyoxolan-2-yl]methyl hydrogen phosphate	Ki	1.0 [1]
	N1-Hydroxy-N8-(3-methoxy-4-(oxazol-5-yl)phenyl)octanediamide	Ki	5000.0 [1]
	N'-[[(2R,3S,4R,5R)-5-(6-Aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methyl]-N-[2-(4-hydroxy-6-methoxy-7-methyl-3-oxo-1H-2-benzofuran-5-yl)ethyl]methanedisulfonamide	Ki	350.0 [1]
	2-[(1,1-Dioxido-1-benzothiophen-3-yl)sulfanyl]-5-(4-methylphenyl)-1,3,4-oxadiazole	IC50	20300.0 [1]
	7-Hydroxy-6-(2-hydroxyethyl)-5-methoxy-4-methylisobenzofuran-1(3H)-one	Ki	15400.0 [1]
	3-[(5-Pyridin-4-yl-1,3,4-oxadiazol-2-yl)sulfanyl]-1-benzothiophene 1,1-dioxide	IC50	8600.0 [1]
	(4E)-6-(4,6-Dimethoxy-7-methyl-3-oxo-1,3-dihydro-2-benzofuran-5-yl)-4-methylhex-4-enoic acid	IC50	67000.0 [1]
	N'-[[(2R,3S,4R,5R)-5-(6-Amino-2-phenylpurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methyl]-N-[2-(4-hydroxy-6-methoxy-7-methyl-3-oxo-1H-2-benzofuran-5-yl)ethyl]methanedisulfonamide	Ki	660.0 [1]
	N'-[[(2R,3S,4R,5R)-5-(6-Amino-2-ethynylpurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methyl]-N-[2-(4-hydroxy-6-methoxy-7-methyl-3-oxo-1H-2-benzofuran-5-yl)ethyl]methanedisulfonamide	Ki	520.0 [1]
	N'-[[(2R,3S,4R,5R)-5-(6-Amino-2-ethylpurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methyl]-N-[2-(4-hydroxy-6-methoxy-7-methyl-3-oxo-1H-2-benzofuran-5-yl)ethyl]methanedisulfonamide	Ki	820.0 [1]
	6-[(E)-4-[4-[[(2R,3S,4R,5R)-5-(6-Aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxymethyl]triazol-1-yl]-3-methylbut-2-enyl]-7-hydroxy-5-methoxy-4-methyl-3H-2-benzofuran-1-one	Ki	70.0 [1]
	Methyl 2-[[(E)-6-(4-hydroxy-6-methoxy-7-methyl-3-oxo-1H-2-benzofuran-5-yl)-4-methylhex-4-enoyl]amino]acetate	Ki	522.0 [1]
	N-(4-Methoxyphenyl)-2-[2-(1,3-thiazol-4-yl)benzimidazol-1-yl]acetamide	IC50	50000.0 [1]
	Methyl (2S)-2-[[(E)-6-(4-hydroxy-6-methoxy-7-methyl-3-oxo-1H-2-benzofuran-5-yl)-4-methylhex-4-enoyl]amino]-3-methylbutanoate	Ki	3771.0 [1]
	(2S)-2-[[(E)-6-(4-Hydroxy-6-methoxy-7-methyl-3-oxo-1H-2-benzofuran-5-yl)-4-methylhex-4-enoyl]amino]-3-methylbutanoic acid	Ki	132.0 [1]
	Methyl (2R)-2-[[(E)-6-(4-hydroxy-6-methoxy-7-methyl-3-oxo-1H-2-benzofuran-5-yl)-4-methylhex-4-enoyl]amino]-3-methylbutanoate	Ki	7723.0 [1]
	(2R)-2-[[(E)-6-(4-Hydroxy-6-methoxy-7-methyl-3-oxo-1H-2-benzofuran-5-yl)-4-methylhex-4-enoyl]amino]-3-methylbutanoic acid	Ki	2035.0 [1]
	Methyl (2R)-2-[[(E)-6-(4-hydroxy-6-methoxy-7-methyl-3-oxo-1H-2-benzofuran-5-yl)-4-methylhex-4-enoyl]amino]-3-phenylpropanoate	Ki	5556.0 [1]
	2-[[(E)-6-(4-Hydroxy-6-methoxy-7-methyl-3-oxo-1H-2-benzofuran-5-yl)-4-methylhex-4-enoyl]amino]acetic acid	Ki	892.0 [1]
	Methyl (2S)-2-[[(E)-6-(4-hydroxy-6-methoxy-7-methyl-3-oxo-1H-2-benzofuran-5-yl)-4-methylhex-4-enoyl]amino]-3-phenylpropanoate	Ki	4362.0 [1]
	(2R)-2-[[(E)-6-(4-Hydroxy-6-methoxy-7-methyl-3-oxo-1H-2-benzofuran-5-yl)-4-methylhex-4-enoyl]amino]-3-phenylpropanoic acid	Ki	4308.0 [1]
	(2S)-2-[[(E)-6-(4-Hydroxy-6-methoxy-7-methyl-3-oxo-1H-2-benzofuran-5-yl)-4-methylhex-4-enoyl]amino]-3-phenylpropanoic acid	Ki	854.0 [1]
	7-Methoxy-2-(4-methoxy-phenyl)-6-oxazol-5-yl-1H-quinolin-4-one	IC50	90.0 [1]
	[Hydroxy-[2-(4-hydroxy-6-methoxy-7-methyl-3-oxo-1H-2-benzofuran-5-yl)ethoxy]phosphoryl]methylphosphonic acid	Ki	890.0 [1]
	[Hydroxy-[2-(4-hydroxy-6-methoxy-7-methyl-3-oxo-1H-2-benzofuran-5-yl)ethoxy]phosphoryl]methyl-[2-(4-hydroxy-6-methoxy-7-methyl-3-oxo-1H-2-benzofuran-5-yl)ethoxy]phosphinic acid	Ki	2300.0 [1]
	N-[3-Methoxy-4-(1,3-oxazol-5-yl)phenyl]-1H-indole-2-carboxamide	IC50	1000.0 [1]
	3-[[5-(3-Chlorophenyl)-1,3,4-oxadiazol-2-yl]sulfanyl]-1-benzothiophene 1,1-dioxide	IC50	10100.0 [1]
	3-[(5-Pyridin-2-yl-1,3,4-oxadiazol-2-yl)sulfanyl]-1-benzothiophene 1,1-dioxide	IC50	13200.0 [1]
	3-[[5-(3-Methoxyphenyl)-1,3,4-oxadiazol-2-yl]sulfanyl]-1-benzothiophene 1,1-dioxide	IC50	4300.0 [1]
	Methyl 4-[5-[(1,1-dioxo-1-benzothiophen-3-yl)sulfanyl]-1,3,4-oxadiazol-2-yl]benzoate	IC50	30000.0 [1]
	N-[4-[5-[(1,1-Dioxo-1-benzothiophen-3-yl)sulfanyl]-1,3,4-oxadiazol-2-yl]phenyl]acetamide	IC50	20400.0 [1]
	3-[(5-Cyclohexyl-1,3,4-oxadiazol-2-yl)sulfanyl]-1-benzothiophene 1,1-dioxide	IC50	7600.0 [1]
	4-[5-[(1,1-Dioxo-1-benzothiophen-3-yl)sulfanyl]-1,3,4-oxadiazol-2-yl]aniline	IC50	13800.0 [1]
	3-[[5-(2-Chlorophenyl)-1,3,4-oxadiazol-2-yl]sulfanyl]-1-benzothiophene 1,1-dioxide	IC50	7200.0 [1]
	3-[2,2-Difluoro-3-[(4-hydroxy-6-methoxy-7-methyl-3-oxo-1H-2-benzofuran-5-yl)methyl]-1-methylcyclopropyl]propanoic acid	IC50	2600.0 [1]
	3-[2,2-Dibromo-3-[(4-hydroxy-6-methoxy-7-methyl-3-oxo-1H-2-benzofuran-5-yl)methyl]-1-methylcyclopropyl]propanoic acid	IC50	3100.0 [1]
	1-Cyclopropane Mycophenolic Acid	IC50	1100.0 [1]
	5-[[(2-Carboxyethyl)thio]methyl]-1,3-dihydro-4-hydroxy-6-methoxy-7-methylisobenzofuran-3-one	IC50	10900.0 [1]
	4-(4-Hydroxy-6-methoxy-7-methyl-3-oxo-1,3-dihydro-isobenzofuran-5-ylmethylsulfanyl)-butyric acid	IC50	22700.0 [1]
	5-(5-Carboxy-2-pentyn-1-yl)-1,3-dihydro-4-hydroxy-6-methoxy-7-methylisobenzofuran-3-one	IC50	2600.0 [1]
	5-(6-Carboxy-2-hexyn-1-yl)-1,3-dihydro-4-hydroxy-6-methoxy-7-methylisobenzofuran-3-one	IC50	2500.0 [1]
	CID 15625192	IC50	1200.0 [1]
	5-(5-Carboxypentyl)-1,3-dihydro-4-hydroxy-6-methoxy-7-methylisobenzofuran-3-one	IC50	940.0 [1]
	5-(6-Carboxyhexyl)-1,3-dihydro-4-hydroxy-6-methoxy-7-methylisobenzofuran-3-one	IC50	1800.0 [1]
	2-[[(E)-4-(6-Ethyl-4-hydroxy-7-methyl-3-oxo-1H-2-benzofuran-5-yl)-2-methylbut-2-enyl]amino]ethylphosphonic acid	IC50	37.0 [1]
	[(2S,3R,4S,5S)-5-(6-Aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-[[hydroxy-[2-(4-hydroxy-6-methoxy-7-methyl-3-oxo-1H-2-benzofuran-5-yl)ethoxy]phosphoryl]oxymethyl]phosphinic acid	Ki	20.0 [1]
	3-{5-[(1,1-Dioxido-1-benzothiophen-3-yl)sulfanyl]-1,3,4-oxadiazol-2-yl}pyridine	IC50	6300.0 [1]
	2-[(1,1-Dioxido-1-benzothiophen-3-yl)sulfanyl]-5-(2-methoxyphenyl)-1,3,4-oxadiazole	IC50	9900.0 [1]
	2-[(2R,3R,4S,5R)-5-[[[(2S,3R,4S,5S)-5-(6-Aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methylsulfamoylmethylsulfonylamino]methyl]-3,4-dihydroxyoxolan-2-yl]-1,3-thiazole-4-carboxamide	Ki	23600.0 [1]
	[[(2R,3S,4R,5R)-5-[6-Amino-2-(2-phenylethylamino)purin-9-yl]-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] [(2R,3S,4R,5R)-5-(4-carbamoyl-1,3-thiazol-2-yl)-3,4-dihydroxyoxolan-2-yl]methyl hydrogen phosphate	Ki	73.0 [1]
	[[(2R,3S,4R,5R)-5-(6-Amino-2-phenylpurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] [(2R,3S,4R,5R)-5-(4-carbamoyl-1,3-thiazol-2-yl)-3,4-dihydroxyoxolan-2-yl]methyl hydrogen phosphate	Ki	20.0 [1]
	[[(2R,3S,4R,5R)-5-(4-Carbamoyl-1,3-thiazol-2-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] [(2R,3S,4R,5R)-5-(2,6-diaminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methyl hydrogen phosphate	Ki	7.0 [1]
	[[(2R,3S,4R,5R)-5-(6-Amino-2-anilinopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] [(2R,3S,4R,5R)-5-(4-carbamoyl-1,3-thiazol-2-yl)-3,4-dihydroxyoxolan-2-yl]methyl hydrogen phosphate	Ki	45.0 [1]
	[[(2R,3S,4R,5R)-5-[6-Amino-2-(benzylamino)purin-9-yl]-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] [(2R,3S,4R,5R)-5-(4-carbamoyl-1,3-thiazol-2-yl)-3,4-dihydroxyoxolan-2-yl]methyl hydrogen phosphate	Ki	45.0 [1]
	[[(2R,3S,4R,5R)-5-(6-Amino-2-ethenylpurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] [(2R,3S,4R,5R)-5-(4-carbamoyl-1,3-thiazol-2-yl)-3,4-dihydroxyoxolan-2-yl]methyl hydrogen phosphate	Ki	96.0 [1]
	N-Hydroxy-6-(4-hydroxy-6-methoxy-7-methyl-3-oxo-1H-2-benzofuran-5-yl)-4-methylhexanamide	Ki	2070.0 [1]
	(E)-N-Hydroxy-7-(4-hydroxy-6-methoxy-7-methyl-3-oxo-1H-2-benzofuran-5-yl)-5-methylhept-5-enamide	Ki	400.0 [1]
	(E)-N-(2-Aminophenyl)-6-(4-hydroxy-6-methoxy-7-methyl-3-oxo-1H-2-benzofuran-5-yl)-4-methylhex-4-enamide	Ki	2830.0 [1]
	(E)-N-Hydroxy-3-[4-[[[3-methoxy-4-(1,3-oxazol-5-yl)phenyl]carbamoylamino]methyl]phenyl]prop-2-enamide	Ki	7800.0 [1]
	(E)-3-[4-[[(4-Cyano-3-methoxyphenyl)carbamoylamino]methyl]phenyl]-N-hydroxyprop-2-enamide	Ki	100000.0 [1]
	(E)-N-Hydroxy-3-[3-[[[3-methoxy-4-(1,3-oxazol-5-yl)phenyl]carbamoylamino]methyl]phenyl]prop-2-enamide	Ki	2300.0 [1]
	(E)-3-[3-[[(4-Cyano-3-methoxyphenyl)carbamoylamino]methyl]phenyl]-N-hydroxyprop-2-enamide	Ki	44000.0 [1]
	6-(4-Methoxy-3-(oxazol-5-yl)phenyl)-4-methylhex-4-enoic acid	Ki	20800.0 [1]
	6-(2,4-Dimethoxy-5-(oxazol-5-yl)phenyl)-4-methylhex-4-enoic acid	Ki	16000.0 [1]
	7-Methoxy-6-oxazol-5-yl-2-m-tolyl-1H-quinolin-4-one	IC50	150.0 [1]
	2-(3,4-Dimethyl-phenyl)-7-methoxy-6-oxazol-5-yl-1H-quinolin-4-one	IC50	83.0 [1]
	[(E)-4-(6-Ethyl-4-hydroxy-7-methyl-3-oxo-1H-2-benzofuran-5-yl)-2-methylbut-2-enyl]phosphonic acid	IC50	71.0 [1]
	[[(3R,4S)-5-(6-Aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl]oxymethyl-[2-(4-hydroxy-6-methoxy-7-methyl-3-oxo-1H-2-benzofuran-5-yl)ethoxy]phosphinic acid	Ki	87.0 [1]
	[(3R,4S)-5-(6-Aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-[[hydroxy-[2-(4-hydroxy-6-methoxy-7-methyl-3-oxo-1H-2-benzofuran-5-yl)ethoxy]phosphoryl]oxymethyl]phosphinic acid	Ki	20.0 [1]
	2-[[(2S,3R,4S,5R)-5-[[[(2R,3S,4R,5R)-5-(6-Aminopurin-7-yl)-3,4-dihydroxyoxolan-2-yl]methylsulfamoylmethylsulfonylamino]methyl]-3,4-dihydroxyoxolan-2-yl]methyl]-1,3-thiazole-4-carboxamide	IC50	23600.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 100 ⟨⟩

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References

This online tool may be cited as follows

MLA	"Quest Database™ Inosine-5'-monophosphate dehydrogenase 1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/inosine-5-monophosphate-dehydrogenase-1-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, May 9). Quest Database™ Inosine-5'-monophosphate dehydrogenase 1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/inosine-5-monophosphate-dehydrogenase-1-inhibitors-ic50-ki.
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