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Integrin alpha-2/beta-3 Inhibitors (IC50, Ki)

Structure
Compound Name
Standard Type
Standard Values (in nM)
Arg-gly-asp-serIC5013000.0 [1]
3-[[3-Oxo-2-(2-piperidin-4-ylethyl)-1H-isoindole-5-carbonyl]amino]propanoic acidIC5025.0 [1]
3-(3-(Carbamoyl)benzamido)-3-(4-methoxyphenyl)propanoic acidIC500.8 [1]
3-(3-(Carbamoyl)benzamido)-3-(3,4-dimethoxyphenyl)propanoic acidIC500.7 [1]
3-(3-(Carbamoyl)benzamido)-3-phenylpropanoic acidIC501.0 [1]
3-(3-(Carbamoyl)benzamido)propanoic acidIC509.0 [1]
3-[[3-Nitro-5-(1,2,3,4-tetrahydroisoquinolin-7-ylcarbamoyl)benzoyl]amino]propanoic acidIC5032.0 [1]
3-[[3-Nitro-5-(1,2,3,4-tetrahydroisoquinolin-7-ylcarbamoyl)benzoyl]amino]-3-phenylpropanoic acidIC508.0 [1]
3-(4-Methoxyphenyl)-3-[[3-nitro-5-(1,2,3,4-tetrahydroisoquinolin-7-ylcarbamoyl)benzoyl]amino]propanoic acidIC505.0 [1]
3-(3,4-Dimethoxyphenyl)-3-[[3-nitro-5-(1,2,3,4-tetrahydroisoquinolin-7-ylcarbamoyl)benzoyl]amino]propanoic acidIC503.7 [1]
3-[3-Oxo-5-(4-piperidin-4-ylbutanoylamino)-1H-isoindol-2-yl]butanoic acidIC50350.0 [1]
3-[3-Oxo-5-[(4-piperazin-1-ylbenzoyl)amino]-1H-isoindol-2-yl]butanoic acidIC5037.0 [1]
3-[3-Oxo-5-[(4-piperidin-4-ylbenzoyl)amino]-1H-isoindol-2-yl]propanoic acidIC506.8 [1]
3-[3-Oxo-5-(1,2,3,4-tetrahydroisoquinoline-7-carbonylamino)-1H-isoindol-2-yl]propanoic acidIC506.5 [1]
3-[3-Oxo-5-(1,2,3,4-tetrahydroisoquinoline-7-carbonylamino)-1H-isoindol-2-yl]butanoic acidIC506.5 [1]
3-[3-Oxo-5-(4-piperidin-4-ylbutanoylamino)-1H-isoindol-2-yl]propanoic acidIC505.5 [1]
2-[3-Oxo-5-[(4-piperidin-4-ylbenzoyl)amino]-1H-isoindol-2-yl]acetic acidIC50270.0 [1]
2-[3-Oxo-5-(1,2,3,4-tetrahydroisoquinoline-7-carbonylamino)-1H-isoindol-2-yl]acetic acidIC501200.0 [1]
3-[3-(1,2,3,4-Tetrahydroisoquinoline-7-carbonylamino)propanoylamino]propanoic acidIC5022.0 [1]



References

This online tool may be cited as follows

MLA

"Quest Database™ Integrin alpha-2/beta-3 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.9 May2024https://www.aatbio.com/data-sets/integrin-alpha-2-beta-3-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024May 9). Quest Database™ Integrin alpha-2/beta-3 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/integrin-alpha-2-beta-3-inhibitors-ic50-ki.
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