Structure | Compound Name | Standard Type | Standard Values (in nM) |
|---|---|---|---|
| (2S)-1-[(2S)-2-[[(2S)-3-Carboxy-2-[[(2S)-4-methyl-2-[[2-[4-[(2-methylphenyl)carbamoylamino]phenyl]acetyl]amino]pentanoyl]amino]propanoyl]amino]-3-methylbutanoyl]pyrrolidine-2-carboxylic acid | IC50 | 0.5 [1] | |
| (3S,6R,11R,14S)-6-[[(2S)-2-Acetamido-3-(4-hydroxyphenyl)propanoyl]amino]-3-(carboxymethyl)-2,5,13-trioxo-8,9-dithia-1,4,12-triazabicyclo[12.3.0]heptadecane-11-carboxylic acid | IC50 | 2.0 [1], 3.0 [2], 200.0 [3], 300.0 [4] | |
| (S)-2-(2-Chloro-6-methyl-benzoylamino)-3-[4-(2,6-dichloro-benzoylamino)-phenyl]-propionic acid | IC50 | 0.3 [1], 10.0 [2], 12.0 [3] | |
| (2S)-2-[[(3S)-2-(3,4-Dimethoxyphenyl)sulfonyl-3,4-dihydro-1H-isoquinoline-3-carbonyl]amino]hexanoic acid | IC50 | 0.53 [1], 58.0 [2] | |
| (2S)-2-[[(2S)-1-(3,5-Dichlorophenyl)sulfonylpyrrolidine-2-carbonyl]amino]-3-[4-[(3,5-dichloropyridine-4-carbonyl)amino]phenyl]propanoic acid | IC50 | 0.03 [1], 0.07 [2], 0.1 [3] | |
MLA | "Quest Database™ Integrin alpha-4/beta-1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 11 Feb. 2026, https://www.aatbio.com/data-sets/integrin-alpha-4-beta-1-inhibitors-ic50-ki. | |
APA | AAT Bioquest, Inc. (2026, February 11). Quest Database™ Integrin alpha-4/beta-1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/integrin-alpha-4-beta-1-inhibitors-ic50-ki. | |
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