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Interleukin-8 receptor A Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
NavarixinIC503.9 [1], 36.0 [2]
NavarixinKi18.0 [1], 20.0 [2]
SporanoxIC50158.49 [1], 5011.87 [2], 19952.62 [3]
ClotrimazoleIC501995.26 [1], 7943.28 [2], 10000.0 [3]
(R)-3-(3,4-Dioxo-2-(1-phenylpropylamino)cyclobut-1-enylamino)-2-hydroxy-N,N-dimethylbenzamideIC50254.0 [1]
(R)-3-(3,4-Dioxo-2-(1-phenylpropylamino)cyclobut-1-enylamino)-2-hydroxy-N,N-dimethylbenzamideKi40.0 [1]
QuercetinIC505011.87 [1], 100000.0 [2]
DiclofenacIC5012.0 [1], 10000.0 [2]
1-(2-Bromophenyl)-3-(2-hydroxy-4-nitrophenyl)ureaIC5022.0 [1], 3000.0 [2]
CID 46897162IC50880.0 [1], 903.0 [2]
[2-[[5-[(4-Fluorophenyl)carbamoyl]pyridin-2-yl]sulfanylmethyl]-4-(trifluoromethoxy)phenyl]boronic acidIC5031.0 [1]
3-[[3,4-Dioxo-2-[[(1R)-1-thiophen-2-ylpropyl]amino]cyclobuten-1-yl]amino]-2-hydroxy-N,N-dimethylbenzamideIC5081.0 [1]
3-[[3,4-Dioxo-2-[[(1R)-1-thiophen-2-ylpropyl]amino]cyclobuten-1-yl]amino]-2-hydroxy-N,N-dimethylbenzamideKi210.0 [1]
2-Hydroxy-N,N-dimethyl-3-[[2-[[(1R)-1-(5-methylthiophen-2-yl)propyl]amino]-3,4-dioxocyclobuten-1-yl]amino]benzamideIC50235.0 [1]
2-Hydroxy-N,N-dimethyl-3-[[2-[[(1R)-1-(5-methylthiophen-2-yl)propyl]amino]-3,4-dioxocyclobuten-1-yl]amino]benzamideKi146.0 [1]
3-(4-Chlorophenyl)-5-[4-[3-(4-methylpiperazin-1-yl)propoxy]phenyl]-1,2-oxazoleIC502100.0 [1], 3600.0 [2]
3-(4-Chlorophenyl)-5-[4-[3-(4-methylpiperazin-1-yl)propoxy]phenyl]-1,2,4-oxadiazoleIC502500.0 [1], 4500.0 [2]
3-[[4-[[(1R)-2,2-Dimethyl-1-(5-methylfuran-2-yl)propyl]amino]-1,2,5-thiadiazol-3-yl]amino]-2-hydroxy-N,N-dimethylbenzamideIC50143.0 [1]
3-[[4-[[(1R)-2,2-Dimethyl-1-(5-methylfuran-2-yl)propyl]amino]-1,2,5-thiadiazol-3-yl]amino]-2-hydroxy-N,N-dimethylbenzamideKi14.0 [1]
2-Hydroxy-N,N-dimethyl-3-[[4-[[(1R)-2-methyl-1-(5-methylfuran-2-yl)propyl]amino]-1,2,5-thiadiazol-3-yl]amino]benzamideIC503910.0 [1]
2-Hydroxy-N,N-dimethyl-3-[[4-[[(1R)-2-methyl-1-(5-methylfuran-2-yl)propyl]amino]-1,2,5-thiadiazol-3-yl]amino]benzamideKi15.0 [1]
3-[[2-[[(1R)-1-(4-Bromofuran-2-yl)propyl]amino]-3,4-dioxocyclobuten-1-yl]amino]-2-hydroxy-N,N-dimethylbenzamideIC5055.0 [1], 917.0 [2]
{4-[5-(4-Fluoro-phenyl)-isoxazol-3-yl]-phenoxymethyl}-dimethyl-amineIC503100.0 [1], 4000.0 [2]
3-(4-Hydroxy-2,6-diiodophenyl)-3-(4-hydroxy-3,5-diiodophenyl)-2-benzofuran-1-oneIC501995.26 [1], 100000.0 [2]
3-(4-Fluorophenyl)-5-[4-[3-(4-methylpiperazin-1-yl)propoxy]phenyl]-1,2-oxazoleIC502000.0 [1], 3800.0 [2]
ReparixinIC501.0 [1]
(S)-N1-((1H-Benzo[d]imidazol-2-yl)methyl)-N1-(5,6,7,8-tetrahydroquinolin-8-yl)butane-1,4-diamineIC5010000.0 [1]
2-Hydroxy-N,N-dimethyl-3-[[2-[1-(5-methylfuran-2-yl)propylamino]-3,4-dioxocyclobuten-1-yl]amino]benzamideIC5099.0 [1]
DanirixinIC5030000.0 [1]
ElubrixinIC5010000.0 [1]
CID 46861584IC5010000.0 [1]
1-[(1R,2S)-2-[[(3S)-3-[(4-Fluorophenyl)methyl]piperidin-1-yl]methyl]cyclohexyl]-3-[3-(1-methyltetrazol-5-yl)phenyl]ureaIC5010000.0 [1]
1-(2-Hydroxy-4-nitrophenyl)-3-phenylureaIC5018200.0 [1]
1-((1R,2S)-2-(((S)-3-(4-Fluorobenzyl)piperidin-1-yl)methyl)cyclohexyl)-3-(3-acetylphenyl)ureaIC5010000.0 [1]
3-[[3,4-Dioxo-2-[[(1R)-1-(4-propan-2-ylfuran-2-yl)propyl]amino]cyclobuten-1-yl]amino]-2-hydroxy-N,N-dimethylbenzamideIC507.3 [1]
3-[[2-[[(1R)-1-(3-Fluorophenyl)propyl]amino]-3,4-dioxocyclobuten-1-yl]amino]-2-hydroxy-N,N-dimethylbenzamideIC50197.0 [1]
1-(1,3-Dimethyl-1H-pyrazolo[3,4-b]pyridine-5-carbonyl)-3-(4-fluoro-3-(trifluoromethyl)phenyl)ureaIC5010000.0 [1]
1-(4-Cyano-2-hydroxyphenyl)-3-phenylureaIC5021000.0 [1]
CCR3 AntagonistIC5010000.0 [1]
(8S)-N-(1H-Benzimidazol-2-ylmethyl)-N-[[4-[(pyridin-2-ylmethylamino)methyl]phenyl]methyl]-5,6,7,8-tetrahydroquinolin-8-amineIC5010000.0 [1]
1-(2-Bromophenyl)-3-(4-cyano-2-hydroxyphenyl)ureaIC5015100.0 [1]
1-(3-Bromo-4-cyano-2-hydroxyphenyl)-3-(2-bromophenyl)ureaIC502600.0 [1]
3-[[3,4-Dioxo-2-(pentan-3-ylamino)cyclobuten-1-yl]amino]-2-hydroxy-N,N-dimethylbenzamideIC50910.0 [1]
3-[[2-[[(1R)-1-(4-Cyclohexylfuran-2-yl)propyl]amino]-3,4-dioxocyclobuten-1-yl]amino]-2-hydroxy-N,N-dimethylbenzamideKi283.0 [1]
1-[4-Chloro-2-hydroxy-3-[(3S)-3-methyloxolan-3-yl]sulfonylphenyl]-3-[(1R)-2-methylcyclopent-2-en-1-yl]ureaIC503800.0 [1]
3-[[2-[[(1S)-2,2-Difluoro-1-(5-methylfuran-2-yl)propyl]amino]-3,4-dioxocyclobuten-1-yl]amino]-2-hydroxy-N,N-dimethylbenzamideKi6.0 [1]
(R)-3-(2-(1-(Furan-2-yl)propylamino)-3,4-dioxocyclobut-1-enylamino)-2-hydroxy-N,N-dimethylbenzamideIC5026.0 [1]
2-Hydroxy-N,N-dimethyl-3-[[2-[[(1R)-1-(4-methylfuran-2-yl)propyl]amino]-3,4-dioxocyclobuten-1-yl]amino]benzamideKi9.0 [1]
3-(4-Fluorophenyl)-5-[4-[3-(4-methylpiperazin-1-yl)propoxy]phenyl]-1,2,4-oxadiazoleIC5010500.0 [1]
3-(3-Chlorophenyl)-5-[4-[3-(4-methylpiperazin-1-yl)propoxy]phenyl]-1,2-oxazoleIC509600.0 [1]
3-[[3,4-Dioxo-2-[[(1R)-1-phenylpropyl]amino]cyclobuten-1-yl]amino]-2-hydroxy-N-methyl-N-propan-2-ylbenzamideKi123.0 [1]
3-[[2-[[(1S)-2,2-Difluoro-1-(4-methylfuran-2-yl)propyl]amino]-3,4-dioxocyclobuten-1-yl]amino]-2-hydroxy-N,N-dimethylbenzamideKi6.0 [1]
3-[2-Hydroxy-3-[(3S)-3-hydroxypyrrolidine-1-carbonyl]anilino]-4-[[(1R)-1-phenylpropyl]amino]cyclobut-3-ene-1,2-dioneKi21.0 [1]
3-[2-Hydroxy-3-(4-methylpiperazine-1-carbonyl)anilino]-4-[[(1R)-1-phenylpropyl]amino]cyclobut-3-ene-1,2-dioneKi41.0 [1]
3-[[2-[[(1R)-1-(4-Ethylfuran-2-yl)propyl]amino]-3,4-dioxocyclobuten-1-yl]amino]-2-hydroxy-N,N-dimethylbenzamideKi7.0 [1]
3-[[3,4-Dioxo-2-[[(1S)-2,2,2-trifluoro-1-(5-methylfuran-2-yl)ethyl]amino]cyclobuten-1-yl]amino]-2-hydroxy-N,N-dimethylbenzamideKi9.0 [1]
3-[[2-[[(R)-Cyclopropyl-(4-propan-2-ylfuran-2-yl)methyl]amino]-3,4-dioxocyclobuten-1-yl]amino]-2-hydroxy-N,N-dimethylbenzamideKi10.0 [1]
2-Hydroxy-N,N-dimethyl-3-[[2-[[(1R)-2-methyl-1-(4-propan-2-ylfuran-2-yl)propyl]amino]-3,4-dioxocyclobuten-1-yl]amino]benzamideKi11.0 [1]
3-[4-[3-(4-Chlorophenyl)-1,2-oxazol-5-yl]phenoxy]-N,N-dimethylpropan-1-amineIC503900.0 [1]
5-[4-[3-(4-Methylpiperazin-1-yl)propoxy]phenyl]-3-phenyl-1,2-oxazoleIC503000.0 [1]
3-(2-(1-(Furan-2-yl)propylamino)-3,4-dioxocyclobut-1-enylamino)-2-hydroxy-N,N-dimethylbenzamideIC5067.0 [1]
3-(3,4-Dioxo-2-(1-(thiophen-2-yl)propylamino)cyclobut-1-enylamino)-2-hydroxy-N,N-dimethylbenzamideIC50179.0 [1]
5-[4-[3-(4-Methylpiperazin-1-yl)propoxy]phenyl]-3-(4-phenoxyphenyl)-1,2-oxazoleIC5022700.0 [1]
3-[[2-[[(1R)-1-(4-Tert-butylfuran-2-yl)propyl]amino]-3,4-dioxocyclobuten-1-yl]amino]-2-hydroxy-N,N-dimethylbenzamideKi10.0 [1]
3-[[2-[[(1R)-1-(4-Cyclopentylfuran-2-yl)propyl]amino]-3,4-dioxocyclobuten-1-yl]amino]-2-hydroxy-N,N-dimethylbenzamideKi53.0 [1]
3-[[3,4-Dioxo-2-[[(1S)-2,2,2-trifluoro-1-(4-propan-2-ylfuran-2-yl)ethyl]amino]cyclobuten-1-yl]amino]-2-hydroxy-N,N-dimethylbenzamideKi16.0 [1]
3-[[2-[[(1R)-1-(4-Butylfuran-2-yl)propyl]amino]-3,4-dioxocyclobuten-1-yl]amino]-2-hydroxy-N,N-dimethylbenzamideKi34.0 [1]
2-Hydroxy-N,N-dimethyl-3-[[2-[[(1R)-1-[4-(4-morpholin-4-ylbutyl)furan-2-yl]propyl]amino]-3,4-dioxocyclobuten-1-yl]amino]benzamideKi14.0 [1]
[(3S,5R,6S,7S,10R,11R,13R,14R,17R)-6,7-Diacetyloxy-5,11-dihydroxy-10,13-dimethyl-17-[(2R)-6-methylheptan-2-yl]-1,2,3,4,6,7,11,12,14,15,16,17-dodecahydrocyclopenta[a]phenanthren-3-yl] acetateIC505500.0 [1]
[(3S,5R,6S,7S,10R,11R,13R,14R,17R)-6-Acetyloxy-3,5,11-trihydroxy-10,13-dimethyl-17-[(2R)-6-methylheptan-2-yl]-1,2,3,4,6,7,11,12,14,15,16,17-dodecahydrocyclopenta[a]phenanthren-7-yl] acetateIC5020000.0 [1]
3-[(2-Chlorophenyl)amino]-7-nitro-4H-1,2,4-benzothiadiazin-5-ol 1,1-dioxideIC5012000.0 [1]
1-(2-Bromophenyl)-3-(3-chloro-4-cyano-2-hydroxyphenyl)ureaIC504200.0 [1]
7-Nitro-3-{[2-(phenyloxy)phenyl]amino}-4H-1,2,4-benzothiadiazin-5-ol 1,1-dioxideIC507600.0 [1]
7-Chloro-3-(2-chloroanilino)-1,1-dioxo-4H-1lambda6,2,4-benzothiadiazin-5-olIC5024000.0 [1]
1-(2-Hydroxy-3-nitro-phenyl)-3-phenyl-ureaIC5033200.0 [1]
3-[(2-Bromophenyl)amino]-7-nitro-4H-1,2,4-benzothiadiazin-5-ol 1,1-dioxideIC503200.0 [1]
[(1R,2S,5S,7R,8S,11R,14R,15R,17R)-5,7-Dihydroxy-2,15-dimethyl-14-[(2R)-6-methylheptan-2-yl]-18-oxapentacyclo[8.8.0.01,17.02,7.011,15]octadec-9-en-8-yl] acetateIC504500.0 [1]
1-(2-Hydroxy-5-nitro-phenyl)-3-phenyl-ureaIC5046200.0 [1]
[3-[[[5-[(4-Fluorophenyl)carbamoyl]pyridin-2-yl]amino]methyl]phenyl]boronic acidIC50611.0 [1]
[3-[[[5-[(4-Fluorophenyl)carbamoyl]pyridin-2-yl]-methylamino]methyl]phenyl]boronic acidIC504100.0 [1]
[4-[[[5-[(4-Fluorophenyl)carbamoyl]pyridin-2-yl]amino]methyl]phenyl]boronic acidIC504300.0 [1]
[6-[[[5-[(4-Fluorophenyl)carbamoyl]pyridin-2-yl]-methylamino]methyl]pyridin-3-yl]boronic acidIC501700.0 [1]
[2-[[[5-[(4-Fluorophenyl)carbamoyl]pyrimidin-2-yl]-methylamino]methyl]phenyl]boronic acidIC505000.0 [1]
[3-[[[5-[(4-Fluorophenyl)carbamoyl]pyrimidin-2-yl]amino]methyl]phenyl]boronic acidIC501340.0 [1]
[3-[[[5-[(4-Fluorophenyl)carbamoyl]pyrimidin-2-yl]-methylamino]methyl]phenyl]boronic acidIC502500.0 [1]
[4-[[[5-[(4-Fluorophenyl)carbamoyl]pyrimidin-2-yl]amino]methyl]phenyl]boronic acidIC501700.0 [1]
[6-[[[5-[(4-Fluorophenyl)carbamoyl]pyrimidin-2-yl]-methylamino]methyl]pyridin-3-yl]boronic acidIC501700.0 [1]
[6-[[Benzyl-[5-[(4-fluorophenyl)carbamoyl]pyridin-2-yl]amino]methyl]pyridin-3-yl]boronic acidIC50326.0 [1]
[6-[[[5-[(4-Fluorophenyl)carbamoyl]pyridin-2-yl]-(pyridin-2-ylmethyl)amino]methyl]pyridin-3-yl]boronic acidIC505000.0 [1]
[6-[[[5-[(4-Fluorophenyl)carbamoyl]pyridin-2-yl]-(oxan-4-ylmethyl)amino]methyl]pyridin-3-yl]boronic acidIC505000.0 [1]
[6-[[[5-[(4-Fluorophenyl)carbamoyl]pyridin-2-yl]-(furan-2-ylmethyl)amino]methyl]pyridin-3-yl]boronic acidIC503.3 [1]
2-[(5-Boronopyridin-2-yl)methyl-[5-[(4-fluorophenyl)carbamoyl]pyrimidin-2-yl]amino]acetic acidIC505000.0 [1]
[6-[[Benzyl-[5-[(4-fluorophenyl)carbamoyl]pyrimidin-2-yl]amino]methyl]pyridin-3-yl]boronic acidIC507.0 [1]
[6-[[[5-[(4-Fluorophenyl)carbamoyl]pyrimidin-2-yl]-(pyridin-2-ylmethyl)amino]methyl]pyridin-3-yl]boronic acidIC502050.0 [1]
[6-[[2-Aminoethyl-[5-[(4-fluorophenyl)carbamoyl]pyrimidin-2-yl]amino]methyl]pyridin-3-yl]boronic acidIC505000.0 [1]
[6-[[[5-[(4-Fluorophenyl)carbamoyl]pyrimidin-2-yl]-(furan-2-ylmethyl)amino]methyl]pyridin-3-yl]boronic acidIC50444.0 [1]
3-[[4-[(1R)-1-(1,3-Benzodioxol-5-yl)-2,2-dimethylpropyl]imino-1,1-dioxo-1,2,5-thiadiazol-3-yl]amino]-2-hydroxy-N,N-dimethylbenzamideKi46.0 [1]
3-[[1,1-Dioxo-4-[(1R)-1-phenylpropyl]imino-1,2,5-thiadiazol-3-yl]amino]-2-hydroxy-N,N-dimethylbenzamideKi8990.0 [1]
2-Hydroxy-N,N-dimethyl-3-[[4-[(1R)-1-(5-methylfuran-2-yl)propyl]imino-1,1-dioxo-1,2,5-thiadiazol-3-yl]amino]benzamideKi5950.0 [1]
3-[[4-[(1R)-1-(Furan-2-yl)-2,2-dimethylpropyl]imino-1,1-dioxo-1,2,5-thiadiazol-3-yl]amino]-2-hydroxy-N,N-dimethylbenzamideKi61.0 [1]
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References

This online tool may be cited as follows

MLA

"Quest Database™ Interleukin-8 receptor A Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/interleukin-8-receptor-a-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 9). Quest Database™ Interleukin-8 receptor A Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/interleukin-8-receptor-a-inhibitors-ic50-ki.
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