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Isoleucyl-tRNA synthetase Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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[(2R,3S,4R,5R)-3,4-Dihydroxy-5-(4-phenyl-1,3-thiazol-2-yl)oxolan-2-yl]methyl N-[(2S,3S)-2-amino-3-methylpentanoyl]sulfamateIC50100.0 [1], 330.0 [2]
[(2R,3S,4R,5R)-3,4-Dihydroxy-5-[4-(4-phenoxyphenyl)-1,3-thiazol-2-yl]oxolan-2-yl]methyl N-[(2S)-2-amino-3-methylpentanoyl]sulfamateIC5045.0 [1], 370.0 [2]
[(2R,3S,4R,5R)-3,4-Dihydroxy-5-[4-(3-methoxyphenyl)-1,3-thiazol-2-yl]oxolan-2-yl]methyl N-[(2S)-2-amino-3-methylpentanoyl]sulfamateIC5015.0 [1], 34.0 [2]
[(2R,3S,4R,5R)-3,4-Dihydroxy-5-[4-(2-methoxyphenyl)-1,3-thiazol-2-yl]oxolan-2-yl]methyl N-[(2S)-2-amino-3-methylpentanoyl]sulfamateIC5030.0 [1], 100.0 [2]
[(2R,3S,4R,5R)-3,4-Dihydroxy-5-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]oxolan-2-yl]methyl N-[(2S)-2-amino-3-methylpentanoyl]sulfamateIC50100.0 [1], 200.0 [2]
[(2R,3S,4R,5R)-3,4-Dihydroxy-5-[4-(6-methoxynaphthalen-2-yl)-1,3-thiazol-2-yl]oxolan-2-yl]methyl N-[(2S)-2-amino-3-methylpentanoyl]sulfamateIC5020.0 [1], 400.0 [2]
[(2R,3S,4R,5R)-3,4-Dihydroxy-5-[4-[2-(4-phenoxyphenyl)ethyl]-1,3-thiazol-2-yl]oxolan-2-yl]methyl N-[(2S)-2-amino-3-methylpentanoyl]sulfamateIC50110.0 [1], 1020.0 [2]
[(2R,3S,4R,5R)-5-[4-(4-Cyanofuran-2-yl)-1,3-thiazol-2-yl]-3,4-dihydroxyoxolan-2-yl]methyl N-[(2S)-2-amino-3-methylpentanoyl]sulfamateIC50120.0 [1]
[(2R,3S,4R,5R)-3,4-Dihydroxy-5-[4-(2-phenylethyl)-1,3-thiazol-2-yl]oxolan-2-yl]methyl N-[(2S)-2-amino-3-methylpentanoyl]sulfamateIC5030.0 [1], 300.0 [2]
MupirocinIC500.8 [1]
Aminoacyl tRNA synthetase-IN-1IC5098.0 [1]
[(2R,3S,4R,5S)-5-[(6-Aminopurin-9-yl)methyl]-3,4-dihydroxyoxolan-2-yl]methyl (2S,3S)-2-amino-3-methylpentanoateIC50128000.0 [1]
(2S,3S)-2-Amino-N-[[(2R,3S,4R,5S)-5-[(6-aminopurin-9-yl)methyl]-3,4-dihydroxyoxolan-2-yl]methyl]-N-hydroxy-3-methylpentanamideIC50128000.0 [1]
2-[Hydroxy-(3-hydroxy-4-methoxybenzoyl)amino]ethyl (2S)-2-amino-3-methylpentanoateIC504500.0 [1]
[(4R)-2-(4-Hydroxy-3-methoxyphenyl)-4,5-dihydro-1,3-oxazol-4-yl]methyl (2S)-2-amino-3-methylpentanoateIC5050000.0 [1]
[3-(4-Hydroxy-3-methoxyphenyl)-4,5-dihydro-1,2-oxazol-5-yl]methyl (2S)-2-amino-3-methylpentanoateIC5079000.0 [1]
[(4S)-2-(4-Hydroxy-3-methoxyphenyl)-4,5-dihydro-1,3-oxazol-4-yl]methyl (2S)-2-amino-3-methylpentanoateIC5038600.0 [1]
[(2R,3S,4R,5R)-3,4-Dihydroxy-5-(4-phenyl-1,3-thiazol-2-yl)oxolan-2-yl]methyl N-[(2S)-2-amino-3-phenylpropanoyl]sulfamateIC50100000.0 [1]
[(2R,3S,4R,5R)-3,4-Dihydroxy-5-(4-phenyl-1,3-thiazol-2-yl)oxolan-2-yl]methyl N-[(2S)-2-aminopropanoyl]sulfamateIC50100000.0 [1]
[(2R,3S,4R,5R)-3,4-Dihydroxy-5-(4-phenyl-1,3-thiazol-2-yl)oxolan-2-yl]methyl N-[(2S)-2-amino-3-(1H-imidazol-5-yl)propanoyl]sulfamateIC50100000.0 [1]
[(2R,3S,4R,5R)-3,4-Dihydroxy-5-(4-phenyl-1,3-thiazol-2-yl)oxolan-2-yl]methyl N-[(2S)-2-amino-3-methylbutanoyl]sulfamateIC5015000.0 [1]
(2S,3S)-2-Amino-N-[[(2R,3S,4R,5R)-5-(6-aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methyl]-N-hydroxy-3-methylpentanamideIC50181000.0 [1]
[(2R,3S,4R,5S)-5-[2-(6-Aminopurin-9-yl)ethyl]-3,4-dihydroxyoxolan-2-yl]methyl (2S,3S)-2-amino-3-methylpentanoateIC50128000.0 [1]
(2S,3S)-2-Amino-N-[[(2R,3S,4R,5S)-5-[2-(6-aminopurin-9-yl)ethyl]-3,4-dihydroxyoxolan-2-yl]methyl]-N-hydroxy-3-methylpentanamideIC50128000.0 [1]
(2S,3S)-2-Amino-N-[[(2R,3S,4R,5S)-3,4-dihydroxy-5-[2-(5-phenyltetrazol-2-yl)ethyl]oxolan-2-yl]methyl]-N-hydroxy-3-methylpentanamideIC50128000.0 [1]
[(2R,3S,4R,5S)-5-[2-[6-(Benzylamino)purin-9-yl]ethyl]-3,4-dihydroxyoxolan-2-yl]methyl (2S,3S)-2-amino-3-methylpentanoateIC5084000.0 [1]
(2S,3S)-2-Amino-N-[[(2R,3S,4R,5S)-5-[2-[6-(benzylamino)purin-9-yl]ethyl]-3,4-dihydroxyoxolan-2-yl]methyl]-N-hydroxy-3-methylpentanamideIC50128000.0 [1]
2-[Hydroxy-[2-(4-hydroxy-3-methoxyphenyl)acetyl]amino]ethyl (2S)-2-amino-3-methylpentanoateIC50228000.0 [1]
[3-(3-Hydroxy-4-methoxyphenyl)-4,5-dihydro-1,2-oxazol-5-yl]methyl (2S)-2-amino-3-methylpentanoateIC5057600.0 [1]
2-[[2-(4-Hydroxy-3-methoxyphenyl)acetyl]amino]ethyl (2S)-2-amino-3-methylpentanoateIC5045000.0 [1]
2-[Hydroxy-(4-hydroxy-3-methoxybenzoyl)amino]ethyl (2S)-2-amino-3-methylpentanoateIC5012800.0 [1]
2-[(3-Hydroxy-4-methoxybenzoyl)amino]ethyl (2S)-2-amino-3-methylpentanoateIC50106000.0 [1]
2-[Hydroxy-[2-(3-hydroxy-4-methoxyphenyl)acetyl]amino]ethyl (2S)-2-amino-3-methylpentanoateIC5021000.0 [1]
[(2R,3S,4R,5R)-5-(6-Aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methyl (2S,3S)-2-amino-3-methylpentanoateIC50183000.0 [1]
[(2R,3S,4R,5S)-3,4-Dihydroxy-5-[2-(5-phenyltetrazol-2-yl)ethyl]oxolan-2-yl]methyl (2S,3S)-2-amino-3-methylpentanoateIC5063600.0 [1]
2-[[2-(3-Hydroxy-4-methoxyphenyl)acetyl]amino]ethyl (2S)-2-amino-3-methylpentanoateIC5056500.0 [1]
2-[(4-Hydroxy-3-methoxybenzoyl)amino]ethyl (2S)-2-amino-3-methylpentanoateIC5064400.0 [1]
[(2R,3S,4R)-5-(6-Amino-2-iodopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methyl N-[(2S,3S)-2-amino-3-methylpentanoyl]sulfamateIC5014.0 [1]
[(2R,3S,4R)-5-(6-Amino-2-chloropurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methyl N-[(2S,3S)-2-amino-3-methylpentanoyl]sulfamateIC505500.0 [1]
(2S,3S)-2-Amino-N-[[(2R,3S,4R)-5-(6-aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxysulfamoyl]-3-methylpentanamideIC5012800.0 [1]
[(2R,3S,4R)-3,4-Dihydroxy-5-[2-iodo-6-(methylamino)purin-9-yl]oxolan-2-yl]methyl N-[(2S,3S)-2-amino-3-methylpentanoyl]sulfamateIC5022200.0 [1]
[(2R,3S,4R)-5-(6-Amino-2-ethynylpurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methyl N-[(2S,3S)-2-amino-3-methylpentanoyl]sulfamateIC5039.0 [1]
(2S,3S)-2-Amino-N-[[(2R,3S,4R)-5-(6-aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methyl-hydroxysulfamoyl]-3-methylpentanamideIC50132000.0 [1]
[(2R,3S,4R)-5-(6-Amino-2-hex-1-ynylpurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methyl N-[(2S,3S)-2-amino-3-methylpentanoyl]sulfamateIC501100.0 [1]
Methyl 9-[(E)-4-[(2S,3R,4R,5S)-5-(butylsulfonylamino)-3,4-dihydroxyoxan-2-yl]but-2-enoyl]oxynonanoateIC50300.0 [1]
Methyl 9-[(E)-4-[(2S,3R,4R,5S)-5-[(3-chlorophenyl)sulfonylamino]-3,4-dihydroxyoxan-2-yl]but-2-enoyl]oxynonanoateIC50300.0 [1]
Methyl 9-[(E)-4-[(2S,3R,4R,5S)-5-(3-chloropropylsulfonylamino)-3,4-dihydroxyoxan-2-yl]but-2-enoyl]oxynonanoateIC50100.0 [1]
Methyl 9-[(E)-4-[(2S,3R,4R,5S)-3,4-dihydroxy-5-(propylsulfonylamino)oxan-2-yl]but-2-enoyl]oxynonanoateIC503000.0 [1]
Methyl 9-[(E)-4-[(2S,3R,4R,5S)-3,4-dihydroxy-5-(methanesulfonamido)oxan-2-yl]but-2-enoyl]oxynonanoateIC5020000.0 [1]
Items per page: 1 - 10 of 49
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References

This online tool may be cited as follows

MLA

"Quest Database™ Isoleucyl-tRNA synthetase Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 8 May. 2024, https://www.aatbio.com/data-sets/isoleucyl-trna-synthetase-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 8). Quest Database™ Isoleucyl-tRNA synthetase Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/isoleucyl-trna-synthetase-inhibitors-ic50-ki.
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