Structure | Compound Name | Standard Type | Standard Values (in nM) |
|---|---|---|---|
| Tofacitinib | IC50 | 170.0 [1] | |
| Filgotinib | IC50 | 1045.0 [1], 3364.0 [2] | |
| N-{cis-3-[Methyl(7H-pyrrolo[2,3-d]pyrimidin-4-yl)amino]cyclobutyl}propane-1-sulfonamide | IC50 | 163.0 [1], 271.0 [2] | |
| Jak-IN-1 | IC50 | 290.0 [1], 291.0 [2] | |
| Ruxolitinib | IC50 | 31.0 [1] | |
MLA | "Quest Database™ JAK2/JAK1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 5 Dec. 2025, https://www.aatbio.com/data-sets/jak2-jak1-inhibitors-ic50-ki. | |
APA | AAT Bioquest, Inc. (2025, December 5). Quest Database™ JAK2/JAK1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/jak2-jak1-inhibitors-ic50-ki. | |
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