logo
Products
Technologies
Applications
Services
Resources
Selection Guides
About
JAK2/JAK1 Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
TofacitinibIC50170.0 [1]
FilgotinibIC501045.0 [1], 3364.0 [2]
N-{cis-3-[Methyl(7H-pyrrolo[2,3-d]pyrimidin-4-yl)amino]cyclobutyl}propane-1-sulfonamideIC50163.0 [1], 271.0 [2]
Jak-IN-1IC50290.0 [1], 291.0 [2]
RuxolitinibIC5031.0 [1]

References
This online resource may be cited as follows
MLA
"Quest DatabaseJAK2/JAK1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.5 Dec2025https://www.aatbio.com/data-sets/jak2-jak1-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 5). Quest DatabaseJAK2/JAK1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/jak2-jak1-inhibitors-ic50-ki.
BibTeXEndNoteRefMan