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JAK3/JAK1 Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
TofacitinibIC5033.0 [1]
FilgotinibIC50148.0 [1], 154.0 [2], 2140.0 [3]
Jak-IN-1IC5031.0 [1], 1008.0 [2]
RuxolitinibIC5023.0 [1], 1850.0 [2]
BaricitinibIC5067.0 [1], 259.0 [2]

References
This online resource may be cited as follows
MLA
"Quest DatabaseJAK3/JAK1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.5 Dec2025https://www.aatbio.com/data-sets/jak3-jak1-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 5). Quest DatabaseJAK3/JAK1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/jak3-jak1-inhibitors-ic50-ki.
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