Structure | Compound Name | Standard Type | Standard Values (in nM) |
|---|---|---|---|
| Camostat mesylate | IC50 | 1480.0 [1], 34100.0 [2] | |
| (4-Carbamimidoylphenyl) 4-[(E)-3-[(2-ethoxy-2-oxoethyl)-prop-2-enylamino]-2-methyl-3-oxoprop-1-enyl]benzoate | IC50 | 190.0 [1], 15700.0 [2] | |
| 4-(4-Guanidinobenzoyloxy)phenylacetate | IC50 | 2320.0 [1], 100000.0 [2] | |
| 6-(N-Phenylcarbamyl)-2-naphthalenecarboxamidine | Ki | 2500.0 [1] | |
| 1-[[5-(5-Chlorothiophen-2-yl)-1,2-oxazol-3-yl]methyl]-N-(1-propan-2-ylpiperidin-4-yl)indole-2-carboxamide | Ki | 10000.0 [1], 15400.0 [2] | |
MLA | "Quest Database™ Kallikrein 1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 7 Dec. 2025, https://www.aatbio.com/data-sets/kallikrein-1-inhibitors-ic50-ki. | |
APA | AAT Bioquest, Inc. (2025, December 7). Quest Database™ Kallikrein 1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/kallikrein-1-inhibitors-ic50-ki. | |
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