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Kallikrein 6 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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CID 38335241IC50130.0 [1], 470.0 [2]
[2-[(3,5-Dimethyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl] 2-(6-carbamimidoyl-2-methyl-1H-indol-3-yl)acetateIC502.5 [1], 23.0 [2]
4-[[(3S)-3-[(7-Methoxynaphthalen-2-yl)sulfonyl-methylamino]-2-oxopyrrolidin-1-yl]methyl]thiophene-2-carboximidamideIC5030000.0 [1]
[2-[(3,5-Dimethyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl] 2-phenylacetateIC5010000.0 [1]
5-[[(3S)-3-[(7-Methoxynaphthalen-2-yl)sulfonylamino]-2-oxopyrrolidin-1-yl]methyl]thiophene-3-carboximidamideIC5030000.0 [1]
5-[[(3S)-3-[(7-Methoxynaphthalen-2-yl)sulfonylamino]-2-oxopyrrolidin-1-yl]methyl]thiophene-2-carboximidamideIC507750.0 [1]
CID 18392356IC501500.0 [1]
8-[(2R,3S)-5,7-Dihydroxy-2-(4-hydroxyphenyl)-4-oxo-2,3-dihydrochromen-3-yl]-2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-2,3-dihydrochromen-4-oneIC5013500.0 [1]
5-[[(3S)-3-[(7-Methoxynaphthalen-2-yl)sulfonyl-methylamino]-2-oxopyrrolidin-1-yl]methyl]thiophene-2-carboximidamideIC508200.0 [1]
[2-[(3,5-Dimethyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl] 2-(1,2-dimethylindol-3-yl)acetateIC506200.0 [1]
[2-[(3,5-Dimethyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl] 2-(2-methyl-1H-indol-3-yl)propanoateIC5028000.0 [1]
[2-[(3,5-Dimethyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl] 3,3,3-trifluoro-2-(2-methyl-1H-indol-3-yl)propanoateIC5023000.0 [1]
[2-Oxo-2-(pyrimidin-5-ylamino)ethyl] 2-(2-methyl-1H-indol-3-yl)acetateIC5017000.0 [1]
[2-[(3,5-Dimethyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl] 3-(2-methyl-1H-indol-3-yl)propanoateIC5058000.0 [1]
[3-[(3,5-Dimethyl-1-phenylpyrazol-4-yl)amino]-1,1,1-trifluoro-3-oxopropan-2-yl] 2-(2-methyl-1H-indol-3-yl)acetateIC5018.0 [1]
(2R)-2-[[(2R)-2-[[2-[[2-[[2-[[(2S)-2-[[(1R,7S,10S,13S,16S,22S,25S,28S,40R,43S,46S,49S,52S,58S,61S)-40-Acetamido-43,52-bis(2-amino-2-oxoethyl)-13-(carboxymethyl)-46-[(1R)-1-hydroxyethyl]-10,49,61-tris(1H-indol-3-ylmethyl)-16-methyl-25-(2-methylpropyl)-2,8,11,14,17,23,26,41,44,47,50,53,59,62-tetradecaoxo-30,38,65-trithia-3,9,12,15,18,24,27,42,45,48,51,54,60,63-tetradecazahexacyclo[32.29.3.132,36.03,7.018,22.054,58]heptahexaconta-32,34,36(67)-triene-28-carbonyl]amino]propanoyl]-methylamino]acetyl]-methylamino]acetyl]-methylamino]acetyl]amino]-5-carbamimidamidopentanoyl]amino]-5-carbamimidamidopentanoic acidKi50000.0 [1]
(2R)-2-[[(2R)-2-[[2-[[2-[[2-[[(2S)-2-[[(7R,10S,13S,16S,22S,25S,28S,31R,34S,37S,45S,48S,51R)-51-Acetamido-45-benzyl-10-[(2S)-butan-2-yl]-34-(4-carbamimidamidobutyl)-13-(carboxymethyl)-48-(hydroxymethyl)-22,25,37-tris[(4-hydroxyphenyl)methyl]-9,12,15,21,24,27,30,33,36,39,44,47,50-tridecaoxo-28-propan-2-yl-5,53,58-trithia-8,11,14,20,23,26,29,32,35,38,43,46,49-tridecazapentacyclo[29.25.3.13,55.016,20.040,43]hexaconta-1(56),2,55(60)-triene-7-carbonyl]amino]propanoyl]-methylamino]acetyl]-methylamino]acetyl]-methylamino]acetyl]amino]-5-carbamimidamidopentanoyl]amino]-5-carbamimidamidopentanoic acidKi50000.0 [1]
(7R,10S,13S,21S,24S,27S,30S,33S,36S,39S,42S,45R)-7-Acetamido-36-(3-amino-3-oxopropyl)-13-benzyl-24-(4-carbamimidamidobutyl)-39-(carboxymethyl)-10-(hydroxymethyl)-21-[(4-hydroxyphenyl)methyl]-33-(1H-imidazol-5-ylmethyl)-30-methyl-42-(2-methylpropyl)-8,11,14,19,22,25,28,34,37,40,43-undecaoxo-5,47,52-trithia-9,12,15,20,23,26,29,32,35,38,41,44-dodecazatetracyclo[25.23.3.13,49.015,18]tetrapentaconta-1,3(54),49-triene-45-carboxylic acidKi50000.0 [1]
[2-[(3,5-Dimethyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl] 2-(5-ethynyl-2-methyl-1H-indol-3-yl)acetateIC50250.0 [1]
[2-[(3,5-Dimethyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl] 2-(5-carbamimidoyl-2-methyl-1H-indol-3-yl)acetateIC50100.0 [1]
[2-[(3,5-Dimethyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl] 2-(6-ethynyl-2-methyl-1H-indol-3-yl)acetateIC50130.0 [1]
[2-[(3,5-Dimethyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl] 2-(2-propan-2-yl-1H-indol-3-yl)acetateIC5013000.0 [1]
2-(2-Methyl-1H-indol-3-yl)-N-[2-oxo-2-[(1-phenylpyrazol-4-yl)amino]ethyl]acetamideIC506990.0 [1]
[2-[(3,5-Dimethyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl] 2-(4-chloro-2-methyl-1H-indol-3-yl)acetateIC507600.0 [1]
N-[(2S)-1-[[(2S)-1-Amino-4-methyl-1-oxopentan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]-4-chlorobenzamideKi1500.0 [1]
N-(3,5-Dimethyl-1-phenylpyrazol-4-yl)-3,3,3-trifluoro-2-[[2-(2-methyl-1H-indol-3-yl)acetyl]amino]propanamideIC50200000.0 [1]
[2-[(3,5-Dimethyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl] 2-(2-methyl-1H-pyrrolo[2,3-b]pyridin-3-yl)acetateIC50190.0 [1]
[2-[(3,5-Dimethyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl] 2-(2-methyl-1H-pyrrolo[3,2-c]pyridin-3-yl)acetateIC50490.0 [1]
[2-[(3,5-Dimethyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl] 2-(4-ethynyl-2-methyl-1H-indol-3-yl)acetateIC5050000.0 [1]
2-(2-Methyl-1H-indol-3-yl)-N-[2-[(5-methyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl]acetamideIC50290.0 [1]
2-(6-Carbamimidoyl-2-methyl-1H-indol-3-yl)-N-[2-[(3,5-dimethyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl]acetamideIC501200.0 [1]
2-(2-Methyl-1H-pyrrolo[3,2-b]pyridin-3-yl)-N-[2-oxo-2-[(1,3,5-trimethylpyrazol-4-yl)amino]ethyl]acetamideIC501400.0 [1]
[2-[(3,5-Dimethyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl] 2-methyl-2-(2-methyl-1H-indol-3-yl)propanoateIC50200000.0 [1]
[2-[(3,5-Dimethyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl] 2-(2-methyl-1H-pyrrolo[2,3-c]pyridin-3-yl)acetateIC50100.0 [1]
[2-[(3,5-Dimethyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl] 2-(2-methylbenzimidazol-1-yl)acetateIC508900.0 [1]
[3-[(3,5-Dimethyl-1-phenylpyrazol-4-yl)amino]-1,1,1-trifluoro-3-oxopropan-2-yl] 2-(2-methyl-1H-indol-3-yl)propanoateIC502310.0 [1]
[2-[(3,5-Dimethyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl] 2-(5-chloro-2-methyl-1H-indol-3-yl)acetateIC50250.0 [1]
N-[2-[(3,5-Dimethyl-1-phenylpyrazol-4-yl)-methylamino]-2-oxoethyl]-2-(2-methyl-1H-pyrrolo[3,2-b]pyridin-3-yl)acetamideIC502800.0 [1]
2-(2-Methyl-1H-indol-3-yl)-N-[2-[(3-methyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl]acetamideIC507500.0 [1]
[2-[(3,5-Dimethyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl] 2-(2-methyl-1H-pyrrolo[3,2-b]pyridin-3-yl)acetateIC506000.0 [1]
[2-[(3,5-Dimethyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl] 2-(2-ethynyl-1H-indol-3-yl)acetateIC50150.0 [1]
[3-[(3,5-Dimethyl-1-phenylpyrazol-4-yl)amino]-3-oxopropyl] 2-(2-methyl-1H-indol-3-yl)acetateIC50110000.0 [1]
N-[2-[(4-Methyl-3-phenyl-1,2-oxazol-5-yl)amino]-2-oxoethyl]-2-(2-methyl-1H-pyrrolo[3,2-b]pyridin-3-yl)acetamideIC501200.0 [1]
[2-[(3,5-Dimethyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl] 2-(2-oxo-1,3-benzoxazol-3-yl)acetateIC509000.0 [1]
[2-[(3,5-Dimethyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl] 2-(4-oxoquinazolin-3-yl)acetateIC50170000.0 [1]
4-[[(3S)-3-[(7-Methoxynaphthalen-2-yl)sulfonyl-(thiophen-3-ylmethyl)amino]-2-oxopyrrolidin-1-yl]methyl]thiophene-2-carboximidamideIC502900.0 [1]
[2-[(3,5-Dimethyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl] 2-methyl-1H-indole-3-carboxylateIC50200000.0 [1]
[2-(4-Morpholin-4-ylanilino)-2-oxoethyl] 2-(2-methyl-1H-indol-3-yl)acetateIC504400.0 [1]
[2-[(3,5-Dimethyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl] 2-(2-methylindol-1-yl)acetateIC50640.0 [1]
2-{[4-(Aminomethyl)phenyl]carbamoyl}-1-[(1-Benzyl-1h-Imidazol-2-Yl)methyl]-3-HydroxypyridiniumIC50890.0 [1]
[2-[(3,5-Dimethyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl] 2-(1H-indol-3-yl)acetateIC5015000.0 [1]
[2-[(3,5-Dimethyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl] 2-(4-methyl-2-oxo-1,3-thiazol-3-yl)acetateIC5043000.0 [1]
Items per page: 1 - 10 of 52
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References

This online tool may be cited as follows

MLA

"Quest Database™ Kallikrein 6 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/kallikrein-6-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 9). Quest Database™ Kallikrein 6 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/kallikrein-6-inhibitors-ic50-ki.
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