Structure | Compound Name | Standard Type | Standard Values (in nM) |
|---|---|---|---|
| trans-3,4-Dichloro-N-methyl-N-[2-(1-pyrrolidinyl)cyclohexyl]-benzeneacetamide | IC50 | 0.3 [1], 0.55 [2], 1.2 [3] | |
| trans-3,4-Dichloro-N-methyl-N-[2-(1-pyrrolidinyl)cyclohexyl]-benzeneacetamide | Ki | 1.4 [1] | |
| Norbinaltorphimine | IC50 | 2.1 [1], 4.6 [2], 9.3 [3] | |
| Norbinaltorphimine | Ki | 0.2 [1], 0.4 [2] | |
| Naltrexone | IC50 | 1.86 [1], 200.0 [2] | |
MLA | "Quest Database™ Kappa opioid receptor Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 19 Dec. 2025, https://www.aatbio.com/data-sets/kappa-opioid-receptor-inhibitors-ic50-ki. | |
APA | AAT Bioquest, Inc. (2025, December 19). Quest Database™ Kappa opioid receptor Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/kappa-opioid-receptor-inhibitors-ic50-ki. | |
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