logo
Products
Technologies
Applications
Services
Resources
Selection Guides
About
Kappa opioid receptor Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
trans-3,4-Dichloro-N-methyl-N-[2-(1-pyrrolidinyl)cyclohexyl]-benzeneacetamideIC500.3 [1], 0.55 [2], 1.2 [3]
trans-3,4-Dichloro-N-methyl-N-[2-(1-pyrrolidinyl)cyclohexyl]-benzeneacetamideKi1.4 [1]
NorbinaltorphimineIC502.1 [1], 4.6 [2], 9.3 [3]
NorbinaltorphimineKi0.2 [1], 0.4 [2]
NaltrexoneIC501.86 [1], 200.0 [2]

References
This online resource may be cited as follows
MLA
"Quest DatabaseKappa opioid receptor Inhibitors (IC50, Ki)." AAT Bioquest, Inc.19 Dec2025https://www.aatbio.com/data-sets/kappa-opioid-receptor-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 19). Quest DatabaseKappa opioid receptor Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/kappa-opioid-receptor-inhibitors-ic50-ki.
BibTeXEndNoteRefMan