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Kinesin-like protein 1 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
▲
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Standard Values (in nM)
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▼
S-Trityl-L-cysteineIC50352.0 [1]
S-Trityl-L-cysteineKi107.3 [1]
MonastrolIC507452.0 [1]
S-4-Methoxyltrityl-L-cysteineIC5028.5 [1], 166.0 [2], 270.0 [3]
S-4-Methoxyltrityl-L-cysteineKi9.1 [1], 15.7 [2], 21.6 [3], 50.0 [4], 200.0 [5]
N-(3-Aminopropyl)-N-[(1R)-1-(3-benzyl-7-chloro-4-oxochromen-2-yl)-2-methylpropyl]-4-methylbenzamideIC50484.0 [1]
N-(3-Aminopropyl)-N-[(1R)-1-(3-benzyl-7-chloro-4-oxochromen-2-yl)-2-methylpropyl]-4-methylbenzamideKi0.5 [1]
2-(Tritylthio)ethanamineIC50241.2 [1], 395.61 [2]
2-(Tritylthio)ethanamineKi150.0 [1], 152.3 [2], 156.1 [3], 245.0 [4], 245.5 [5]
N-(4-Acetyl-5-methyl-5-phenyl-4,5-dihydro-1,3,4-thiadiazol-2-yl)acetamideIC501300.0 [1]
IspinesibIC501.2 [1], 5.0 [2], 47.0 [3]
IspinesibKi2.3 [1], 2.5 [2]
N-[3-Fluoro-4'-(trifluoromethyl)-4-biphenylyl]ureaIC5015.0 [1], 100.0 [2]
N-[3-Fluoro-4'-(trifluoromethyl)-4-biphenylyl]ureaKi6.8 [1], 8.8 [2], 10.0 [3]
6-[4-(Trifluoromethyl)phenyl]-3,4-dihydro-2(1H)-quinolinoneIC5046.0 [1]
6-[4-(Trifluoromethyl)phenyl]-3,4-dihydro-2(1H)-quinolinoneKi1.4 [1], 1.8 [2], 2.2 [3], 66.0 [4]
FilanesibIC506.0 [1], 18.0 [2]
Adociasulfate-2IC503500.0 [1], 5300.0 [2], 7300.0 [3], 13900.0 [4]
trans-HR22C16IC50800.0 [1], 7100.0 [2]
(2R)-2-Amino-3-[(naphthalen-2-yldiphenylmethyl)sulfanyl]propanoic acidIC5016.3 [1]
(2R)-2-Amino-3-[(naphthalen-2-yldiphenylmethyl)sulfanyl]propanoic acidKi4.2 [1], 50.0 [2], 200.0 [3]
(2R)-2-Amino-3-{[(4-methylphenyl)diphenylmethyl]sulfanyl}propanoic acidIC5061.7 [1]
(2R)-2-Amino-3-{[(4-methylphenyl)diphenylmethyl]sulfanyl}propanoic acidKi13.6 [1], 50.0 [2], 100.0 [3]
[(4R)-4-(3-Hydroxyphenyl)-1,6-dimethyl-2-thioxo-1,2,3,4-tetrahydropyrimidin-5-YL](phenyl)methanoneIC50110.0 [1], 150.0 [2]
(S)-(4-(3-Hydroxyphenyl)-1,6-dimethyl-2-thioxo-1,2,3,4-tetrahydropyrimidin-5-yl)(phenyl)methanoneIC50150.0 [1], 520.0 [2], 650.0 [3]
4-(3-Methylphenyl)-4,4-diphenylbutan-1-amineKi8.8 [1], 10.8 [2], 13.7 [3]
S-Trityl-D-CysteineIC50306.2 [1], 1000.0 [2]
S-Trityl-D-CysteineKi98.6 [1]
Terpendole EIC5023000.0 [1], 34700.0 [2]
N-[1-(3-Benzyl-7-chloro-4-oxoquinazolin-2-yl)propyl]-4-bromo-N-[3-(dimethylamino)propyl]benzamideIC5029.0 [1], 49.0 [2], 53.0 [3]
(R)-2-Amino-3-(diphenyl(4-(trifluoromethyl)phenyl)methylthio)propanoic acidIC50116.4 [1], 262.0 [2]
(R)-2-Amino-3-(diphenyl(4-(trifluoromethyl)phenyl)methylthio)propanoic acidKi50.0 [1]
5-(2,5-Difluorophenyl)-N,N-dimethyl-3-phenyl-3,4-dihydropyrazole-2-carboxamideIC5084.0 [1]
2-(Trifluoromethyl)-9H-carbazoleIC50210.0 [1], 260.0 [2]
(5S)-5-(3-Aminopropyl)-3-(2,5-difluorophenyl)-N,N-dimethyl-5-phenyl-4H-pyrazole-1-carboxamideIC501.9 [1], 2.0 [2]
(2r)-2-Amino-3-[(4-Chlorophenyl)-Diphenyl-Methyl]sulfanyl-Propanoic AcidIC5053.3 [1]
(2r)-2-Amino-3-[(4-Chlorophenyl)-Diphenyl-Methyl]sulfanyl-Propanoic AcidKi50.0 [1], 200.0 [2]
(2R)-2-Amino-3-[(2-methyl-1,1-diphenylpropyl)sulfanyl]propanoic acidIC501152.6 [1]
(2R)-2-Amino-3-[(2-methyl-1,1-diphenylpropyl)sulfanyl]propanoic acidKi150.0 [1], 174.5 [2]
(2R)-2-Amino-3-{[(4-bromophenyl)diphenylmethyl]sulfanyl}propanoic acidIC5026.8 [1]
(2R)-2-Amino-3-{[(4-bromophenyl)diphenylmethyl]sulfanyl}propanoic acidKi50.0 [1], 250.0 [2]
3-(2,5-Difluorophenyl)-N-methyl-5-phenyl-4,5-dihydro-1H-pyrazole-1-carboxamideIC503100.0 [1], 3140.0 [2]
1-[(5S)-3-(2-Chlorophenyl)-5-(3-hydroxyphenyl)-4,5-dihydro-1H-pyrazol-1-yl]ethan-1-oneIC50450.0 [1]
(2R)-2-Amino-3-[(1,1-diphenylpentyl)sulfanyl]propanoic acidIC50318.8 [1]
(2R)-2-Amino-3-[(1,1-diphenylpentyl)sulfanyl]propanoic acidKi50.0 [1], 175.0 [2]
(5S)-5-(3-Aminopropyl)-3-(2,5-difluorophenyl)-N,N-dimethyl-5-phenyl-2H-pyrrole-1-carboxamideIC502.2 [1], 23.0 [2]
(2r)-2-Amino-5-(3-Methylphenyl)-5,5-Diphenylpropanoic AcidKi6.4 [1], 7.1 [2], 10.2 [3]
4-(4-Methylphenyl)-4,4-diphenylbutan-1-amineKi9.7 [1], 16.4 [2]
(5S)-5-[(3S)-3-Amino-4,4-difluorobutyl]-3-(2,5-difluorophenyl)-N,N-dimethyl-5-phenyl-2H-pyrrole-1-carboxamideIC505.2 [1], 24.0 [2], 123.0 [3]
N-[2-[2-(2-Aminoethoxy)ethoxy]ethyl]-4-(3-hydroxyphenyl)-6-methyl-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxamideIC503900.0 [1], 18300.0 [2], 22000.0 [3]
GossypolIC5010800.0 [1], 25000.0 [2]
(S)-MonastrolIC5010000.0 [1]
DimethylenastronIC50200.0 [1]
LitronesibIC507.0 [1], 26.0 [2]
(4R)-4-(3-Hydroxyphenyl)-N,N,7,8-tetramethyl-3,4-dihydroisoquinoline-2(1H)-carboxamideIC50104.0 [1]
2-Hydroxyethyl N-[(2S)-1-[(2S)-4-(2,5-difluorophenyl)-2-phenyl-2,5-dihydropyrrol-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]carbamateIC507.4 [1]
N-(3-Aminopropyl)-N-[(1R)-1-(3-benzyl-7-chloro-4-oxoquinazolin-2-yl)-2-methylpropyl]-3-fluoro-4-methylbenzamideKi1.0 [1], 350.0 [2]
2-(3-Fluoro-4-methoxyanilino)-1-[[2-(trifluoromethyl)phenyl]methyl]benzimidazole-5-carboxylic acidIC50458.8 [1], 2300.0 [2]
1-(3-(2-Fluorophenyl)-5-phenyl-4,5-dihydropyrazol-1-yl)ethanoneIC503600.0 [1]
1-[3-(2,5-Difluorophenyl)-5-phenyl-4,5-dihydro-1H-pyrazol-1-yl]ethan-1-oneIC5094.0 [1]
1-(3-(3-Chlorophenyl)-5-phenyl-4,5-dihydropyrazol-1-yl)ethanoneIC509800.0 [1]
3-(2,5-Difluoro-phenyl)-1-methanesulfonyl-5-phenyl-4,5-dihydro-1H-pyrazoleIC501800.0 [1]
1-(3-(2-Chlorophenyl)-5-phenyl-4,5-dihydropyrazol-1-yl)ethanoneIC503600.0 [1]
Methyl (2R)-2-amino-3-[(triphenylmethyl)sulfanyl]propanoateIC505800.0 [1]
Methyl (2R)-2-amino-3-[(triphenylmethyl)sulfanyl]propanoateKi120.0 [1]
N-[4'-(Trifluoromethyl)-4-biphenylyl]sulfamideKi6.2 [1], 7.0 [2]
2-Fluoro-4-[4-(sulfamoylamino)phenyl]-1-(trifluoromethyl)benzeneIC5015.0 [1], 20.0 [2]
[4-[4-(Trifluoromethyl)phenyl]phenyl]ureaIC5039.0 [1], 140.0 [2]
1-[(3R,3Ar)-3-[3-(4-acetylpiperazin-1-yl)propyl]-8-fluoro-3-phenyl-3a,4-dihydropyrazolo[5,1-c][1,4]benzoxazin-2-yl]ethanoneIC501.6 [1]
Urea, [7-(trifluoromethyl)-9H-carbazol-3-yl]-IC50120.0 [1]
2-{[(4-Methoxyphenyl)(diphenyl)methyl]sulfanyl}ethan-1-amineIC50136.0 [1]
2-{[(4-Methoxyphenyl)(diphenyl)methyl]sulfanyl}ethan-1-amineKi21.5 [1]
N,N-Diethyl-5,5-dimethyl-2-(thiophene-2-carbonylamino)-6,7-dihydro-4H-1-benzothiophene-3-carboxamideIC503100.0 [1]
9H-Pyrido[3,4-b]indole, 7-(trifluoromethyl)-IC5052.0 [1]
(2S)-N-(1-Acetylpiperidin-4-yl)-4-(2,5-difluorophenyl)-N-methyl-2-phenyl-2,5-dihydropyrrole-1-carboxamideIC5050.0 [1]
(2S)-N-(3-Aminopropyl)-4-(2,5-difluorophenyl)-N-methyl-2-phenyl-2,5-dihydropyrrole-1-carboxamideIC5016.0 [1]
3-Amino-1-[(2S)-4-(2,5-difluorophenyl)-2-phenyl-2,5-dihydropyrrol-1-yl]-2,2-dimethylpropan-1-oneIC505.2 [1]
(1S)-1-Cyclopropyl-2-[(2S)-4-(2,5-difluorophenyl)-2-phenyl-2,5-dihydro-1H-pyrrol-1-yl]-2-oxoethanolIC5011.0 [1]
1-[(5S)-3-(2,5-Difluorophenyl)-5-(3-hydroxyphenyl)-4,5-dihydro-1H-pyrazol-1-yl]ethan-1-oneIC5024.7 [1], 26.0 [2]
7,8-Dimethyl-4-phenyl-1,2,3,4-tetrahydroisoquinolineIC508230.0 [1], 8330.0 [2]
2-Ethyl-7,8-dimethyl-4-phenyl-1,2,3,4-tetrahydroisoquinolineIC5025200.0 [1]
2-(7,8-Dimethyl-4-phenyl-1,2,3,4-tetrahydroisoquinolin-2-yl)ethan-1-amineIC502270.0 [1]
4-(3-Hydroxyphenyl)-N,N,7,8-tetramethyl-3,4-dihydro-1H-isoquinoline-2-carboxamideIC50306.0 [1]
7-Bromo-4-(3-hydroxyphenyl)-N,N-dimethyl-3,4-dihydro-1H-isoquinoline-2-carboxamideIC50808.0 [1]
1-(3-(2,5-Difluorophenyl)-5-phenyl-4,5-dihydropyrazol-1-yl)ethanethioneIC50250.0 [1]
1-(3-(2,5-Difluorophenyl)-5-(thiophen-2-yl)-4,5-dihydropyrazol-1-yl)ethanoneIC501800.0 [1]
(2S)-1-[(2S)-4-(2,5-Difluorophenyl)-2-(3-hydroxyphenyl)-2,5-dihydropyrrol-1-yl]-2-hydroxy-3,3-dimethylbutan-1-oneIC501.3 [1]
(2S)-4-(2,5-Difluorophenyl)-N-(2-hydroxyethyl)-2-(3-hydroxyphenyl)-N-methyl-2,5-dihydropyrrole-1-carboxamideIC504.0 [1]
(2S)-2-Amino-1-[(2S)-4-(2,5-difluorophenyl)-2-(3-hydroxyphenyl)-2,5-dihydropyrrol-1-yl]-3-methylbutan-1-oneIC501.2 [1]
(2S)-2-Amino-2-cyclopropyl-1-[(2S)-4-(2,5-difluorophenyl)-2-(3-hydroxyphenyl)-2,5-dihydropyrrol-1-yl]ethanoneIC500.5 [1]
4-(3-Hydroxyphenyl)-6-methyl-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxylic acidIC5032000.0 [1], 72200.0 [2]
CID 44435336IC5011500.0 [1], 23000.0 [2]
5H-Pyrido[4,3-b]indole, 7-(trifluoromethyl)-IC5095.0 [1]
(4s)-4-(3-Hydroxyphenyl)-7,7-Dimethyl-2-Thioxo-2,3,4,6,7,8-Hexahydroquinazolin-5(1h)-OneIC50200.0 [1]
(2R)-2-Amino-3-[(4-cyclohexylphenyl)-diphenylmethyl]sulfanylpropanoic acidIC501578.0 [1]
(2R)-2-Amino-3-[(4-cyclohexylphenyl)-diphenylmethyl]sulfanylpropanoic acidKi3263.7 [1]
(2R)-2-Amino-3-[diphenyl-(4-phenylphenyl)methyl]sulfanylpropanoic acidIC501970.0 [1]
(2R)-2-Amino-3-[diphenyl-(4-phenylphenyl)methyl]sulfanylpropanoic acidKi1349.7 [1]
(2R)-2-Amino-3-[(4-tert-butylphenyl)-diphenylmethyl]sulfanylpropanoic acidIC501244.0 [1]
(2R)-2-Amino-3-[(4-tert-butylphenyl)-diphenylmethyl]sulfanylpropanoic acidKi428.6 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Kinesin-like protein 1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 10 May. 2024, https://www.aatbio.com/data-sets/kinesin-like-protein-1-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 10). Quest Database™ Kinesin-like protein 1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/kinesin-like-protein-1-inhibitors-ic50-ki.
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