Structure | Compound Name | Standard Type | Standard Values (in nM) |
|---|---|---|---|
| 5-[[(5S,9R)-9-(4-Cyanophenyl)-3-(3,5-dichlorophenyl)-1-methyl-2,4-dioxo-1,3,7-triazaspiro[4.4]nonan-7-yl]methyl]thiophene-3-carboxylic acid | IC50 | 18.0 [1], 276.0 [2], 280.0 [3] | |
| Bms-688521 | IC50 | 2.5 [1], 60.0 [2], 276.0 [3] | |
| 2-[(5S,9R)-9-(4-Cyanophenyl)-3-(3,5-dichlorophenyl)-1-methyl-2,4-dioxo-1,3,7-triazaspiro[4.4]nonan-7-yl]pyrimidine-5-carboxylic acid | IC50 | 11.0 [1], 260.0 [2] | |
| 5-[(5S,9R)-9-(4-Cyanophenyl)-3-(3,5-dichlorophenyl)-1-methyl-2,4-dioxo-1,3,7-triazaspiro[4.4]nonan-7-yl]pyrazine-2-carboxylic acid | IC50 | 19.0 [1], 1260.0 [2] | |
| 6-[(5S,9R)-9-(4-Cyanophenyl)-3-(3,5-dichlorophenyl)-1-methyl-2,4-dioxo-1,3,7-triazaspiro[4.4]nonan-7-yl]pyridazine-3-carboxylic acid | IC50 | 13.0 [1], 270.0 [2] | |
MLA | "Quest Database™ Leukocyte adhesion glycoprotein LFA-1 alpha Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 4 Nov. 2025, https://www.aatbio.com/data-sets/leukocyte-adhesion-glycoprotein-lfa-1-alpha-inhibitors-ic50-ki. | |
APA | AAT Bioquest, Inc. (2025, November 4). Quest Database™ Leukocyte adhesion glycoprotein LFA-1 alpha Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/leukocyte-adhesion-glycoprotein-lfa-1-alpha-inhibitors-ic50-ki. | |
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