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Liver glycogen phosphorylase Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
(2S)-2-[[3-[(2-Chloro-6-methylphenyl)carbamoylamino]naphthalene-2-carbonyl]amino]-2-cyclohexylacetic acidIC5073.0 [1], 80.0 [2], 460.0 [3], 600.0 [4], 1290.0 [5]
5-Chloro-1H-indole-2-carboxylic acid [1-(4-fluorobenzyl)-2-(4-hydroxypiperidin-1YL)-2-oxoethyl]amideIC50205.0 [1], 920.0 [2], 2400.0 [3]
(2S)-2-Cyclohexyl-2-[[3-[(2,6-dichlorophenyl)carbamoylamino]naphthalene-2-carbonyl]amino]acetic acidIC5021.0 [1], 100.0 [2], 320.0 [3]
(2S)-2-Cyclohexyl-2-[[3-[(2,6-dimethylphenyl)carbamoylamino]naphthalene-2-carbonyl]amino]acetic acidIC50120.0 [1], 1060.0 [2], 1100.0 [3]
(2S)-2-[[3-[(2-Chloro-6-methylphenyl)carbamoylamino]naphthalene-2-carbonyl]amino]-3-cyclohexylpropanoic acidIC502200.0 [1], 7400.0 [2], 51000.0 [3]
(2S)-2-[[3-[(2-Chloro-6-methylphenyl)carbamoylamino]naphthalene-2-carbonyl]amino]butanedioic acidIC50390.0 [1], 1600.0 [2], 4700.0 [3]
CP-91149IC5082.0 [1], 110.0 [2]
5-Chloro-N-(2-oxo-1,2,3,4-tetrahydroquinolin-3-yl)-1H-indole-2-carboxamideIC5044.0 [1], 86.0 [2]
alpha-D-GlucoseKi4280000.0 [1], 4900000.0 [2]
AfegostatIC50670.0 [1], 700.0 [2]
8,9,10-Trihydroxy-7-hydroxymethyl-2-thioxo-6-oxa-1,3-diaza-spiro[4.5]decan-4-oneKi10900.0 [1], 29800.0 [2]
Glycogen Phosphorylase InhibitorIC5052.48 [1], 53.0 [2]
(5R,6R,7S,8S,9R)-9-(Hydroxymethyl)-3-naphthalen-2-yl-1,10-dioxa-2-azaspiro[4.5]dec-2-ene-6,7,8-triolIC5014180.0 [1], 19950.0 [2]
5-Chloro-N-(2-oxo-1,3,4,5-tetrahydro-1-benzazepin-3-yl)-1H-indole-2-carboxamideIC50105.0 [1]
(S)-5-Chloro-N-(1-(dimethylamino)-1-oxo-3-phenylpropan-2-yl)-1H-indole-2-carboxamideIC5051.0 [1], 82.0 [2]
5-Chloro-N-[1-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-2-oxo-3,4-dihydroquinolin-3-yl]-1H-indole-2-carboxamideIC50140.0 [1]
5-Chloro-N-[1-[[3-(1H-imidazol-2-yl)-1H-1,2,4-triazol-5-yl]methyl]-2-oxo-3,4-dihydroquinolin-3-yl]-1H-indole-2-carboxamideIC50160.0 [1]
2,3-Dichloro-N-(2-oxo-1,2,3,4-tetrahydroquinolin-3-yl)-4H-thieno[3,2-b]pyrrole-5-carboxamideIC50132.0 [1]
2-Chloro-N-(2-oxo-1,2,3,4-tetrahydroquinolin-3-yl)-6H-thieno[2,3-b]pyrrole-5-carboxamideIC5041.0 [1]
5-Chloro-N-(1-methyl-2-oxo-3,4-dihydroquinolin-3-yl)-1H-indole-2-carboxamideIC5025.0 [1]
O-Tert-Butyl-N-[(3-{[(2,4,6-Trimethylphenyl)carbamoyl]amino}naphthalen-2-Yl)carbonyl]-L-ThreonineIC507.0 [1], 139.0 [2]
5-Methyl-N-(1-methyl-2-oxo-3,4-dihydroquinolin-3-yl)-1H-indole-2-carboxamideIC50120.0 [1]
5-Fluoro-N-(1-methyl-2-oxo-3,4-dihydroquinolin-3-yl)-1H-indole-2-carboxamideIC50120.0 [1]
5-Bromo-N-(1-methyl-2-oxo-3,4-dihydroquinolin-3-yl)-1H-indole-2-carboxamideIC5030.0 [1]
N-(1-Methyl-2-oxo-3,4-dihydroquinolin-3-yl)-1H-indole-2-carboxamideIC50160.0 [1]
5-Chloro-N-(1-methyl-2-oxo-4,5-dihydro-3H-1-benzazepin-3-yl)-1H-indole-2-carboxamideIC50305.0 [1]
5-Chloro-N-[(3R)-2-oxo-1,3,4,5-tetrahydro-1-benzazepin-3-yl]-1H-indole-2-carboxamideIC5099.0 [1]
5-Chloro-N-[(3S)-2-oxo-3,4-dihydro-1H-quinolin-3-yl]-1H-indole-2-carboxamideIC5047.0 [1]
5-Chloro-N-[(3S)-2-oxo-1,3,4,5-tetrahydro-1-benzazepin-3-yl]-1H-indole-2-carboxamideIC50240.0 [1]
5-Chloro-N-[(3S)-1-methyl-2-oxo-3,4-dihydroquinolin-3-yl]-1H-indole-2-carboxamideIC5057.0 [1]
5-Chloro-N-[(3R)-1-methyl-2-oxo-3,4-dihydroquinolin-3-yl]-1H-indole-2-carboxamideIC5061.0 [1]
5-Chloro-N-[2-oxo-1-(pyridin-2-ylmethyl)-3,4-dihydroquinolin-3-yl]-1H-indole-2-carboxamideIC50110.0 [1]
N-(1-Methyl-2-oxo-3,4-dihydroquinolin-3-yl)-5-phenyl-1H-indole-2-carboxamideIC5020000.0 [1]
N-(1-Methyl-2-oxo-3,4-dihydroquinolin-3-yl)-5-(trifluoromethyl)-1H-indole-2-carboxamideIC501500.0 [1]
Methyl 2-[(1-methyl-2-oxo-3,4-dihydroquinolin-3-yl)carbamoyl]-1H-indole-5-carboxylateIC505300.0 [1]
5-Cyano-N-(1-methyl-2-oxo-3,4-dihydroquinolin-3-yl)-1H-indole-2-carboxamideIC50180.0 [1]
5-Methoxy-N-(1-methyl-2-oxo-3,4-dihydroquinolin-3-yl)-1H-indole-2-carboxamideIC501700.0 [1]
5-Ethyl-N-(1-methyl-2-oxo-3,4-dihydroquinolin-3-yl)-1H-indole-2-carboxamideIC502500.0 [1]
4-Chloro-N-(1-methyl-2-oxo-3,4-dihydroquinolin-3-yl)-1H-indole-2-carboxamideIC501600.0 [1]
7-Chloro-N-(1-methyl-2-oxo-3,4-dihydroquinolin-3-yl)-1H-indole-2-carboxamideIC5088.0 [1]
N-(1-Methyl-2-oxo-3,4-dihydroquinolin-3-yl)-6-phenyl-1H-indole-2-carboxamideIC5020000.0 [1]
6-Chloro-N-(1-methyl-2-oxo-3,4-dihydroquinolin-3-yl)-1H-indole-2-carboxamideIC5099.0 [1]
Methyl 5-chloro-2-[(1-methyl-2-oxo-3,4-dihydroquinolin-3-yl)carbamoyl]-1H-indole-4-carboxylateIC5020000.0 [1]
7-Amino-N-(1-methyl-2-oxo-3,4-dihydroquinolin-3-yl)-1H-indole-2-carboxamideIC501200.0 [1]
5-Chloro-N-[2-oxo-1-(pyridin-3-ylmethyl)-3,4-dihydroquinolin-3-yl]-1H-indole-2-carboxamideIC50130.0 [1]
5-Chloro-7-fluoro-N-(1-methyl-2-oxo-3,4-dihydroquinolin-3-yl)-1H-indole-2-carboxamideIC5083.0 [1]
Methyl 5-chloro-2-[(1-methyl-2-oxo-3,4-dihydroquinolin-3-yl)carbamoyl]-1H-indole-6-carboxylateIC5020000.0 [1]
3,4-Dichloro-N-(2-oxo-1,2,3,4-tetrahydro-quinolin-3-yl)-benzamideIC501370.0 [1], 1400.0 [2]
3,4-Dichloro-N-(2-oxo-1,3,4,5-tetrahydro-1-benzazepin-3-yl)benzamideIC506400.0 [1]
N-(1-Methyl-2-oxo-3,4-dihydroquinolin-3-yl)-7-nitro-1H-indole-2-carboxamideIC50300.0 [1]
5-Chloro-N-[4-(hydroxymethyl)phenyl]-1H-indole-2-carboxamideIC501600.0 [1]
5-Chloro-N-[(3R)-2-oxo-3,4-dihydro-1H-quinolin-3-yl]-1H-indole-2-carboxamideIC5025.0 [1]
3-Chloro-4-[3-(2,4-dichloro-benzoyl)-ureido]-benzoic acidIC50416.87 [1], 420.0 [2]
4-[3-(2-Chloro-benzoyl)-ureido]-3-methoxy-benzoic acidIC50850.0 [1], 851.14 [2]
4-[3-(2,4-Dichloro-benzoyl)-ureido]-benzoic acidIC507000.0 [1], 7079.46 [2]
2-Chloro-4-fluoro-N-(1,2,3,4-tetrahydroquinolin-7-ylcarbamoyl)benzamideIC503467.37 [1], 3500.0 [2]
1-(2-Chloro-benzoyl)-3-(5-hydroxy-2-methoxy-phenyl)-ureaIC5064.57 [1], 65.0 [2]
2-Amino-4-[3-(2-chloro-4-fluoro-benzoyl)-ureido]-benzoic acidIC50700.0 [1], 707.95 [2]
(2S)-3-Ethoxy-2-[[3-[(2,4,6-trimethylphenyl)carbamoylamino]naphthalene-2-carbonyl]amino]propanoic acidIC5056.0 [1], 4467.0 [2]
(2S)-3-[(2-Methylpropan-2-yl)oxy]-2-[[3-[(2,4,6-trimethylphenyl)carbamoylamino]naphthalene-2-carbonyl]amino]propanoic acidIC5044.0 [1], 387.0 [2]
4-[(2-Chloro-4,5-difluorobenzoyl)carbamoylamino]-2-hydroxy-5-methoxybenzoic acidIC5050.0 [1], 50.12 [2]
3-Chloro-4-[3-(2-chloro-benzoyl)-ureido]-benzoic acidIC50933.25 [1], 940.0 [2]
4-[3-(2,4-Dichloro-benzoyl)-ureido]-2-hydroxy-benzoic acidIC50537.03 [1], 540.0 [2]
(2S)-2-[[3-[(2,4,6-Trimethylphenyl)carbamoylamino]naphthalene-2-carbonyl]amino]hexanoic acidIC5023.0 [1], 501.0 [2]
(2S)-5-Methyl-2-[[3-[(2,4,6-trimethylphenyl)carbamoylamino]naphthalene-2-carbonyl]amino]hexanoic acidIC509.0 [1], 452.0 [2]
2-(1,4-Dioxaspiro[4.5]decan-8-yl)-2-[[3-[(2,4,6-trimethylphenyl)carbamoylamino]naphthalene-2-carbonyl]amino]acetic acidIC50106.0 [1], 2053.0 [2]
N-[(5-Acetamido-2-chlorophenyl)carbamoyl]-2-chloro-4,5-difluorobenzamideIC5060.0 [1], 60.26 [2]
1-[[3-[(2,4,6-Trimethylphenyl)carbamoylamino]naphthalene-2-carbonyl]amino]cyclooctane-1-carboxylic acidIC505.0 [1], 498.0 [2]
(2S)-4-Methyl-2-[[3-[(2,4,6-trimethylphenyl)carbamoylamino]naphthalene-2-carbonyl]amino]pentanoic acidIC50101.0 [1], 1427.0 [2]
3-Chloro-4-[3-(2-chloro-4-fluoro-benzoyl)-ureido]-benzoic acidIC50158.49 [1], 160.0 [2]
2-[[3-[(2,4,6-Trimethylphenyl)carbamoylamino]naphthalene-2-carbonyl]amino]-1,3-dihydroindene-2-carboxylic acidIC5091.0 [1], 4788.0 [2]
1-(2-Chloro-4-fluorobenzoyl)-3-[2-chloro-4-(1H-tetrazol-5-yl)phenyl]ureaIC50190.0 [1], 190.55 [2]
4-[3-(2-Fluoro-benzoyl)-ureido]-3-methoxy-benzoic acid methyl esterIC5015000.0 [1], 15135.61 [2]
4-[(2-Chloro-4-fluorobenzoyl)carbamoylamino]-2-hydroxy-5-methoxybenzoic acidIC50158.49 [1], 160.0 [2]
4-[3-(2-Chloro-4-fluoro-benzoyl)-ureido]-3-trifluoromethoxy-benzoic acidIC50150.0 [1], 151.36 [2]
(2S)-3-(2,2-Dimethylpropoxy)-2-[[3-[(2,4,6-trimethylphenyl)carbamoylamino]naphthalene-2-carbonyl]amino]propanoic acidIC5079.0 [1], 949.0 [2]
1-(2,4-Dichloro-benzoyl)-3-(1H-indol-6-yl)-ureaIC5027542.29 [1], 35000.0 [2]
4-[3-(2-Chloro-4-fluoro-benzoyl)-ureido]-2-hydroxy-benzoic acidIC50510.0 [1], 512.86 [2]
1-(2-Chloro-4-fluoro-benzoyl)-3-(4-hydroxymethyl-2-methoxy-phenyl)-ureaIC50800.0 [1], 831.76 [2]
1-[[3-[(2,4,6-Trimethylphenyl)carbamoylamino]naphthalene-2-carbonyl]amino]cycloheptane-1-carboxylic acidIC5036.0 [1], 585.0 [2]
4-[(2-Chloro-4,5-difluorobenzoyl)carbamoylamino]-3-(2,2,2-trifluoroethoxy)benzoic acidIC50446.68 [1], 450.0 [2]
1-(2-Chloro-4-fluoro-benzoyl)-3-[4-(1H-tetrazol-5-yl)-2-trifluoromethoxy-phenyl]-ureaIC5079.43 [1], 80.0 [2]
(2S)-Cyclohexyl{[3-({[(2,4,6-trichlorophenyl)amino]carbonyl}amino)-2-naphthoyl]amino}ethanoic acidIC5065.0 [1], 224.0 [2]
4-[3-(2-Bromo-benzoyl)-ureido]-3-methoxy-benzoic acidIC501200.0 [1], 1202.26 [2]
(2S)-3-Propan-2-yloxy-2-[[3-[(2,4,6-trimethylphenyl)carbamoylamino]naphthalene-2-carbonyl]amino]propanoic acidIC50148.0 [1], 451.0 [2]
4-[3-(2,4-Dichloro-benzoyl)-ureido]-3-methoxy-N-methyl-benzamideIC50407.38 [1], 410.0 [2]
(2S)-2-Cyclopentyl-2-[[3-[(2,4,6-trimethylphenyl)carbamoylamino]naphthalene-2-carbonyl]amino]acetic acidIC5014.0 [1], 321.0 [2]
1-(2-Chloro-4-fluoro-benzoyl)-3-(3,4-dihydroxy-phenyl)-ureaIC50120.0 [1], 120.23 [2]
4-[3-(2-Fluoro-benzoyl)-ureido]-3-methoxy-benzoic acidIC502137.96 [1], 2150.0 [2]
4-[3-(2-Chloro-4-fluoro-benzoyl)-ureido]-3-methoxy-benzoic acidIC50208.93 [1], 210.0 [2]
1-[[3-[(2,4,6-Trimethylphenyl)carbamoylamino]naphthalene-2-carbonyl]amino]cyclodecane-1-carboxylic acidIC5014.0 [1], 443.0 [2]
4-[3-(2-Chloro-4-fluoro-benzoyl)-ureido]-3-methoxy-benzamideIC50300.0 [1], 302.0 [2]
4-Chloro-3-[3-(2-chloro-4-fluoro-benzoyl)-ureido]-benzenesulfonamideIC502000.0 [1], 2041.74 [2]
5-Chloro-4-[3-(2,4-dichloro-benzoyl)-ureido]-2-hydroxy-benzoic acidIC50150.0 [1], 151.36 [2]
(2S)-3-Butoxy-2-[[3-[(2,4,6-trimethylphenyl)carbamoylamino]naphthalene-2-carbonyl]amino]propanoic acidIC5095.0 [1], 1139.0 [2]
5-Chloro-4-[(2-chloro-4,5-difluorobenzoyl)carbamoylamino]-2-hydroxybenzoic acidIC5089.13 [1], 90.0 [2]
2,4-Dichloro-N-[[2-chloro-5-(methylcarbamoylamino)phenyl]carbamoyl]benzamideIC50158.49 [1], 160.0 [2]
(2S)-2-[[3-[(2,4,6-Trimethylphenyl)carbamoylamino]naphthalene-2-carbonyl]amino]pentanoic acidIC5039.0 [1], 1019.0 [2]
1-(2,4-Dichloro-benzoyl)-3-(3-hydroxy-phenyl)-ureaIC50970.0 [1], 977.24 [2]
2-[[3-[(2,4,6-Trimethylphenyl)carbamoylamino]naphthalene-2-carbonyl]amino]-3,4-dihydro-1H-naphthalene-2-carboxylic acidIC5027.0 [1], 1070.0 [2]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Liver glycogen phosphorylase Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 10 May. 2024, https://www.aatbio.com/data-sets/liver-glycogen-phosphorylase-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 10). Quest Database™ Liver glycogen phosphorylase Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/liver-glycogen-phosphorylase-inhibitors-ic50-ki.
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