Long-chain fatty acid transport protein 1 Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	N-[[4-Ethyl-5-[[5-(trifluoromethoxy)-1,3-benzoxazol-2-yl]methylsulfanyl]-1,2,4-triazol-3-yl]methyl]aniline	IC50	100.0 [1]
	2-[4-(4-Fluorophenyl)piperazin-1-yl]-N-(1,3-thiazol-2-yl)acetamide	IC50	1000.0 [1]
	CID 71601847	IC50	46.0 [1]
	2-{[4-Allyl-5-(anilinomethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}-N-(4-methoxyphenyl)acetamide	IC50	6600.0 [1]
	2-(4-Phenylpiperazin-1-yl)-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)acetamide	IC50	280.0 [1]
	2-[4-(4-Fluorophenyl)piperazin-1-yl]-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)acetamide	IC50	77.0 [1]
	N-(4,5-Dimethyl-1,3-thiazol-2-yl)-2-[4-(4-fluorophenyl)piperazin-1-yl]acetamide	IC50	430.0 [1]
	2-[[5-(Anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]-N-(6-propanoylpyridin-3-yl)acetamide	IC50	400.0 [1]
	2-[[5-(Anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]-N-methyl-N-(4-propanoylphenyl)acetamide	IC50	580.0 [1]
	2-[[5-(Anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]-N-ethyl-N-(4-propanoylphenyl)acetamide	IC50	1000.0 [1]
	Ethyl 1-[2-[[5-(anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]acetyl]-3,4-dihydro-2H-quinoline-6-carboxylate	IC50	1000.0 [1]
	Ethyl 1-[2-[[5-(anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]acetyl]-2,3-dihydroindole-5-carboxylate	IC50	1000.0 [1]
	Ethyl 4-[[2-[[5-(anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]acetyl]amino]benzoate	IC50	330.0 [1]
	Ethyl 3-[[2-[[5-(anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]acetyl]amino]benzoate	IC50	1000.0 [1]
	Methyl 4-[[2-[[5-(anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]acetyl]amino]benzoate	IC50	540.0 [1]
	Tert-butyl 4-[[2-[[5-(anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]acetyl]amino]benzoate	IC50	1000.0 [1]
	4-[[2-[[5-(Anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]acetyl]amino]benzoic acid	IC50	1000.0 [1]
	4-[[2-[[5-(Anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]acetyl]amino]-N-methylbenzamide	IC50	1000.0 [1]
	4-[[2-[[5-(Anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]acetyl]amino]-N,N-dimethylbenzamide	IC50	1000.0 [1]
	4-[[2-[[5-(Anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]acetyl]amino]-N-ethylbenzamide	IC50	1000.0 [1]
	1-[2-[[5-(Anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanylmethyl]-1,3-benzoxazol-5-yl]propan-1-one	IC50	190.0 [1]
	Ethyl 2-[[5-(anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanylmethyl]-1,3-benzoxazole-5-carboxylate	IC50	680.0 [1]
	1-[2-[[5-(Anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanylmethyl]-1,3-benzoxazol-6-yl]propan-1-one	IC50	900.0 [1]
	1-[2-[[5-(Anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfonylmethyl]-1,3-benzoxazol-5-yl]propan-1-one	IC50	1670.0 [1]
	1-[2-[[5-(Anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanylmethyl]-1,3-benzoxazol-5-yl]propan-1-ol	IC50	1000.0 [1]
	(NZ)-N-[1-[2-[[5-(anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanylmethyl]-1,3-benzoxazol-5-yl]propylidene]hydroxylamine	IC50	260.0 [1]
	N-[[4-Ethyl-5-[[5-[(Z)-C-ethyl-N-methoxycarbonimidoyl]-1,3-benzoxazol-2-yl]methylsulfanyl]-1,2,4-triazol-3-yl]methyl]aniline	IC50	1000.0 [1]
	N-[[4-Ethyl-5-[[5-(trifluoromethyl)-1,3-benzoxazol-2-yl]methylsulfanyl]-1,2,4-triazol-3-yl]methyl]aniline	IC50	360.0 [1]
	1-[2-[[5-(Anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanylmethyl]-1,3-benzoxazol-5-yl]-2-methylpropan-1-one	IC50	600.0 [1]
	N-(1,3-Benzothiazol-2-yl)-2-[4-(4-fluorophenyl)piperazin-1-yl]acetamide	IC50	490.0 [1]
	2-[[5-(Anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]-N-(4-methylsulfonylphenyl)acetamide	IC50	1000.0 [1]
	N-[[5-[(6-Chloro-1,3-benzoxazol-2-yl)methylsulfanyl]-4-ethyl-1,2,4-triazol-3-yl]methyl]aniline	IC50	1000.0 [1]
	N-[[4-Ethyl-5-[(5-ethyl-1,3-benzoxazol-2-yl)methylsulfanyl]-1,2,4-triazol-3-yl]methyl]aniline	IC50	1000.0 [1]
	N-[[4-Ethyl-5-[(5-methoxy-1,3-benzoxazol-2-yl)methylsulfanyl]-1,2,4-triazol-3-yl]methyl]aniline	IC50	1000.0 [1]
	2-[[5-(Anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]-N-(4-methoxyphenyl)acetamide	IC50	1000.0 [1]
	2-[[5-(Anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]-N-(4-chlorophenyl)acetamide	IC50	1000.0 [1]
	2-[[5-(Anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]-N-(4-propanoylphenyl)acetamide	IC50	400.0 [1]
	N-[[5-(1,3-Benzoxazol-2-ylmethylsulfanyl)-4-ethyl-1,2,4-triazol-3-yl]methyl]aniline	IC50	1000.0 [1]
	N-[[4-Ethyl-5-[(5-fluoro-1,3-benzoxazol-2-yl)methylsulfanyl]-1,2,4-triazol-3-yl]methyl]aniline	IC50	1000.0 [1]
	N-[[5-[(5-Chloro-1,3-benzoxazol-2-yl)methylsulfanyl]-4-ethyl-1,2,4-triazol-3-yl]methyl]aniline	IC50	1000.0 [1]
	2-[[5-(Anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]-N-phenylacetamide	IC50	1000.0 [1]
	N-(4-Acetylphenyl)-2-[[5-(anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]acetamide	IC50	1000.0 [1]
	2-[[5-(Anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]-N-(4-benzoylphenyl)acetamide	IC50	1000.0 [1]
	N-[[4-Ethyl-5-[(5-methyl-1,3-benzoxazol-2-yl)methylsulfanyl]-1,2,4-triazol-3-yl]methyl]aniline	IC50	1000.0 [1]
	2-[[5-(Anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]-N-(4-cyanophenyl)acetamide	IC50	1000.0 [1]
	2-[[5-(Anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]-N-[4-(2-ethyltetrazol-5-yl)phenyl]acetamide	IC50	1000.0 [1]
	2-[[5-(Anilinomethyl)-4-ethyl-1,2,4-triazol-3-yl]sulfanyl]-N-(4-butanoylphenyl)acetamide	IC50	230.0 [1]
	2-[4-(4-Fluorophenyl)piperazin-1-yl]-N-(4,5,6,7-tetrahydro-1,3-benzoxazol-2-yl)acetamide	IC50	180.0 [1]
	N-(5,6-Dihydro-4H-cyclopenta[d][1,3]thiazol-2-yl)-2-[4-(4-fluorophenyl)piperazin-1-yl]acetamide	IC50	490.0 [1]
	2-[4-(4-Fluorophenyl)piperazin-1-yl]-N-(5,6,7,8-tetrahydro-4H-cyclohepta[d][1,3]thiazol-2-yl)acetamide	IC50	120.0 [1]
	2-[4-(4-Methylphenyl)piperazin-1-yl]-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)acetamide	IC50	250.0 [1]
	2-[4-(3-Fluorophenyl)piperazin-1-yl]-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)acetamide	IC50	1000.0 [1]
	2-(4-Benzoylpiperazin-1-yl)-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)acetamide	IC50	1000.0 [1]
	2-(4-Cyclohexylpiperazin-1-yl)-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)acetamide	IC50	1000.0 [1]
	2-(4-Pyridin-2-ylpiperazin-1-yl)-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)acetamide	IC50	200.0 [1]
	2-(4-Pyridin-3-ylpiperazin-1-yl)-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)acetamide	IC50	1000.0 [1]
	2-(4-Pyridin-4-ylpiperazin-1-yl)-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)acetamide	IC50	1000.0 [1]
	2-(4-Pyrimidin-2-ylpiperazin-1-yl)-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)acetamide	IC50	1000.0 [1]
	N-(4,5,6,7-Tetrahydro-1,3-benzothiazol-2-yl)-2-[4-(1,3-thiazol-2-yl)piperazin-1-yl]acetamide	IC50	520.0 [1]
	2-[4-(5-Fluoropyridin-2-yl)piperazin-1-yl]-N-(4,5,6,7-tetrahydro-1,3-benzoxazol-2-yl)acetamide	IC50	100.0 [1]
	2-[4-(5-Fluoropyridin-2-yl)piperazin-1-yl]-N-methyl-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)acetamide	IC50	41.0 [1]
	N-Ethyl-2-[4-(5-fluoropyridin-2-yl)piperazin-1-yl]-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)acetamide	IC50	780.0 [1]
	2-[4-(5-Fluoropyridin-2-yl)piperazin-1-yl]-1-(2-methylimidazo[1,2-a]pyridin-3-yl)ethanone	IC50	430.0 [1]
	2-[4-(5-Fluoropyridin-2-yl)piperazin-1-yl]-1-imidazo[1,2-a]pyridin-3-ylethanone	IC50	130.0 [1]
	2-[4-(5-Fluoropyridin-2-yl)piperazin-1-yl]-1-imidazo[1,5-a]pyridin-3-ylethanone	IC50	1000.0 [1]
	2-[4-(5-Fluoropyridin-2-yl)piperazin-1-yl]-1-(1H-indazol-3-yl)ethanone	IC50	1000.0 [1]
	2-[4-(5-Fluoropyridin-2-yl)piperazin-1-yl]-1-pyrazolo[1,5-a]pyridin-3-ylethanone	IC50	330.0 [1]
	2-[4-(5-Fluoropyridin-2-yl)piperazin-1-yl]-1-(1H-indol-3-yl)ethanone	IC50	1000.0 [1]
	1-(1-Benzofuran-3-yl)-2-[4-(5-fluoropyridin-2-yl)piperazin-1-yl]ethanone	IC50	470.0 [1]
	2-[4-(5-Fluoropyridin-2-yl)piperazin-1-yl]-1-(2-methyl-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-3-yl)ethanone	IC50	190.0 [1]
	2-[4-(5-Fluoropyridin-2-yl)piperazin-1-yl]-1-(5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-3-yl)ethanone	IC50	100.0 [1]
	2-[4-(4-Fluorophenyl)piperazin-1-yl]-N-(5-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)acetamide	IC50	26.0 [1]
	1-(2-Methylimidazo[1,2-a]pyridine-3-yl)-2-(4-phenylpiperazino)ethanone	IC50	3000.0 [1]
	Ethyl 4-{[({5-[(benzylsulfanyl)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}sulfanyl)acetyl]amino}benzoate	IC50	7600.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 74 ⟨⟩

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References

This online tool may be cited as follows

MLA	"Quest Database™ Long-chain fatty acid transport protein 1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/long-chain-fatty-acid-transport-protein-1-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, May 9). Quest Database™ Long-chain fatty acid transport protein 1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/long-chain-fatty-acid-transport-protein-1-inhibitors-ic50-ki.
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