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Lysine-specific demethylase 5A Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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2-[[3-[[(E)-4-(Dimethylamino)but-2-enoyl]amino]phenyl]-(2-piperidin-1-ylethoxy)methyl]thieno[3,2-b]pyridine-7-carboxylic acidIC50180.0 [1]
2-[(3-Aminophenyl)-(2-piperidin-1-ylethoxy)methyl]thieno[3,2-b]pyridine-7-carboxylic acidIC504900.0 [1]
3-[4-(2-Butyl-1-benzofuran-3-carbonyl)-2,6-diiodophenoxy]propyl-trimethylazaniumIC5030000.0 [1]
Kdm5A-IN-1IC5045.0 [1], 500.0 [2], 570.0 [3], 2400.0 [4], 22000.0 [5]
2-{5-[(4-Chloro-2-Methylphenyl)methoxy]-1h-Pyrazol-1-Yl}pyridine-4-Carboxylic AcidIC5013.0 [1], 100.0 [2]
N-{(3S)-1-[5-(Propan-2-yl)-1H-pyrazole-3-carbonyl]pyrrolidin-3-yl}cyclopropanecarboxamideIC501800.0 [1], 4300.0 [2], 11000.0 [3], 140000.0 [4]
2-[5-[(4-Chlorophenyl)methoxy]pyrazol-1-yl]pyridine-4-carboxylic acidIC5014.0 [1], 100.0 [2]
3-[4-(2-Butyl-1-benzofuran-3-carbonyl)phenoxy]propyl-trimethylazanium;iodideIC5037000.0 [1], 80000.0 [2], 340000.0 [3]
3-[4-(2-Butyl-1-benzofuran-3-carbonyl)phenoxy]propyl-trimethylazanium;iodideKi74000.0 [1]
AmiodaroneIC5099000.0 [1], 1000000.0 [2]
Kdoam-25IC501700.0 [1], 3200.0 [2], 18000.0 [3]
2-[5-(4-Methoxyphenyl)-1-methylimidazol-4-yl]pyridine-4-carboxylic acidIC50100.0 [1], 1000.0 [2]
2-[5-[(4-Fluorophenyl)methoxy]-4-(2-hydroxyethyl)pyrazol-1-yl]pyridine-4-carboxylic acidIC5080.0 [1], 100.0 [2]
(2-Butyl-1-benzofuran-3-yl)-[4-[3-(dimethylamino)propoxy]phenyl]methanoneIC50166000.0 [1], 1000000.0 [2]
2-(1-Methylimidazol-4-yl)pyridine-4-carboxylic acidIC50100.0 [1], 10000.0 [2]
2-(1-Methylimidazol-4-yl)-4-(2H-tetrazol-5-yl)pyridineIC50100.0 [1], 10000.0 [2]
2-[5-[4-(Cyclopropylmethoxy)phenyl]-1-methylimidazol-4-yl]pyridine-4-carboxylic acidIC50100.0 [1], 1000.0 [2]
2-[4-(2-Butyl-1-benzofuran-3-carbonyl)-2,6-diiodophenoxy]ethyl-trimethylazaniumIC5026000.0 [1], 30000.0 [2], 1658000.0 [3]
N-OxalylglycineIC50250000.0 [1], 640000.0 [2]
Pyridine-2,4-dicarboxylic acidIC50760.0 [1], 100000.0 [2]
(2-(Phenylamino)-1,4-phenylene)bis((4-(pyrrolidin-1-yl)piperidin-1-yl)methanone)IC5010000.0 [1], 30000.0 [2]
(5-Bromopyridin-3-yl)(4-(pyrrolidin-1-yl)piperidin-1-yl)methanoneIC5010000.0 [1], 30000.0 [2]
1,4-Phenylenebis(1,4'-bipiperidin-1'-ylmethanone)IC5010000.0 [1], 30000.0 [2]
[3-[6-Methyl-4-(1-methylpyrazol-4-yl)pyridin-2-yl]pyrrolidin-1-yl]-(5-propan-2-yl-1H-pyrazol-3-yl)methanoneIC50160.0 [1], 30000.0 [2]
3-[(1-Cyclopentyl-5-fluoroindazol-3-yl)amino]pyridine-4-carboxylic acidIC50100.0 [1]
2-(5-(Benzyloxy)-1H-pyrazol-1-yl)isonicotinic acidIC50100.0 [1], 550.0 [2]
2-[5-[(4-Cyanophenyl)methoxy]pyrazol-1-yl]pyridine-4-carboxylic acidIC504.0 [1], 100.0 [2]
2-[5-[(4-Chloro-2-methoxyphenyl)methoxy]pyrazol-1-yl]pyridine-4-carboxylic acidIC5012.0 [1], 100.0 [2]
2-[5-[[4-(Trifluoromethyl)phenyl]methoxy]pyrazol-1-yl]pyridine-4-carboxylic acidIC50100.0 [1], 240.0 [2]
2-[5-[(4-Methoxyphenyl)methoxy]pyrazol-1-yl]pyridine-4-carboxylic acidIC50100.0 [1], 1700.0 [2]
2-[5-[(4-Fluorophenyl)methoxy]-4-methylpyrazol-1-yl]pyridine-4-carboxylic acidIC5077.0 [1], 100.0 [2]
2-[5-[(4-Bromophenyl)methoxy]pyrazol-1-yl]pyridine-4-carboxylic acidIC506.0 [1], 100.0 [2]
2-[5-[(4-Cyclopropylphenyl)methoxy]pyrazol-1-yl]pyridine-4-carboxylic acidIC50100.0 [1], 250.0 [2]
2-[5-[[4-Chloro-2-(cyclopropylmethoxy)phenyl]methoxy]pyrazol-1-yl]pyridine-4-carboxylic acidIC5075.0 [1], 100.0 [2]
2-[5-[(2-Fluorophenyl)methoxy]pyrazol-1-yl]pyridine-4-carboxylic acidIC50100.0 [1], 270.0 [2]
2-[5-[(4-Chloro-2-fluorophenyl)methoxy]pyrazol-1-yl]pyridine-4-carboxylic acidIC5018.0 [1], 100.0 [2]
2-[5-[(4-Methylphenyl)methoxy]pyrazol-1-yl]pyridine-4-carboxylic acidIC5032.0 [1], 100.0 [2]
2-[5-[(4-Ethylphenyl)methoxy]pyrazol-1-yl]pyridine-4-carboxylic acidIC5044.0 [1], 100.0 [2]
2-[5-[(4-Chloro-2-ethoxyphenyl)methoxy]pyrazol-1-yl]pyridine-4-carboxylic acidIC5019.0 [1], 100.0 [2]
2-[4-[2-(Dimethylamino)ethyl]-5-[(4-fluorophenyl)methoxy]pyrazol-1-yl]pyridine-4-carboxylic acidIC503.0 [1], 100.0 [2]
2-[5-[(3-Fluorophenyl)methoxy]pyrazol-1-yl]pyridine-4-carboxylic acidIC50100.0 [1], 430.0 [2]
2-[5-[(4-Fluorophenyl)methoxy]pyrazol-1-yl]pyridine-4-carboxylic acidIC5038.0 [1], 100.0 [2]
2-[5-[(4-Chloro-2-phenylmethoxyphenyl)methoxy]pyrazol-1-yl]pyridine-4-carboxylic acidIC5032.0 [1], 100.0 [2]
2-[4-Ethyl-5-[(4-fluorophenyl)methoxy]pyrazol-1-yl]pyridine-4-carboxylic acidIC5029.0 [1], 100.0 [2]
2-[5-[1-(4-Fluorophenyl)ethoxy]pyrazol-1-yl]pyridine-4-carboxylic acidIC50100.0 [1], 180.0 [2]
3-[(1-Methylpyrazolo[3,4-b]pyridin-3-yl)amino]pyridine-4-carboxylic acidIC50100.0 [1]
DisulfiramIC5010000.0 [1]
DaminozideIC502200000.0 [1]
4-HydroxybenzohydrazideIC5013000.0 [1]
3-[[2-Pyridin-2-Yl-6-(1,2,4,5-Tetrahydro-3-Benzazepin-3-Yl)pyrimidin-4-Yl]amino]propanoic AcidIC50110000.0 [1]
(E)-5-Chloro-2-(2-(phenyl(pyridin-2-yl)methylene)hydrazinyl)pyridineIC50251.19 [1]
Di-N-desethylamiodaroneIC5026000.0 [1]
3-Benzyl-6-(2-pyridinyl)[1,2,4]triazolo[3,4-b][1,3,4]thiadiazoleIC5025000.0 [1]
2-[(2-Chlorophenyl)-[2-(1-methylpyrrolidin-2-yl)ethoxy]methyl]-1H-pyrrolo[3,2-b]pyridine-7-carboxylic acidIC50290.0 [1]
5,7-Dichloro-4-((3-(4-methoxyphenylthio)benzyl)(methyl)amino)quinoline-2-carboxylic acidIC503800.0 [1]
2-[(2-Chlorophenyl)-propoxymethyl]-1H-pyrrolo[3,2-b]pyridine-7-carboxylic acidIC506700.0 [1]
CID 127030711IC5010000.0 [1]
2-[(2-Chlorophenyl)-[2-(1-methylimidazol-2-yl)ethoxy]methyl]-1H-pyrrolo[3,2-b]pyridine-7-carboxylic acidIC501400.0 [1]
N-[6-(4-Acryloyl-1,4-diazepan-1-yl)-2-(pyridin-2-yl)pyrimidin-4-yl]-beta-alanineIC5071000.0 [1]
2-[(2-Chlorophenyl)-[(4,4-difluorocyclohexyl)methoxy]methyl]-1H-pyrrolo[3,2-b]pyridine-7-carboxylic acidIC5022000.0 [1]
2-[(2-Chlorophenyl)-(2-piperidin-1-ylethoxy)methyl]-1H-pyrrolo[3,2-b]pyridine-7-carboxylic acidIC50690.0 [1]
8-(1-Methyl-1h-Imidazol-4-Yl)-2-(4,4,4-Trifluorobutoxy)pyrido[3,4-D]pyrimidin-4-OlIC50100.0 [1]
3-[9-(Dimethylamino)nonanoyl-hydroxyamino]propanoic acidIC5013000.0 [1]
(2S)-2-[[(2S)-2-[[(2S)-5-Amino-2-[[(2S)-6-amino-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-6-amino-2-[[2-[[2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-6-amino-2-[[(2S)-2-[[(2S)-2-[[(2S,3R)-2-[[(2S)-5-amino-2-[[(2S)-6-amino-2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-2-aminopropanoyl]amino]-5-carbamimidamidopentanoyl]amino]-3-hydroxybutanoyl]amino]hexanoyl]amino]-5-oxopentanoyl]amino]-3-hydroxybutanoyl]amino]propanoyl]amino]-5-carbamimidamidopentanoyl]amino]hexanoyl]amino]-3-hydroxypropanoyl]amino]-3-hydroxybutanoyl]amino]acetyl]amino]acetyl]amino]hexanoyl]amino]propanoyl]pyrrolidine-2-carbonyl]amino]-5-carbamimidamidopentanoyl]amino]hexanoyl]amino]-5-oxopentanoyl]amino]-4-methylpentanoyl]amino]propanoic acidIC50571000.0 [1]
9H-Xanthen-9-one, 1,4-dihydroxy-IC5025000.0 [1]
9-Oxo-4,5,6,7,8,9-hexahydro-pyrazolo[5,1-b]quinazoline-3-carbonitrileIC501000.0 [1]
6-Ethyl-3-[1-[4-(hydroxymethyl)pyridin-2-yl]pyrazol-4-yl]-5-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-oneIC502.3 [1]
6-Bromo-3-(4-methylbenzoyl)-1-benzofuran-4,5-dioneIC505000.0 [1]
1,4-Bis(4-(pyrrolidinyl)piperidinyl)benzamideIC5010000.0 [1]
6-Hydroxy-1-methoxy-9H-xanthen-9-oneIC5015000.0 [1]
Kdm5-IN-1IC5014.0 [1]
[3-[6-Methyl-4-(1-methylpyrazol-4-yl)pyridin-2-yl]pyrrolidin-1-yl]-(5-propyl-1H-pyrazol-3-yl)methanoneIC50458.0 [1]
(5-Cyclopropyl-1H-pyrazol-3-yl)-[3-[6-methyl-4-(1-methylpyrazol-4-yl)pyridin-2-yl]pyrrolidin-1-yl]methanoneIC50357.0 [1]
N-[1-(5-Propan-2-yl-1H-pyrazole-3-carbonyl)pyrrolidin-3-yl]propanamideIC50251.0 [1]
N-[1-(5-Propan-2-yl-1H-pyrazole-3-carbonyl)pyrrolidin-3-yl]acetamideIC501100.0 [1]
N,N,2-Trimethyl-6-[1-(5-propan-2-yl-1H-pyrazole-3-carbonyl)pyrrolidin-3-yl]pyridine-4-carboxamideIC507200.0 [1]
[3-(6-Methyl-4-phenoxypyridin-2-yl)pyrrolidin-1-yl]-(5-propan-2-yl-1H-pyrazol-3-yl)methanoneIC50128.0 [1]
[3-[6-Methyl-4-(1-methylpyrazol-4-yl)pyridin-2-yl]-2,5-dihydropyrrol-1-yl]-(5-propan-2-yl-1H-pyrazol-3-yl)methanoneIC5025000.0 [1]
(5-Propan-2-yl-1H-pyrazol-3-yl)-[3-(pyridin-2-ylamino)pyrrolidin-1-yl]methanoneIC508900.0 [1]
[3-(6-Methyl-4-pyridin-3-ylpyridin-2-yl)pyrrolidin-1-yl]-(5-propan-2-yl-1H-pyrazol-3-yl)methanoneIC50469.0 [1]
[3-[4-(Furan-3-yl)-6-methylpyridin-2-yl]pyrrolidin-1-yl]-(5-propan-2-yl-1H-pyrazol-3-yl)methanoneIC50265.0 [1]
(5-Ethyl-1H-pyrazol-3-yl)-[3-[6-methyl-4-(1-methylpyrazol-4-yl)pyridin-2-yl]pyrrolidin-1-yl]methanoneIC50878.0 [1]
(5-Tert-butyl-1H-pyrazol-3-yl)-[3-[6-methyl-4-(1-methylpyrazol-4-yl)pyridin-2-yl]pyrrolidin-1-yl]methanoneIC50897.0 [1]
N-[2-Methyl-6-[1-(5-propan-2-yl-1H-pyrazole-3-carbonyl)pyrrolidin-3-yl]pyridin-4-yl]acetamideIC501500.0 [1]
[3-[6-Methyl-4-(1-methylpyrazol-4-yl)pyridin-2-yl]pyrrolidin-1-yl]-(5-methyl-1H-pyrazol-3-yl)methanoneIC502600.0 [1]
[3-[6-Methyl-4-(3-methylphenyl)pyridin-2-yl]pyrrolidin-1-yl]-(5-propan-2-yl-1H-pyrazol-3-yl)methanoneIC50122.0 [1]
[3-[4-(1-Benzylpyrazol-4-yl)-6-methylpyridin-2-yl]pyrrolidin-1-yl]-(5-propan-2-yl-1H-pyrazol-3-yl)methanoneIC50105.0 [1]
[3-(4-Bromopyrazol-1-yl)pyrrolidin-1-yl]-(5-propan-2-yl-1H-pyrazol-3-yl)methanoneIC50727.0 [1]
(5-Propan-2-yl-1H-pyrazol-3-yl)-(3-pyridin-2-yloxypyrrolidin-1-yl)methanoneIC5014300.0 [1]
N-[1-(5-Propan-2-yl-1H-pyrazole-3-carbonyl)pyrrolidin-3-yl]cyclobutanecarboxamideIC5060.0 [1]
3-[5-[Butyl(methyl)amino]pentanoyl-hydroxyamino]propanoic acidIC504300.0 [1]
3-[3-[Butyl(methyl)amino]propanoyl-hydroxyamino]propanoic acidIC5053000.0 [1]
3-[4-[Butyl(methyl)amino]butanoyl-hydroxyamino]propanoic acidIC506300.0 [1]
3-[7-[Butyl(methyl)amino]heptanoyl-hydroxyamino]propanoic acidIC501800.0 [1]
3-[5-[Ethyl(methyl)amino]pentanoyl-hydroxyamino]propanoic acidIC507800.0 [1]
3-[Hydroxy-[5-[methyl(propyl)amino]pentanoyl]amino]propanoic acidIC508900.0 [1]
3-[Hydroxy-[5-[methyl(pentyl)amino]pentanoyl]amino]propanoic acidIC502300.0 [1]
3-[5-[Hexyl(methyl)amino]pentanoyl-hydroxyamino]propanoic acidIC503300.0 [1]
3-[5-[Butyl(ethyl)amino]pentanoyl-hydroxyamino]propanoic acidIC5014000.0 [1]
3-[5-(Dibutylamino)pentanoyl-hydroxyamino]propanoic acidIC5019000.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Lysine-specific demethylase 5A Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/lysine-specific-demethylase-5a-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 9). Quest Database™ Lysine-specific demethylase 5A Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/lysine-specific-demethylase-5a-inhibitors-ic50-ki.
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