Lysophosphatidic acid receptor Edg-7 Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	[(2R)-2-[[(Z)-Octadec-9-enoyl]amino]-3-[4-(pyridin-2-ylmethoxy)phenyl]propyl] dihydrogen phosphate	IC50	175.0 [1]
	[(2R)-2-[[(Z)-Octadec-9-enoyl]amino]-3-[4-(pyridin-2-ylmethoxy)phenyl]propyl] dihydrogen phosphate	Ki	175.0 [1]
	CID 10367662	IC50	301.0 [1]
	CID 10367662	Ki	148.0 [1]
	Dodecyl dihydrogen phosphate	IC50	384.0 [1]
	Dodecyl dihydrogen phosphate	Ki	121.0 [1]
	Tetradecylphosphonic acid	IC50	3100.0 [1]
	Tetradecylphosphonic acid	Ki	1120.0 [1]
	Dioctanoylglycerol pyrophosphate	IC50	454.0 [1]
	Dioctanoylglycerol pyrophosphate	Ki	202.0 [1]
	Decyl dihydrogen phosphate	IC50	384.0 [1]
	Decyl dihydrogen phosphate	Ki	121.0 [1]
	Decylphosphonic acid	IC50	1200.0 [1]
	Decylphosphonic acid	Ki	680.0 [1]
	Dodecylphosphonic acid	IC50	654.0 [1]
	Dodecylphosphonic acid	Ki	303.0 [1]
	2-(1,3-Dioxo-5-(p-tolyloxy)isoindolin-2-yl)acetic acid	IC50	2992.0 [1]
	2-(1,3-Dioxo-5-(p-tolyloxy)isoindolin-2-yl)acetic acid	Ki	1084.0 [1]
	Tetradecyl dihydrogen phosphate	IC50	422.0 [1]
	Tetradecyl dihydrogen phosphate	Ki	211.0 [1]
	Dodecyl-thiophosphate	IC50	28.0 [1]
	Dodecyl-thiophosphate	Ki	14.0 [1]
	3-(4-{3-[4-(3-Carboxy-acryloylamino)-phenoxy]-phenoxy}-phenylcarbamoyl)-acrylic acid	IC50	1230.0 [1]
	3-(4-{3-[4-(3-Carboxy-acryloylamino)-phenoxy]-phenoxy}-phenylcarbamoyl)-acrylic acid	Ki	310.0 [1]
	[(2S)-2-[[(Z)-Octadec-9-enoyl]amino]-3-[4-(pyridin-2-ylmethoxy)phenyl]propyl] dihydrogen phosphate	IC50	940.0 [1]
	[(2S)-2-[[(Z)-Octadec-9-enoyl]amino]-3-[4-(pyridin-2-ylmethoxy)phenyl]propyl] dihydrogen phosphate	Ki	940.0 [1]
	Phosphoric acid mono-((E)-tetradec-9-enyl) ester	IC50	96.0 [1]
	Phosphoric acid mono-((E)-tetradec-9-enyl) ester	Ki	58.0 [1]
	Thiophosphoric acid (E)-dodec-9-enyl ester	IC50	27.0 [1]
	Thiophosphoric acid (E)-dodec-9-enyl ester	Ki	14.0 [1]
	Phosphoric acid mono-((E)-dodec-9-enyl) ester	IC50	32.0 [1]
	Phosphoric acid mono-((E)-dodec-9-enyl) ester	Ki	27.0 [1]
	Dihydroxy-sulfanylidene-[(E)-tetradec-9-enoxy]-lambda5-phosphane	IC50	28.0 [1]
	Dihydroxy-sulfanylidene-[(E)-tetradec-9-enoxy]-lambda5-phosphane	Ki	14.0 [1]
	Thiophosphoric acid decyl ester	IC50	122.0 [1]
	Thiophosphoric acid decyl ester	Ki	49.0 [1]
	Phosphoric acid mono-((E)-dec-4-enyl) ester	IC50	830.0 [1]
	Phosphoric acid mono-((E)-dec-4-enyl) ester	Ki	370.0 [1]
	Thiophosphoric acid dec-9-enyl ester	IC50	340.0 [1]
	Thiophosphoric acid dec-9-enyl ester	Ki	128.0 [1]
	Phosphoric acid mono-((E)-tetradec-11-enyl) ester	IC50	103.0 [1]
	Phosphoric acid mono-((E)-tetradec-11-enyl) ester	Ki	40.0 [1]
	Thiophosphoric acid tetradecyl ester	IC50	162.0 [1]
	Thiophosphoric acid tetradecyl ester	Ki	76.0 [1]
	(1,1-Difluoro-pentadecyl)-phosphonic acid	IC50	1513.0 [1]
	(1,1-Difluoro-pentadecyl)-phosphonic acid	Ki	575.0 [1]
	Phosphoric acid monodec-9-enyl ester	IC50	770.0 [1]
	Phosphoric acid monodec-9-enyl ester	Ki	504.0 [1]
	2-Hexadecanoylamino-3-(4-phosphonooxy-phenyl)-propionic acid	IC50	5570.0 [1]
	2-Hexadecanoylamino-3-(4-phosphonooxy-phenyl)-propionic acid	Ki	2325.0 [1]
	2-(3-(4-Nitrophenoxy)phenyl)-1,3-dioxoisoindoline-5-carboxylic acid	IC50	752.0 [1]
	2-(3-(4-Nitrophenoxy)phenyl)-1,3-dioxoisoindoline-5-carboxylic acid	Ki	230.0 [1]
	[(2S)-2-(Octadecanoylamino)-3-(4-phenylmethoxyphenyl)propyl] dihydrogen phosphate	IC50	1186.0 [1]
	[(2S)-2-(Octadecanoylamino)-3-(4-phenylmethoxyphenyl)propyl] dihydrogen phosphate	Ki	588.0 [1]
	1-[4-[4-[1-Methyl-5-[[(1R)-1-phenylethoxy]carbonylamino]triazol-4-yl]phenyl]phenyl]cyclopropane-1-carboxylic acid	IC50	2290.0 [1]
	[(1R)-1-Phenylethyl] N-[3-methyl-5-[4-[4-[1-(methylsulfonylcarbamoyl)cyclopropyl]phenyl]phenyl]triazol-4-yl]carbamate	IC50	2310.0 [1]
	2-[4-[4-[1-Methyl-5-[[(1R)-1-phenylethoxy]carbonylamino]triazol-4-yl]phenyl]phenyl]acetic acid	IC50	21940.0 [1]
	1-[4-[3-Fluoro-4-[1-methyl-5-[[(1R)-1-phenylethoxy]carbonylamino]triazol-4-yl]phenyl]phenyl]cyclopropane-1-carboxylic acid	IC50	27350.0 [1]
	1-[4-[4-[1-Methyl-5-[[(1S)-1-[3-(trifluoromethyl)phenyl]ethoxy]carbonylamino]triazol-4-yl]phenyl]phenyl]cyclopropane-1-carboxylic acid	IC50	6300.0 [1], 6310.0 [2]
	1-[4-[4-[1-Methyl-5-[[(1R)-1-[3-(trifluoromethyl)phenyl]ethoxy]carbonylamino]triazol-4-yl]phenyl]phenyl]cyclopropane-1-carboxylic acid	IC50	132.0 [1]
	[(1R)-1-[3-(Trifluoromethyl)phenyl]ethyl] N-[3-methyl-5-[4-[4-[1-(methylsulfonylcarbamoyl)cyclopropyl]phenyl]phenyl]triazol-4-yl]carbamate	IC50	65.0 [1], 65.7 [2]
	2-[4-[4-[1-Methyl-5-[[(1R)-1-phenylethoxy]carbonylamino]triazol-4-yl]phenyl]cyclohexyl]acetic acid	IC50	18600.0 [1], 18640.0 [2]
	[(2S)-2-[[(Z)-Octadec-9-enoyl]amino]-3-(4-phenylmethoxyphenyl)propyl] dihydrogen phosphate	IC50	6450.0 [1], 10000.0 [2]
	[(2R)-2-[[(Z)-Octadec-9-enoyl]amino]-3-[4-(pyridin-3-ylmethoxy)phenyl]propyl] dihydrogen phosphate	Ki	1688.0 [1]
	[(2R)-2-[[(Z)-Octadec-9-enoyl]amino]-3-(4-phenylmethoxyphenyl)propyl] dihydrogen phosphate	IC50	10000.0 [1]
	(4'-(4-((R)-1-(2-Chlorophenyl)ethoxycarbonylamino)-3-methylisoxazol-5-yl)biphenyl-4-yl)acetic acid	IC50	1600.0 [1]
	4-(3-Benzamidophenylamino)-4-oxobut-2-enoic acid	Ki	316.6 [1]
	LPA2 antagonist 1	IC50	50000.0 [1]
	AM095 free acid	IC50	8000.0 [1]
	CID 66775043	IC50	10000.0 [1]
	[1-Bromo-(3S)-hydrox-4-(palmitoyloxy)butyl]phosphate	Ki	170.0 [1]
	2-((3-(1,3-Dioxo-1H-benzo[de]isoquinolin-2(3H)-yl)propyl)thio)benzoic acid	IC50	6600.0 [1]
	2-[4-[[(3,5-Dimethoxybenzoyl)-(3-phenylpropyl)amino]methyl]phenoxy]benzoic acid	IC50	40.0 [1]
	E,E-3-[4'-(3-Carboxy-acryloylamino)-biphenyl-4-ylcarbamoyl]-acrylic acid	Ki	7020.0 [1]
	[(2S)-2-[[(Z)-Octadec-9-enoyl]amino]-3-(4-prop-2-ynoxyphenyl)propyl] dihydrogen phosphate	IC50	10000.0 [1]
	[(2S)-2-[[(Z)-Octadec-9-enoyl]amino]-3-(4-prop-2-enoxyphenyl)propyl] dihydrogen phosphate	IC50	10000.0 [1]
	[(2S)-3-[4-[(3-Methoxyphenyl)methoxy]phenyl]-2-[[(Z)-octadec-9-enoyl]amino]propyl] dihydrogen phosphate	IC50	642.0 [1]
	(2-Hydroxy-2-sulfanylidene-1,2lambda5-oxaphospholan-5-yl)methyl hexadecanoate	IC50	2340.0 [1]
	(2-Hydroxy-2-sulfanylidene-1,2lambda5-oxaphospholan-5-yl)methyl octadecanoate	Ki	636.0 [1]
	(2r)-3-(Phosphonooxy)propane-1,2-Diyl Diheptanoate	IC50	143.0 [1]
	[2-(Octanoylamino)-3-(4-phenylmethoxyphenyl)propyl] dihydrogen phosphate	IC50	10000.0 [1]
	[3-(4-Phenylmethoxyphenyl)-2-(tetradecanoylamino)propyl] dihydrogen phosphate	IC50	10000.0 [1]
	[(2R)-2-[[(Z)-Octadec-9-enoyl]amino]-3-[4-[(3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxyphenyl]propyl] dihydrogen phosphate	IC50	10000.0 [1]
	[2-[[(9Z,12Z)-Octadeca-9,12-dienoyl]amino]-3-(4-phenylmethoxyphenyl)propyl] dihydrogen phosphate	IC50	10000.0 [1]
	[(2R)-3-(4-Methoxyphenyl)-2-[[(Z)-octadec-9-enoyl]amino]propyl] dihydrogen phosphate	IC50	10000.0 [1]
	[(2S)-3-(4-Ethoxyphenyl)-2-[[(Z)-octadec-9-enoyl]amino]propyl] dihydrogen phosphate	IC50	6930.0 [1]
	[(2S)-3-[4-(3-Methylbutoxy)phenyl]-2-[[(Z)-octadec-9-enoyl]amino]propyl] dihydrogen phosphate	IC50	5920.0 [1]
	[(2R)-3-[4-(3-Methylbutoxy)phenyl]-2-[[(Z)-octadec-9-enoyl]amino]propyl] dihydrogen phosphate	IC50	351.0 [1]
	[(2R)-3-(4-Hex-5-ynoxyphenyl)-2-[[(Z)-octadec-9-enoyl]amino]propyl] dihydrogen phosphate	IC50	3280.0 [1]
	[(2R)-3-(4-Ethoxyphenyl)-2-[[(Z)-octadec-9-enoyl]amino]propyl] dihydrogen phosphate	IC50	6410.0 [1]
	[(2R)-3-[4-(Cyclohexylmethoxy)phenyl]-2-[[(Z)-octadec-9-enoyl]amino]propyl] dihydrogen phosphate	IC50	4030.0 [1]
	[(2R)-3-[4-[(3-Methoxyphenyl)methoxy]phenyl]-2-[[(Z)-octadec-9-enoyl]amino]propyl] dihydrogen phosphate	IC50	35.6 [1]
	[4-[(2R)-2-[[(Z)-Octadec-9-enoyl]amino]-3-phosphonooxypropyl]phenyl] 3,4,5-trimethoxybenzoate	IC50	427.0 [1]
	[(2R)-3-[4-(2,3-Dihydro-1H-inden-2-yloxy)phenyl]-2-[[(Z)-octadec-9-enoyl]amino]propyl] dihydrogen phosphate	IC50	2310.0 [1]
	[4-[(2S)-2-[[(Z)-Octadec-9-enoyl]amino]-3-phosphonooxypropyl]phenyl] 4-pentylbenzoate	IC50	10000.0 [1]
	4-Amino-benzoic acid 4-[(S)-2-((Z)-octadec-9-enoylamino)-3-phosphonooxy-propyl]-phenyl ester	IC50	10000.0 [1]
	[2-(Hexadecanoylamino)-3-(4-phenylmethoxyphenyl)propyl] dihydrogen phosphate	IC50	6840.0 [1]
	[2-(Hexadecanoylamino)-3-[4-[(3-methoxyphenyl)methoxy]phenyl]propyl] dihydrogen phosphate	IC50	7220.0 [1]
	[(2S)-3-[4-(1H-Indol-2-yloxy)phenyl]-2-[[(Z)-octadec-9-enoyl]amino]propyl] dihydrogen phosphate	IC50	9260.0 [1]
	[(2R)-3-[4-(1H-Indol-2-yloxy)phenyl]-2-[[(Z)-octadec-9-enoyl]amino]propyl] dihydrogen phosphate	IC50	2630.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 100 ⟨⟩

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References

This online tool may be cited as follows

MLA	"Quest Database™ Lysophosphatidic acid receptor Edg-7 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 10 May. 2024, https://www.aatbio.com/data-sets/lysophosphatidic-acid-receptor-edg-7-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, May 10). Quest Database™ Lysophosphatidic acid receptor Edg-7 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/lysophosphatidic-acid-receptor-edg-7-inhibitors-ic50-ki.
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