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Lysosomal protective protein Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
3-[3-Chloro-5-[2-(trifluoromethoxy)phenyl]phenyl]-3-(5-methyl-1,3-thiazol-2-yl)propanoic acidIC50221.0 [1]
BortezomibIC509200.0 [1]
Diisopropyl fluorophosphateIC5010000.0 [1]
CarfilzomibIC5030000.0 [1]
e-64IC50300000.0 [1]
3,4-DichloroisocoumarinIC50600.0 [1]
VaborbactamIC501000000.0 [1]
(S)-3-{[1-(2-Fluoro-Phenyl)-5-Hydroxy-1h-Pyrazole-3-Carbonyl]-Amino}-3-O-Tolyl-Propionic AcidIC5038.0 [1]
(3S)-3-[[1-(2-Fluorophenyl)-5-methoxypyrazole-3-carbonyl]amino]-3-(2-methylphenyl)propanoic acidIC5026.0 [1]
(3S)-3-[[1-(2-Fluorophenyl)-5-[(2R)-2-hydroxy-3,3-dimethylbutoxy]pyrazole-3-carbonyl]amino]-3-(2-methylphenyl)propanoic acidIC505.0 [1]
(3S)-3-[[1-(2-Fluorophenyl)-5-[(2S)-2-hydroxy-3,3-dimethylbutoxy]pyrazole-3-carbonyl]amino]-3-(2-methylphenyl)propanoic acidIC5010.0 [1]
(3S)-3-[[5-(3,3-Dimethyl-2-oxobutoxy)-1-(2-fluorophenyl)pyrazole-3-carbonyl]amino]-3-(2-methylphenyl)propanoic acidIC503.0 [1]
(3S)-3-(2,4-Dichlorophenyl)-3-[[1-(2-fluorophenyl)-5-[(2S)-2-hydroxy-3,3-dimethylbutoxy]pyrazole-3-carbonyl]amino]propanoic acidIC5070.0 [1]
(3S)-3-(2,4-Dichlorophenyl)-3-[[1-(2-fluorophenyl)-5-[(2R)-2-hydroxy-3,3-dimethylbutoxy]pyrazole-3-carbonyl]amino]propanoic acidIC5050.0 [1]
(3S)-3-[[5-Ethoxy-1-(2-fluorophenyl)pyrazole-3-carbonyl]amino]-3-(2-methylphenyl)propanoic acidIC5015.0 [1]
(3S)-3-[[2-(4-Fluorophenyl)-3-oxo-1H-pyrazole-5-carbonyl]amino]-3-(2-methylphenyl)propanoic acidIC5087.0 [1]
3-[(3-Oxo-2-phenyl-1H-pyrazole-5-carbonyl)amino]-3-(4-phenoxyphenyl)propanoic acidIC50200.0 [1]
(3S)-3-(2-Methylphenyl)-3-[(3-oxo-2-phenyl-1H-pyrazole-5-carbonyl)amino]propanoic acidIC5070.0 [1]
(3S)-3-[[2-(3-Fluorophenyl)-3-oxo-1H-pyrazole-5-carbonyl]amino]-3-(2-methylphenyl)propanoic acidIC5059.0 [1]
(3S)-3-[[2-(3-Chlorophenyl)-3-oxo-1H-pyrazole-5-carbonyl]amino]-3-(2-methylphenyl)propanoic acidIC50102.0 [1]
3-[[2-(2-Fluorophenyl)-3-oxo-1H-pyrazole-5-carbonyl]amino]-3-phenylpropanoic acidIC50226.0 [1]
3-(2,3-Dichlorophenyl)-3-[[2-(2,4-difluorophenyl)-3-oxo-1H-pyrazole-5-carbonyl]amino]propanoic acidIC50120.0 [1]
(3S)-3-[[5-(Cyclopropylmethoxy)-1-(2-fluorophenyl)pyrazole-3-carbonyl]amino]-3-(2-methylphenyl)propanoic acidIC5015.0 [1]
3-(2,3-Dichlorophenyl)-3-[(3-oxo-2-phenyl-1H-pyrazole-5-carbonyl)amino]propanoic acidIC50100.0 [1]
(3R)-3-(2-Methylphenyl)-3-[(3-oxo-2-phenyl-1H-pyrazole-5-carbonyl)amino]propanoic acidIC507800.0 [1]
(3S)-3-[[2-(2-Fluorophenyl)-3-oxo-1H-pyrazole-5-carbonyl]amino]-3-[2-(trifluoromethyl)phenyl]propanoic acidIC50375.0 [1]
(3S)-3-[[4-Chloro-1-(2-fluorophenyl)-5-methoxypyrazole-3-carbonyl]amino]-3-(2-methylphenyl)propanoic acidIC50110.0 [1]
(3S)-3-[(4-Hydroxy-1-phenylpyrazole-3-carbonyl)amino]-3-(2-methylphenyl)propanoic acidIC50110.0 [1]
3-[[2-(2,5-Dimethylphenyl)-3-oxo-1H-pyrazole-5-carbonyl]amino]-3-(4-fluorophenyl)propanoic acidIC505380.0 [1]
3-[[2-(4-Chlorophenyl)-3-oxo-1H-pyrazole-5-carbonyl]amino]-3-(2,5-dichlorophenyl)propanoic acidIC5030000.0 [1]
(3S)-3-[[4-Fluoro-1-(2-fluorophenyl)-5-methoxypyrazole-3-carbonyl]amino]-3-(2-methylphenyl)propanoic acidIC5030.0 [1]
3-(5-Fluoro-2-methylphenyl)-3-[[2-(2-fluorophenyl)-3-oxo-1H-pyrazole-5-carbonyl]amino]propanoic acidIC5076.0 [1]
(3S)-3-[[2-(2-Fluorophenyl)-3-oxo-1H-pyrazole-5-carbonyl]amino]-3-(3-methylphenyl)propanoic acidIC50252.0 [1]
(3S)-3-[[2-(2-Fluorophenyl)-3-oxo-1H-pyrazole-5-carbonyl]amino]-3-(4-methylphenyl)propanoic acidIC50274.0 [1]
(3S)-3-[[2-(2-Fluorophenyl)-3-oxo-1H-pyrazole-5-carbonyl]amino]-3-(2-methoxyphenyl)propanoic acidIC50357.0 [1]
3-[[2-(2,5-Dimethylphenyl)-3-oxo-1H-pyrazole-5-carbonyl]amino]-3-(4-phenylphenyl)propanoic acidIC50803.0 [1]
(3S)-3-(2,4-Dichlorophenyl)-3-[[5-(3,3-dimethyl-2-oxobutoxy)-1-(2-fluorophenyl)pyrazole-3-carbonyl]amino]propanoic acidIC5060.0 [1]
(3S)-3-[(4-Methoxy-1-phenylpyrazole-3-carbonyl)amino]-3-(2-methylphenyl)propanoic acidIC50100.0 [1]
3-[[2-(2-Fluorophenyl)-3-oxo-1H-pyrazole-5-carbonyl]amino]-3-[4-(4-fluorophenyl)phenyl]propanoic acidIC5025.0 [1]
(3S)-3-[[2-(2-Chlorophenyl)-3-oxo-1H-pyrazole-5-carbonyl]amino]-3-(2-methylphenyl)propanoic acidIC5057.0 [1]
(2S)-2-Acetamido-N-[(1R)-3-methyl-1-[(1S,2S,6R,8S)-2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl]butyl]-N'-[4-phenylmethoxy-3-(phenylmethoxymethyl)butyl]butanediamideIC5030000.0 [1]
(2S)-2-Acetamido-N-[(1R)-3-methyl-1-[(1S,2S,6R,8S)-2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl]butyl]-N'-(4-phenylmethoxybutyl)butanediamideIC5030000.0 [1]
(3S)-3-(2-Methylphenyl)-3-[(2-piperidin-1-yl-1,2-dihydropyridine-6-carbonyl)amino]propanoic acidIC508930.0 [1]
(3S)-3-[(2-Methoxy-6-pyridin-4-ylpyridine-4-carbonyl)amino]-3-(2-methylphenyl)propanoic acidIC5030000.0 [1]
(3S)-3-[(5-Methoxy-6-pyridin-4-ylpyridine-2-carbonyl)amino]-3-(4-methylphenyl)propanoic acidIC509660.0 [1]
(3S)-3-[(5-Methoxy-6-pyridin-3-ylpyridine-2-carbonyl)amino]-3-(4-methylphenyl)propanoic acidIC5010000.0 [1]
(3S)-3-[[6-(6-Fluoropyridin-3-yl)-5-methoxypyridine-2-carbonyl]amino]-3-(4-methylphenyl)propanoic acidIC507630.0 [1]
(3S)-3-[[6-(6-Fluoro-2-methoxypyridin-3-yl)-5-methoxypyridine-2-carbonyl]amino]-3-(4-methylphenyl)propanoic acidIC50609.0 [1]
(3S)-3-(2-Chlorophenyl)-3-[(5-methoxy-6-pyridin-3-ylpyridine-2-carbonyl)amino]propanoic acidIC507540.0 [1]
(3S)-3-(2-Fluorophenyl)-3-[(5-methoxy-6-pyridin-4-ylpyridine-2-carbonyl)amino]propanoic acidIC5010000.0 [1]
(3S)-3-(2-Fluorophenyl)-3-[[5-(5-methoxypyridin-2-yl)pyridine-2-carbonyl]amino]propanoic acidIC5010000.0 [1]
(3S)-3-(2-Fluorophenyl)-3-[[6-(6-fluoropyridin-3-yl)-5-methoxypyridine-2-carbonyl]amino]propanoic acidIC5010000.0 [1]
(3S)-3-[[6-(2-Chloro-5-methylpyridin-3-yl)-5-methoxypyridine-2-carbonyl]amino]-3-(2-fluorophenyl)propanoic acidIC5010000.0 [1]
(3S)-3-(2-Fluorophenyl)-3-[[5-methoxy-6-(2-morpholin-4-ylpyridin-4-yl)pyridine-2-carbonyl]amino]propanoic acidIC5010000.0 [1]
(3S)-3-[(5-Methoxy-6-pyridin-4-ylpyridine-2-carbonyl)amino]-3-(2-methylphenyl)propanoic acidIC505450.0 [1]
(3S)-3-[[6-(6-Fluoropyridin-3-yl)-5-methoxypyridine-2-carbonyl]amino]-3-(2-methylphenyl)propanoic acidIC501600.0 [1]
(3S)-3-[[5-Methoxy-6-(2-morpholin-4-ylpyridin-4-yl)pyridine-2-carbonyl]amino]-3-(2-methylphenyl)propanoic acidIC5010000.0 [1]
(3S)-3-(2-Chlorophenyl)-3-[[5-(3-chlorophenyl)-6-methoxypyridine-3-carbonyl]amino]propanoic acidIC5010300.0 [1]
(3S)-3-(2-Chlorophenyl)-3-[(5-methoxy-6-pyridin-4-ylpyridine-2-carbonyl)amino]propanoic acidIC508040.0 [1]
(3S)-3-(2-Chlorophenyl)-3-[[6-(6-fluoropyridin-3-yl)-5-methoxypyridine-2-carbonyl]amino]propanoic acidIC506490.0 [1]
(3S)-3-[[6-(2-Chloro-5-methylpyridin-3-yl)-5-methoxypyridine-2-carbonyl]amino]-3-(2-methylphenyl)propanoic acidIC505630.0 [1]
(3S)-3-[[6-(5-Fluoro-2-methylpyridin-4-yl)-5-methoxypyridine-2-carbonyl]amino]-3-(2-methylphenyl)propanoic acidIC50118.2 [1]
(3S)-3-[[6-(2-Chloro-5-methylpyridin-3-yl)-5-methoxypyridine-2-carbonyl]amino]-3-(2-chlorophenyl)propanoic acidIC508770.0 [1]
(3S)-3-(2-Chlorophenyl)-3-[[5-methoxy-6-(2-methyl-6-morpholin-4-ylpyridin-4-yl)pyridine-2-carbonyl]amino]propanoic acidIC509080.0 [1]
(3S)-3-(2-Methylphenyl)-3-[(2-piperidin-1-yl-2,3-dihydropyridine-4-carbonyl)amino]propanoic acidIC5010000.0 [1]
(3S)-3-[3-(2-Methoxy-5-propan-2-ylphenyl)phenyl]-3-(5-methyl-1,3,4-oxadiazol-2-yl)propanoic acidIC506259.0 [1]
3-[3-(2-Methoxy-5-propan-2-ylphenyl)phenyl]-3-(5-methyl-1,3,4-oxadiazol-2-yl)propanoic acidIC5049.0 [1]
3-[3-(5-Tert-butyl-2-methoxyphenyl)phenyl]-3-(1,3-thiazol-2-yl)propanoic acidIC50119.0 [1]
3-[5-(5-Chloro-2-methoxyphenyl)pyridin-3-yl]-3-(5-methyl-1,3,4-oxadiazol-2-yl)propanoic acidIC503910.0 [1]
3-[5-(2,6-Dimethoxyphenyl)pyridin-3-yl]-3-(5-methyl-1,3,4-oxadiazol-2-yl)propanoic acidIC50160.0 [1]
3-[5-(5-Fluoro-2-methoxyphenyl)pyridin-3-yl]-3-(5-methyl-1,3,4-oxadiazol-2-yl)propanoic acidIC507070.0 [1]
3-[2-Methoxy-5-(4-methoxyphenyl)phenyl]-3-(5-methyl-1,3-thiazol-2-yl)propanoic acidIC507810.0 [1]
3-[2-Methoxy-5-(2-methylphenyl)phenyl]-3-(5-methyl-1,3-thiazol-2-yl)propanoic acidIC503280.0 [1]
3-[3-(2-Cyanophenyl)phenyl]-3-(5-methyl-1,3,4-oxadiazol-2-yl)propanoic acidIC504740.0 [1]
3-[5-(5-Fluoro-2-methylphenyl)-2-methoxyphenyl]-3-(5-methyl-1,3-thiazol-2-yl)propanoic acidIC501200.0 [1]
3-[3-(2-Fluoro-4-methoxyphenyl)phenyl]-3-(5-methyl-1,3-thiazol-2-yl)propanoic acidIC50989.0 [1]
3-[3-(2-Carbamoylphenyl)phenyl]-3-(5-methyl-1,3-thiazol-2-yl)propanoic acidIC505384.0 [1]
3-[3-(6-Amino-2-fluoropyridin-3-yl)phenyl]-3-(1,3-thiazol-2-yl)propanoic acidIC501390.0 [1]
3-[5-(4-Fluoro-2-methylphenyl)-2-methoxyphenyl]-3-(5-methyl-1,3-thiazol-2-yl)propanoic acidIC503730.0 [1]
3-[3-Chloro-5-(2-fluoro-4-methoxyphenyl)phenyl]-3-(5-methyl-1,3-thiazol-2-yl)propanoic acidIC50563.0 [1]
3-[3-(2-Acetylphenyl)-5-fluorophenyl]-3-(1,3-oxazol-2-yl)propanoic acidIC502030.0 [1]
3-[2-Methoxy-5-[3-(trifluoromethyl)phenyl]phenyl]-3-(5-methyl-1,3-thiazol-2-yl)propanoic acidIC507770.0 [1]
3-[3-(2,5-Difluorophenyl)-5-fluorophenyl]-3-(1,3-oxazol-2-yl)propanoic acidIC501490.0 [1]
3-[5-(4-Chlorophenyl)-2-methoxyphenyl]-3-(5-methyl-1,3-thiazol-2-yl)propanoic acidIC503200.0 [1]
3-[3-(3-Phenylmethoxyphenyl)phenyl]-3-(1,3-thiazol-2-yl)propanoic acidIC502772.0 [1]
3-(2-Methoxy-5-phenylphenyl)-3-(1,3-thiazol-2-yl)propanoic acidIC504942.0 [1]
3-[5-(3-Chloro-2-fluorophenyl)-2-methoxyphenyl]-3-(5-methyl-1,3-thiazol-2-yl)propanoic acidIC50954.0 [1]
3-[3-(3-Fluoro-4-phenylmethoxyphenyl)phenyl]-3-(1,3-thiazol-2-yl)propanoic acidIC502426.0 [1]
3-[5-(5-Chloro-2-fluorophenyl)-2-methoxyphenyl]-3-(5-methyl-1,3-thiazol-2-yl)propanoic acidIC501230.0 [1]
3-[5-(2,3-Dimethylphenyl)-2-methoxyphenyl]-3-(5-methyl-1,3-thiazol-2-yl)propanoic acidIC502300.0 [1]
3-[3-(2-Fluoropyridin-4-yl)phenyl]-3-(1,3-thiazol-2-yl)propanoic acidIC5023600.0 [1]
3-[3-[3-(Cyanomethoxy)phenyl]phenyl]-3-(1,3-thiazol-2-yl)propanoic acidIC501940.0 [1]
3-[3-(2-Formyl-5-methoxyphenyl)phenyl]-3-(1,3-thiazol-2-yl)propanoic acidIC503202.0 [1]
3-[2-Methoxy-5-[2-(trifluoromethyl)phenyl]phenyl]-3-(5-methyl-1,3-thiazol-2-yl)propanoic acidIC5010200.0 [1]
3-[3-(2-Acetylphenyl)phenyl]-3-(5-methyl-1,3,4-oxadiazol-2-yl)propanoic acidIC501720.0 [1]
3-[5-(3-Chloro-2-methylphenyl)-2-methoxyphenyl]-3-(5-methyl-1,3-thiazol-2-yl)propanoic acidIC501310.0 [1]
3-[3-(2,5-Dimethylpyrazol-3-yl)phenyl]-3-(1,3-thiazol-2-yl)propanoic acidIC509540.0 [1]
3-[3-Fluoro-5-(2-fluoro-3-methylphenyl)phenyl]-3-(1,3-oxazol-2-yl)propanoic acidIC50488.0 [1]
3-[3-Chloro-5-(2-fluorophenyl)phenyl]-3-(5-methyl-1,3-thiazol-2-yl)propanoic acidIC50328.0 [1]
3-(3-Fluoro-5-pyridin-4-ylphenyl)-3-(5-methyl-1,3-thiazol-2-yl)propanoic acidIC508650.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Lysosomal protective protein Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 10 May. 2024, https://www.aatbio.com/data-sets/lysosomal-protective-protein-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 10). Quest Database™ Lysosomal protective protein Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/lysosomal-protective-protein-inhibitors-ic50-ki.
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