Structure | Compound Name | Standard Type | Standard Values (in nM) |
|---|---|---|---|
| Tomivosertib | IC50 | 6.0 [1] | |
| (4-Methylpiperazin-1-yl)-[4-[3-[4-(trifluoromethyl)phenyl]imidazo[1,2-a]pyrazin-6-yl]phenyl]methanone | IC50 | 1990.0 [1] | |
| [4-[3-(4-Chlorophenyl)imidazo[1,2-a]pyrazin-6-yl]phenyl]-(4-methylpiperazin-1-yl)methanone | IC50 | 759.0 [1] | |
| CID 118598634 | IC50 | 73.0 [1] | |
| N-[6-[(8-Chloro-1,5-dioxospiro[2H-imidazo[1,5-a]pyridine-3,1'-cyclohexane]-6-yl)amino]pyrimidin-4-yl]cyclopropanecarboxamide | IC50 | 0.31 [1] | |
MLA | "Quest Database™ MAP kinase-interacting serine/threonine-protein kinase 1/2 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 15 Dec. 2025, https://www.aatbio.com/data-sets/map-kinase-interacting-serine-threonine-protein-kinase-1-2-inhibitors-ic50-ki. | |
APA | AAT Bioquest, Inc. (2025, December 15). Quest Database™ MAP kinase-interacting serine/threonine-protein kinase 1/2 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/map-kinase-interacting-serine-threonine-protein-kinase-1-2-inhibitors-ic50-ki. | |
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